ONLINE DATABASE SEARCH - HIV-LS-303-MEMO
1. 43914 HIV-LS-303; SCIFINDER-HIV-8/17/2004
Synthesis of certain 6-(arylthio)uracils and related derivatives as potential antiviral agents
El-Emam, Ali A, Massoud, Mohamed AM, El-Bendary, Eman R, and El-Sayed, Magda A
Bulletin of the Korean Chemical Society 2004. 25(7): 991-996
2. 43915 HIV-LS-303; PUBMED-HIV-8/24/2004
Resistance to HIV Protease Inhibitors: Mechanisms and Clinical Consequences
De Mendoza, C and Soriano, V
Curr Drug Metab 2004. 5(4): 321-328
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15320704&dopt=abstract
3. 43916 HIV-LS-303; PUBMED-HIV-8/24/2004
Structural Determinants and Molecular Mechanisms for the Resistance of HIV-1 RT to Nucleoside Analogues
Deval, J, Courcambeck, J, Selmi, B, Boretto, J, and Canard, B
Curr Drug Metab 2004. 5(4): 305-16
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15320702&dopt=abstract
4. 43917 HIV-LS-303; PUBMED-HIV-8/24/2004
HIV-1 Reverse Transcriptase Inhibitors: Current Issues and Future Perspectives
Locatelli, GA, Cancio, R, Spadari, S, and Maga, G
Curr Drug Metab 2004. 5(4): 283-90
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15320700&dopt=abstract
5. 43918 HIV-LS-303; SCIFINDER-HIV-8/17/2004
Antiviral Drugs: Third strike against HIV enzymes
Kirkpatrick, Peter
Nature Reviews Drug Discovery 2004. 3(8): 645
6. 43919 HIV-LS-303; PUBMED-HIV-8/24/2004
Statins Inhibit HIV-1 Infection by Down-regulating Rho Activity
Del Real, G, Jimenez-Baranda, S, Mira, E, Lacalle, RA, Lucas, P, Gomez-Mouton, C, Alegret, M, Pena, JM, Rodriguez-Zapata, M, Alvarez-Mon, M, Martinez-A, C, and Manes, S
J Exp Med 2004. 200(4): 541-547
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15314078&dopt=abstract
7. 43920 HIV-LS-303; SCIFINDER-HIV-8/17/2004
Preparation of tetrahydro-4H-pyrido[1,2-a]pyrimidines and related compounds as HIV integrase inhibitors ((Istituto Di Ricerche Di Biologia Molecolare P. Angeletti Spa, Italy)
Crescenzi, Benedetta, Kinzel, Olaf, Muraglia, Ester, Orvieto, Federica, Pescatore, Giovanna, Rowley, Michael, and Summa, Vincenzo
PATENT: WO 2004058756 A1; ISSUE DATE: 20040715
APPLICATION: 2003; PP: 113 pp.
8. 43921 HIV-LS-303; PUBMED-HIV-8/24/2004
Synthesis and application of methyleneoxy pseudodipeptide building blocks in biologically active peptides
Hlavacek, J, Marik, J, Konvalinka, J, Bennettova, B, and Tykva, R
Amino Acids 2004. 27(1): 19-27
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15309568&dopt=abstract
9. 43922 HIV-LS-303; PUBMED-HIV-8/24/2004
Inhibition of HIV-1 fusion with small interfering RNAs targeting the chemokine coreceptor CXCR4
Zhou, N, Fang, J, Mukhtar, M, Acheampong, E, and Pomerantz, RJ
Gene Ther 2004
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15306840&dopt=abstract
10. 43923 HIV-LS-303; SCIFINDER-HIV-8/17/2004
Preparation of pyrrolidine and azetidine compounds as CCR5 antagonists ((Smithkline Beecham Corporation, USA)
Yang, Hanbiao, Kazmierski, Wieslaw Mieczyslaw, and Aquino, Christopher Joseph
PATENT: WO 2004055016 A1; ISSUE DATE: 20040701
APPLICATION: 2003; PP: 130 pp.
11. 43924 HIV-LS-303; SCIFINDER-HIV-8/17/2004
Preparation of indane compounds and analogs as CCR5 antagonists ((Smithkline Beecham Corporation, USA)
Youngman, Michael, Kazmierski, Wieslaw Mieczyslaw, Yang, Hanbiao, and Aquino, Christopher Joseph
PATENT: WO 2004055012 A1; ISSUE DATE: 20040701
APPLICATION: 2003; PP: 129 pp.
12. 43925 HIV-LS-303; PUBMED-HIV-8/24/2004
PHI-443: A Novel Noncontraceptive Broad-Spectrum Anti- Human Immunodeficiency Virus Microbicide
D'Cruz, OJ, Samuel, P, and Uckun, FM
Biol Reprod 2004
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15306558&dopt=abstract
13. 43926 HIV-LS-303; PUBMED-HIV-8/24/2004
Small-Molecule Dimerization Inhibitors of Wild-Type and Mutant HIV Protease: A Focused Library Approach
Shultz, MD, Ham, YW, Lee, SG, Davis, DA, Brown, C, and Chmielewski, J
J Am Chem Soc 2004. 126(32): 9886-7
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15303839&dopt=abstract
14. 43927 HIV-LS-303; PUBMED-HIV-8/24/2004
Inhibition of human immunodeficiency virus type 1 replication by Z-100, an immunomodulator extracted from human-type tubercle bacilli, in macrophages
Emori, Y, Ikeda, T, Ohashi, T, Masuda, T, Kurimoto, T, Takei, M, and Kannagi, M
J Gen Virol 2004. 85(Pt 9): 2603-13
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15302954&dopt=abstract
15. 43928 HIV-LS-303; PUBMED-HIV-8/24/2004
l-Chicoric acid inhibits human immunodeficiency virus type 1 integration in vivo and is a noncompetitive but reversible inhibitor of HIV-1 integrase in vitro
Reinke, RA, Lee, DJ, McDougall, BR, King, PJ, Victoria, J, Mao, Y, Lei, X, Reinecke, MG, and Robinson, WE Jr
Virology 2004. 326(2): 203-19
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15302207&dopt=abstract
16. 43929 HIV-LS-303; PUBMED-HIV-8/24/2004
2-(2,6-Dihalophenyl)-3-(pyrimidin-2-yl)-1,3-thiazolidin-4-ones as non-nucleoside HIV-1 reverse transcriptase inhibitors
Rao, A, Balzarini, J, Carbone, A, Chimirri, A, De, Clercq E, Monforte, AM, Monforte, P, Pannecouque, C, and Zappala, M
Antiviral Res 2004. 63(2): 79-84
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15302136&dopt=abstract
17. 43930 HIV-LS-303; PUBMED-HIV-8/24/2004
Protecting from R5-tropic HIV: individual and combined effectiveness of a hammerhead ribozyme and a single-chain Fv antibody that targets CCR5
Cordelier, P, Kulkowsky, JW, Ko, C, Matskevitch, AA, McKee, HJ, Rossi, JJ, Bouhamdan, M, Pomerantz, RJ, Kari, G, and Strayer, DS
Gene Ther 2004
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15295615&dopt=abstract
18. 43931 HIV-LS-303; SCIFINDER-HIV-8/17/2004
Preparation of 5,11-dihydro-8-(2-hydroxyethyl)-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepin-6-one derivatives as non-nucleoside reverse transcriptase inhibitors ((Boehringer Ingelheim (Canada) Ltd., Can.)
Yoakim, Christiane, Malenfant, Eric, Thavonekham, Bounkham, Ogilvie, William, and Deziel, Robert
PATENT: US 2004106791 A1; ISSUE DATE: 20040603
APPLICATION: 2003-7496; PP: 27 pp.
19. 43932 HIV-LS-303; PUBMED-HIV-8/24/2004
Lamellarins, from A to Z: a family of anticancer marine pyrrole alkaloids
Bailly, C
Curr Med Chem Anti-Canc Agents 2004. 4(4): 363-78
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15281908&dopt=abstract
20. 43933 HIV-LS-303; SCIFINDER-HIV-8/17/2004
Quinolones with anti-HIV activity, and preparation thereof ((IRM LLC, Bermuda)
He, Yun, Ellis, David Archer, Anaclerio, Beth Marie, Kuhen, Kelli L, Wu, Baogen, and Jiang, Tao
PATENT: WO 2004037853 A2; ISSUE DATE: 20040506
APPLICATION: 2003; PP: 71 pp.
21. 43934 HIV-LS-303; SCIFINDER-HIV-8/17/2004
Structures of HIV-1 RT-DNA complexes before and after incorporation of the anti-AIDS drug tenofovir
Tuske, Steve, Sarafianos, Stefan G, Clark, Arthur D, Ding, Jianping, Naeger, Lisa K, White, Kirsten L, Miller, Michael D, Gibbs, Craig S, Boyer, Paul L, Clark, Patrick, Wang, Gang, Gaffney, Barbara L, Jones, Roger A, Jerina, Donald M, Hughes, Stephen H, and Arnold, Eddy
Nature Structural & Molecular Biology 2004. 11(5): 469-474
22. 43935 HIV-LS-303; SCIFINDER-HIV-8/17/2004
Use of soluble monovalent oligosaccharides as inhibitors of HIV-1 fusion and replication((USA))
Leach, James L, Garber, Stacey Ann, Prieto, Pedro A, Alarcon, Balbino, Rueda, Ricardo, and Vazquez, Enrique
PATENT: US 2004077590 A1; ISSUE DATE: 20040422
APPLICATION: 2002-15115; PP: 13 pp.
23. 43936 HIV-LS-303; PUBMED-HIV-8/24/2004
Drug Targeting of HIV-1 RNA.DNA Hybrid Structures: Thermodynamics of Recognition and Impact on Reverse Transcriptase-Mediated Ribonuclease H Activity and Viral Replication
Li, TK, Barbieri, CM, Lin, HC, Rabson, AB, Yang, G, Fan, Y, Gaffney, BL, Jones, RA, and Pilch, DS
Biochemistry 2004. 43(30): 9732-9742
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15274628&dopt=abstract
24. 43937 HIV-LS-303; SCIFINDER-HIV-8/17/2004
Short-term safety and antiretroviral activity of T-1249, a second-generation fusion inhibitor of HIV
Eron, Joseph J, Gulick, Roy M, Bartlett, John A, Merigan, Thomas, Arduino, Roberto, Kilby, JMichael, Yangco, Bienvenido, Diers, Adriann, Drobnes, Claude, DeMasi, Ralph, Greenberg, Michael, Melby, Thomas, Raskino, Claire, Rusnak, Pam, Zhang, Ying, Spence, Rebecca, and Miralles, GDiego
Journal of Infectious Diseases 2004. 189(6): 1075-1083
25. 43938 HIV-LS-303; SCIFINDER-HIV-8/17/2004
Antiviral random sequence oligonucleotides lacking complementarity to target genomes and their therapeutic uses ((Replicor, Inc. Can.)
Vaillant, Andrew and Juteau, Jean-Marc
PATENT: WO 2004024919 A1; ISSUE DATE: 20040325
APPLICATION: 2003; PP: 161 pp.
26. 43939 HIV-LS-303; WOS-HIV-8/15/2004
The HIV protease inhibitor ritonavir blocks osteoclastogenesis and function by impairing RANKL-induced signaling
Wang, MWH, Wei, S, Faccio, R, Takeshita, S, Tebas, P, Powderly, WG, Teitelbaum, SL, and Ross, FP
J CLIN INVEST 2004. 114(2): 206-213
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000222667600011
27. 43940 HIV-LS-303; WOS-HIV-8/15/2004
Exploring binding mode for styrylquinoline HIV-1 integrase inhibitors using comparative molecular field analysis and docking studies
Ma, XH, Zhang, XY, Tan, JJ, Chen, WZ, and Wang, CX
ACTA PHARMACOL SIN 2004. 25(7): 950-958
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000222574700016
28. 43941 HIV-LS-303; WOS-HIV-8/23/2004
Improved preparation and structural investigation of 4-aryl-4-oxo-2-hydroxy-2-butenoic acids and methyl esters
Maurin, C, Bailly, F, and Cotelle, P
TETRAHEDRON 2004. 60(31): 6479-6486
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000222863600007
29. 43942 HIV-LS-303; WOS-HIV-8/23/2004
In-water reactivity of nucleosides and nucleotides: one-step preparation and biological evaluation of novel ferrocenyl-derivatives
de Champdore, M, Di Fabio, G, Messere, A, Montesarchio, D, Piccialli, G, Loddo, R, La Colla, M, and La Colla, P
TETRAHEDRON 2004. 60(31): 6555-6563
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000222863600015
30. 43943 HIV-LS-303; WOS-HIV-8/23/2004
Synthesis of peptidomimetics based on iminosugar and beta-D-glucopyranoside scaffolds and inhibiton of HIV-protease
Chery, F, Cronin, L, O'Brien, JL, and Murphy, PV
TETRAHEDRON 2004. 60(31): 6597-6608
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000222863600021
31. 43944 HIV-LS-303; WOS-HIV-8/23/2004
Actinchinin, a novel antifungal protein from the gold kiwi fruit
Xia, LX and Ng, TB
PEPTIDES 2004. 25(7): 1093-1098
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000222855100004
32. 43945 HIV-LS-303; WOS-HIV-8/23/2004
Expression of HIV-1 accessory protein Vif is controlled uniquely to be low and optimal by proteasome degradation
Fujita, M, Akari, H, Sakurai, A, Yoshida, A, Chiba, T, Tanaka, K, Strebel, K, and Adachi, A
MICROBES INFECT 2004. 6(9): 791-798
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000222860200001
33. 43946 HIV-LS-303; WOS-HIV-8/23/2004
Lysine sulfonamides as novel HIV-protease inhibitors: N epsilon-disubstituted ureas
Stranix, BR, Sauve, G, Bouzide, A, Cote, A, Sevigny, G, Yelle, J, and Perron, V
BIOORG MED CHEM LETT 2004. 14(15): 3971-3974
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000222792800025
34. 43947 HIV-LS-303; WOS-HIV-8/23/2004
Rigid backbone moiety of KNI-272, a highly selective HIV protease inhibitor: methanol, acetone and dimethylsulfoxide solvated forms of 3-[3-benzyl-2-hydroxy-9-(isoquinoli -5-yloxy)-6-methyl-sulfanylmethyl-5 8-dioxo-4,7-diazanonanoyl]-N-tert-b tyl-1,3-thiazolidine-4-carboxamide
Doi, M, Kimura, T, Ishida, T, and Kiso, Y
ACTA CRYSTALLOGR B 2004. 60: 433-437
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000222725100009