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ONLINE DATABASE SEARCH - HIV-LS-295-MEMO

1. 43307 HIV-LS-295; PUBMED-HIV-5/3/2004

Rational Design and Synthesis of Novel Dimeric Diketoacid-Containing Inhibitors of HIV-1 Integrase: Implication for Binding to Two Metal Ions on the Active Site of Integrase

Long, YQ, Jiang, XH, Dayam, R, Sanchez, T, Shoemaker, R, Sei, S, and Neamati, N

J Med Chem 2004. 47(10): 2561-2573

HYPERLINK:  http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15115398&dopt=abstract


2. 43308 HIV-LS-295; SCIFINDER-HIV-4/27/2004

The Reverse Transcriptase (RT) Mutation V118I is Associated with Virologic Failure on Abacavir-based Antiretroviral Treatment (ART) in HIV-1 Infection

Saeberg, Paer, Koppel, Kristina, Bratt, Goeran, Fredriksson, Eva Lena, Hejdeman, Bo, Sitbon, Gisela, and Sandstroem, Eric

Scandinavian Journal of Infectious Diseases 2004. 36(1): 40-45

 

3. 43309 HIV-LS-295; PUBMED-HIV-5/3/2004

An unusual "senseless" 2',5'-oligoribonucleotide with potent anti-HIV activity

Aboul-Fadl, T, Agrawal, VK, Buckheit, RW Jr, and Broom, AD

Nucleosides Nucleotides Nucleic Acids 2004. 23(3): 545-54

HYPERLINK:  http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15113022&dopt=abstract


4. 43310 HIV-LS-295; PUBMED-HIV-5/3/2004

Design, synthesis and evaluation of potential inhibitors of HIV gp120-CD4 interactions

Boussard, C, Klimkait, T, Mahmood, N, Pritchard, M, and Gilbert, IH

Bioorg Med Chem Lett 2004. 14(10): 2673-6

HYPERLINK:  http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15109676&dopt=abstract


5. 43311 HIV-LS-295; PUBMED-HIV-5/3/2004

Bis-Anthracycline Antibiotics Inhibit Human Immunodeficiency Virus Type 1 Transcription

Kutsch, O, Levy, DN, Bates, PJ, Decker, J, Kosloff, BR, Shaw, GM, Priebe, W, and Benveniste, EN

Antimicrob Agents Chemother 2004. 48(5): 1652-1663

HYPERLINK:  http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15105117&dopt=abstract


6. 43312 HIV-LS-295; PUBMED-HIV-5/3/2004

Novel 4'-Substituted Stavudine Analog with Improved Anti-Human Immunodeficiency Virus Activity and Decreased Cytotoxicity

Dutschman, GE, Grill, SP, Gullen, EA, Haraguchi, K, Takeda, S, Tanaka, H, Baba, M, and Cheng, YC

Antimicrob Agents Chemother 2004. 48(5): 1640-1646

HYPERLINK:  http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15105115&dopt=abstract


7. 43313 HIV-LS-295; PUBMED-HIV-5/3/2004

Effects of Drug Resistance Mutations L100I and V106A on the Binding of Pyrrolobenzoxazepinone Nonnucleoside Inhibitors to the Human Immunodeficiency Virus Type 1 Reverse Transcriptase Catalytic Complex

Locatelli, GA, Campiani, G, Cancio, R, Morelli, E, Ramunno, A, Gemma, S, Hubscher, U, Spadari, S, and Maga, G

Antimicrob Agents Chemother 2004. 48(5): 1570-1580

HYPERLINK:  http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15105107&dopt=abstract


8. 43314 HIV-LS-295; SCIFINDER-HIV-4/27/2004

Synergistic attachment inhibitor-fusion inhibitor compositions for the prevention and treatment of acquired immunodeficiency syndrome((Tanox, Inc. USA)

Fung, Sek Chung

PATENT: WO 2004028473 A2; ISSUE DATE: 20040408

APPLICATION: 2003; PP: 22 pp.

 

9. 43315 HIV-LS-295; SCIFINDER-HIV-4/27/2004

Treatment of viral diseases by 1,3,5-triazine nucleoside and nucleotide analogs, and preparation thereof ((Koronis Pharmaceuticals, Incorporated USA)

Daifuku, Richard, Gall, Alexander, and Sergueev, Dmitri

PATENT: WO 2004028454 A2; ISSUE DATE: 20040408

APPLICATION: 2003; PP: 108 pp.

 

10. 43316 HIV-LS-295; PUBMED-HIV-5/3/2004

Tipranavir: the first nonpeptidic protease inhibitor

Cheonis, N

BETA 2004. 16(2): 15-7

HYPERLINK:  http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15104065&dopt=abstract


11. 43317 HIV-LS-295; SCIFINDER-HIV-4/27/2004

Preparation and pharmaceutical compositions of indole, azaindole and related heterocyclic 4-alkenyl piperidine amides ((USA))

Wang, Tao, Kadow, John F, Meanwell, Nicholas A, Yeung, Kap-Sun, Zhang, Zhongxing, Yin, Zhiwei, Qiu, Zhilei, Deon, Daniel H, James, Clint A, Ruediger, Edward H, and Bachand, Carol

PATENT: US 20040063744 A1; ISSUE DATE: 20040401

APPLICATION: 2003-32154; PP: 181 pp.

 

12. 43318 HIV-LS-295; PUBMED-HIV-5/3/2004

A 14-Day Dose-Response Study of the Efficacy, Safety, and Pharmacokinetics of the Nonpeptidic Protease Inhibitor Tipranavir in Treatment-Naive HIV-1-Infected Patients

McCallister, S, Valdez, H, Curry, K, MacGregor, T, Borin, M, Freimuth, W, Wang, Y, and Mayers, DL

J Acquir Immune Defic Syndr 2004. 35(4): 376-382

HYPERLINK:  http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15097154&dopt=abstract


13. 43319 HIV-LS-295; SCIFINDER-HIV-4/27/2004

Cellular protein Inip76, its presence in HIV-1 integrase protein complex, role in retroviral integration, and use as drug target((K U Leuven Research & Development, Belg.)

Cherepanov, Peter, Debyser, Zeger, and De Clercq, Erik

PATENT: GB 2393440 A1; ISSUE DATE: 20040331

APPLICATION: 2002-22361; PP: 50 pp.

 

14. 43320 HIV-LS-295; PUBMED-HIV-5/3/2004

Pharmacokinetic Evaluation and Short-Term Activity of Stavudine, Nevirapine, and Nelfinavir Therapy in HIV-1-Infected Adults

Skowron, G, Leoung, G, Hall, DB, Robinson, P, Lewis, R, Grosso, R, Jacobs, M, Kerr, B, MacGregor, T, Stevens, M, Fisher, A, Odgen, R, and Yen-Lieberman, B

J Acquir Immune Defic Syndr 2004. 35(4): 351-358

HYPERLINK:  http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15097151&dopt=abstract


15. 43321 HIV-LS-295; SCIFINDER-HIV-4/27/2004

TAT-gp120 interaction-based mechanism for HIV-1 entry into host cells, and peptides inhibiting this mechanism ((Creabilis Therapeutics S.R.L., Italy)

Bussolino, Federico and Marchio, Serena

PATENT: WO 2004024173 A2; ISSUE DATE: 20040325

APPLICATION: 2003; PP: 87 pp.

 

16. 43322 HIV-LS-295; SCIFINDER-HIV-4/27/2004

Mutational profiles in HIV-1 protease correlated with phenotypic drug resistance((Tibotec Pharmaceuticals Ltd., Ire.)

De Meyer, Sandra, Azijn, Hilde, and De Bethune, Marie-pierre TMMG

PATENT: WO 2004003817 A1; ISSUE DATE: 20040108

APPLICATION: 2003; PP: 32 pp.

 

17. 43323 HIV-LS-295; PUBMED-HIV-5/3/2004

Phase II trial of infusional cyclophosphamide, doxorubicin, and etoposide in patients with HIV-associated non-Hodgkin's lymphoma: an Eastern Cooperative Oncology Group Trial (E1494)

Sparano, JA, Lee, S, Chen, MG, Nazeer, T, Einzig, A, Ambinder, RF, Henry, DH, Manalo, J, Li, T, and Von, Roenn JH

J Clin Oncol 2004. 22(8): 1491-500

HYPERLINK:  http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15084622&dopt=abstract


18. 43324 HIV-LS-295; PUBMED-HIV-5/3/2004

Novel halogenated nitrobenzylthioinosine analogs as es nucleoside transporter inhibitors

Gupte, A and Buolamwini, JK

Bioorg Med Chem Lett 2004. 14(9): 2257-60

HYPERLINK:  http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15081020&dopt=abstract


19. 43325 HIV-LS-295; PUBMED-HIV-5/3/2004

Measurement of anti-HIV activity of marketed vaginal products and excipients using a PBMC-based in vitro assay

Rohan, LC, Ratner, D, McCullough, K, Hiller, SL, and Gupta, P

Sex Transm Dis 2004. 31(3): 143-8

HYPERLINK:  http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15076925&dopt=abstract


20. 43326 HIV-LS-295; SCIFINDER-HIV-4/27/2004

The human immunodeficiency virus type 1 ribosomal frameshifting site is an invariant sequence determinant and an important target for antiviral therapy

Biswas, Preetha, Jiang, Xi, Pacchia, Annmarie L, Dougherty, Joseph P, and Peltz, Stuart W

Journal of Virology 2004. 78(4): 2082-2087

 

21. 43327 HIV-LS-295; PUBMED-HIV-5/3/2004

Synthesis and biological evaluation of novel tert-azido or tert-amino substituted penciclovir analogs

Ok, Kim H, Won, Baek H, Ryong, Moon H, Kim, DK, Woo, Chun M, and Shin, Jeong L

Org Biomol Chem 2004. 2(8): 1164-8

HYPERLINK:  http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15064793&dopt=abstract


22. 43328 HIV-LS-295; SCIFINDER-HIV-4/27/2004

Polymer conjugates with HIV gp41-derived peptides and their therapeutic use((Trimeris, Inc. USA)

Bray, Brian, Kang, Myung-Chol, Tvermoes, Nicolai, Kinder, Daniel, and Lackey, John William

PATENT: WO 2004029073 A2; ISSUE DATE: 20040408

APPLICATION: 2003; PP: 79 pp.

 

23. 43329 HIV-LS-295; WOS-HIV-4/25/2004

Synthesis and anti HIV-1 activity of 2-[[2-(3,5-dimethylphenoxy)ethyl]thio]pyrimidin4(3 H)-ones

Novikov, MS, Ozerov, AA, Sim, OG, and Buckheit, RW

KHIM GETEROTSIKL+ 2004(1): 42-47

HYPERLINK:  http://publishorperish.nih.gov/isicgi/gateway/Gateway.cgi?KeyUT=000220011500005


24. 43330 HIV-LS-295; WOS-HIV-4/25/2004

Design, synthesis and preliminary evaluation of peptidomimetic inhibitors of HIV aspartic protease with an epoxyalcohol core

Benedetti, F, Berti, F, Miertus, S, Romeo, D, Schillani, F, and Tossi, A

ARKIVOC 2003: 140-154

HYPERLINK:  http://publishorperish.nih.gov/isicgi/gateway/Gateway.cgi?KeyUT=000220561500013


25. 43331 HIV-LS-295; WOS-HIV-4/25/2004

Synthesis of the 5 '-phosphonate of 4(S)-(6-amino-9H-purin-9-yl)tetrahy ro-2(S)-furanmethanol [S,S-IsoddA]

Nair, V and Sharma, PK

ARKIVOC 2003: 10-14

HYPERLINK:  http://publishorperish.nih.gov/isicgi/gateway/Gateway.cgi?KeyUT=000220561700002


26. 43332 HIV-LS-295; WOS-HIV-5/2/2004

Pharmacokinetic characteristics of ritonavir, zidovudine, lamivudine, and stavudine in children with human immunodeficiency virus infection

Fletcher, CV, Yogev, R, Nachman, SA, Wiznia, A, Pelton, S, McIntosh, K, and Stanley, K

PHARMACOTHERAPY 2004. 24(4): 453-459

HYPERLINK:  http://publishorperish.nih.gov/isicgi/gateway/Gateway.cgi?KeyUT=000220624600004


27. 43333 HIV-LS-295; WOS-HIV-5/2/2004

Orally bioavailable competitive CCR5 antagonists

Thoma, G, Nuninger, F, Schaefer, M, Akyel, KG, Albert, R, Beerli, C, Bruns, C, Francotte, E, Luyten, M, MacKenzie, D, Oberer, L, Streiff, MB, Wagner, T, Walter, H, Weckbecker, G, and Zerwes, HG

J MED CHEM 2004. 47(8): 1939-1955

HYPERLINK:  http://publishorperish.nih.gov/isicgi/gateway/Gateway.cgi?KeyUT=000220642100010


28. 43334 HIV-LS-295; WOS-HIV-5/2/2004

Selective inhibition of HIV-1 reverse transcriptase (HIV-1 RT) RNase H by small RNA hairpins and dumbbells

Hannoush, RN, Carriero, S, Min, KL, and Damha, MJ

CHEMBIOCHEM 2004. 5(4): 527-533

HYPERLINK:  http://publishorperish.nih.gov/isicgi/gateway/Gateway.cgi?KeyUT=000220773500016


29. 43335 HIV-LS-295; WOS-HIV-5/2/2004

On the role of interferon regulatory factors in HIV-1 replication

Marsili, G, Borsetti, A, Sgarbanti, M, Remoli, AL, Ridolfi, B, Stellacci, E, Ensoli, B, and Battistini, A

ANN NY ACAD SCI 2003. 1010: 29-42

HYPERLINK:  http://publishorperish.nih.gov/isicgi/gateway/Gateway.cgi?KeyUT=000189446300005


30. 43336 HIV-LS-295; WOS-HIV-5/2/2004

Six-year follow-up of HIV-1-infected adults in a clinical trial of antiretroviral therapy with indinavir, zidovudine, and lamivudine

Gulick, RM, Meibohm, A, Havlir, D, Eron, JJ, Mosley, A, Chodakewitz, JA, Isaacs, R, Gonzalez, C, McMahon, D, Richman, DD, Robertson, M, and Mellors, JW

AIDS 2003. 17(16): 2345-2349

HYPERLINK:  http://publishorperish.nih.gov/isicgi/gateway/Gateway.cgi?KeyUT=000220672200009


31. 43337 HIV-LS-295; WOS-HIV-5/2/2004

Resistance of HIV-1 to multiple antiretroviral drugs in France: a 6-year survey (1997-2002) based on an analysis of over 7000 genotypes

Tamalet, C, Fantini, J, Tourres, C, and Yahi, N

AIDS 2003. 17(16): 2383-2388

HYPERLINK:  http://publishorperish.nih.gov/isicgi/gateway/Gateway.cgi?KeyUT=000220672200014


32. 43338 HIV-LS-295; WOS-HIV-5/2/2004

An open-label assessment of TMC 125-a new, next-generation NNRTI, for 7 days in HIV-1 infected individuals with NNRT1 resistance

Gazzard, BG, Pozniak, AL, Rosenbaum, W, Yeni, GP, Staszewski, S, Arasteh, K, De, Dier K, Peeters, M, Woodfall, B, Stebbing, J, and Vant', Klooster GAE

AIDS 2003. 17(18): F49-F54

HYPERLINK:  http://publishorperish.nih.gov/isicgi/gateway/Gateway.cgi?KeyUT=000220672800001


33. 43339 HIV-LS-295; WOS-HIV-5/2/2004

HIV biological variability unveiled: frequent isolations and chimeric receptors reveal unprecedented variation of coreceptor use

Karlsson, I, Antonsson, L, Shi, Y, Karlsson, A, Albert, J, Leitner, T, Olde, B, Owman, C, and Fenyo, EM

AIDS 2003. 17(18): 2561-2569

HYPERLINK:  http://publishorperish.nih.gov/isicgi/gateway/Gateway.cgi?KeyUT=000220672800003


34. 43340 HIV-LS-295; WOS-HIV-5/2/2004

Molecular mapping of epitopes for interaction of HIV-1 as well as natural ligands with the chemokine receptors, CCR5 and CXCR4

Antonsson, L, Boketoft, A, Garzino-Demo, A, Olde, B, and Owman, C

AIDS 2003. 17(18): 2571-2579

HYPERLINK:  http://publishorperish.nih.gov/isicgi/gateway/Gateway.cgi?KeyUT=000220672800004


35. 43341 HIV-LS-295; WOS-HIV-5/2/2004

Clinical and immunological impact of HIV envelope V3 sequence variation after starting initial triple antiretroviral therapy

Brumme, ZL, Dong, WWY, Yip, B, Wynhoven, B, Hoffman, NG, Swanstrom, R, Jensen, MA, Mullins, JI, Hogg, RS, Montaner, JSG, and Harrigan, PR

AIDS 2004. 18(4): F1-F9

HYPERLINK:  http://publishorperish.nih.gov/isicgi/gateway/Gateway.cgi?KeyUT=000220647400001


36. 43342 HIV-LS-295; WOS-HIV-5/2/2004

Evaluation of nevirapine and/or hydroxyurea with nucleoside reverse transcriptase inhibitors in treatment-naive HIV-1-infected subjects

Blanckenberg, DH, Wood, R, Horban, A, Beniowski, M, Boron-Kaczmarska, A, Trocha, H, Halota, W, Schmidt, RE, Fatkenheuer, G, Jessen, H, and Lange, JMA

AIDS 2004. 18(4): 631-640

HYPERLINK:  http://publishorperish.nih.gov/isicgi/gateway/Gateway.cgi?KeyUT=000220647400007

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