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Protozoal Drugs in Development


OrganismDrug ClassCompanyDrug NameAlt NameDrug StatusNotesAIDS#
Plasmodium sppAntimalarial AminoquinolineSanofiFerroquineSR-97193Phase IITerminated
Plasmodium sppAntimalarial EndoperoxidesGlaxoSmithKlineTafenoquine; EtaquineWR 238605; SB-252263Phase II/IIIRecruiting 006901
Plasmodium sppAntimalarial SpiroindoloneNovartisKAE-609NITD-609Phase IIRecruiting
Plasmodium sppAntimalarial TrioxolaneMedicines for Malaria VentureOZ-439MMV-08/1019Phase IINot Yet Recruiting
Plasmodium sppCombinationPoliclinique Medicale UniversitaireCotrifazidRifampicin and Cotrimoxazole and Isoniazid Phase IITerminated
Plasmodium sppCombinationPfizerAzithromycin and ChloroquineAZCQ; Zithromax and Chloroquine; Zmax and ChloroquinePhase IIIRecruiting
Plasmodium sppCombinationHolley Pharm; Holleykin PharmEurartesim; Artekin™; Duocotecxin™Dihydroartemisinin and PiperaquinePhase IIICompleted
Plasmodium sppCombinationJomaa PharmaFosclin; JP-01Clindamycin and FosmidomycinPhase IIICompleted
Plasmodium sppDNA Synthesis InhibitorPfizer; Mission PharmacalTindamax™; Fasigyn™; Simplotan™TinidazolePhase IIUnknown 007940
Plasmodium sppElectron Transport Chain InhibitorGlaxoSmithKlineGSK932121 Phase ITerminated (Toxicity)
Plasmodium sppHemozoin InhibitorTulane University Health CenterAQ-13AminoquinolinePhase IINot Yet Recruiting
Plasmodium sppInhibition of Phospholipid Metabolism Sanofi-AventisSAR97276A1,12-Bis[5-(2-hydroxyethyl)-4-methyl-1,3-thiazol-3-ium]dodecane dibromidePhase IITerminated
Toxoplasma gondiiProtein Synthesis Inhibitor (binds to 50S subunit)Rhone-Poulenc PharmaceuticalsRovamycine™SpiramycinPhase IIIRecruiting 007350

Last Updated: January 2013