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ONLINE DATABASE SEARCH - HIV-LS-317-MEMO

1. 44932 HIV-LS-317; SCIFINDER-HIV-3/1/2005

A novel HIV-1 antiviral high throughput screening approach for the discovery of HIV-1 inhibitors

Blair, Wade S, Isaacson, Jason, Li, Xinqiang, Cao, Joan, Peng, Qinghai, Kong, George FZ, and Patick, Amy K

Antiviral Research 2005. 65(2): 107-116


2. 44933 HIV-LS-317; PUBMED-HIV-3/9/2005

Activity profiles of deoxynucleoside kinases and 5'-nucleotidases in cultured adipocytes and myoblastic cells: insights into mitochondrial toxicity of nucleoside analogs

Rylova, SN, Albertioni, F, Flygh, G, and Eriksson, S

Biochem Pharmacol 2005. 69(6): 951-60


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15748706&dopt=abstract


3. 44934 HIV-LS-317; PUBMED-HIV-3/9/2005

Artificial zinc-finger fusions targeting Sp1 binding sites and TAR potently repress transcription and replication of HIV-1

Kim, YS, Kim, JM, Jung, DL, Kang, JE, Lee, S, Kim, JS, Seol, W, Shin, HC, Kwon, HS, Lint, CV, Hernandez, N, and Hur, MW

J Biol Chem 2005.


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15743774&dopt=abstract


4. 44935 HIV-LS-317; PUBMED-HIV-3/9/2005

Synthesis of Phosphonated Carbocyclic 2'-Oxa-3'-aza-nucleosides: Novel Inhibitors of Reverse Transcriptase

Chiacchio, U, Balestrieri, E, Macchi, B, Iannazzo, D, Piperno, A, Rescifina, A, Romeo, R, Saglimbeni, M, Sciortino, MT, Valveri, V, Mastino, A, and Romeo, G

J Med Chem 2005. 48(5): 1389-1394


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15743182&dopt=abstract


5. 44936 HIV-LS-317; SCIFINDER-HIV-3/1/2005

Synthesis and evaluation of CCR5 antagonists containing modified 4-piperidinyl-2-phenyl-1-(phenylsulfonylamino)-butane

Shah, Shrenik K, Chen, Natalie, Guthikonda, Ravindra N, Mills, Sander G, Malkowitz, Lorraine, Springer, Martin S, Gould, Sandra L, DeMartino, Julie A, Carella, Anthony, Carver, Gwen, Holmes, Karen, Schleif, William A, Danzeisen, Renee, Hazuda, Daria, Kessler, Joseph, Lineberger, Janet, Miller, Michael, Emini, Emilio A, and MacCoss, Malcolm

Bioorganic & Medicinal Chemistry Letters 2005. 15(4): 977-982



6. 44937 HIV-LS-317; PUBMED-HIV-3/9/2005

Synergistic anti-viral effect of oxanosine and ddI against human immunodeficiency virus

Nakamura, M, Ogawa, T, Yokono, A, Nakamori, S, Ohno, T, and Umezawa, K

Biomed Pharmacother 2005. 59(1-2): 47-50


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15740935&dopt=abstract


7. 44938 HIV-LS-317; PUBMED-HIV-3/9/2005

Design of novel bioisosteres of beta-diketo acid inhibitors of HIV-1 integrase

Sechi, M, Sannia, L, Carta, F, Palomba, M, Dallocchio, R, Dessi, A, Derudas, M, Zawahir, Z, and Neamati, N

Antivir Chem Chemother 2005. 16(1): 41-61


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15739621&dopt=abstract


8. 44939 HIV-LS-317; PUBMED-HIV-3/9/2005

Inhibition of Phosphorolysis Catalyzed by HIV-1 Reverse Transcriptase Is Responsible for the Synergy Found in Combinations of 3'-Azido-3'-deoxythymidine with Nonnucleoside Inhibitors

Cruchaga, C, Odriozola, L, Andreola, M, Tarrago-Litvak, L, and Martinez-Irujo, JJ

Biochemistry 2005. 44(9): 3535-3546


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15736963&dopt=abstract


9. 44940 HIV-LS-317; SCIFINDER-HIV-3/1/2005

Trimeric envelope protein gp41 helical conformation stabilization by peptide mimetics inhibits membrane fusion-mediated cell entry by HIV-1

Tam, James P, Yu, Qitao, Lu, Yi-An, and Yang, Jin-Long

PATENT: WO 2005007831 ISSUE DATE: 20050127

APPLICATION: 2004 PP: 71 pp.

ASSIGNEE: (Vanderbilt University, USA


10. 44941 HIV-LS-317; PUBMED-HIV-3/9/2005

In Vitro Activity of Structurally Diverse Nucleoside Analogs against Human Immunodeficiency Virus Type 1 with the K65R Mutation in Reverse Transcriptase

Parikh, UM, Koontz, DL, Chu, CK, Schinazi, RF, and Mellors, JW

Antimicrob Agents Chemother 2005. 49(3): 1139-44


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15728915&dopt=abstract



11. 44942 HIV-LS-317; PUBMED-HIV-3/9/2005

Crystal structure of a cross-reaction complex between an anti-HIV-1 protease antibody and an HIV-2 protease peptide

Rezacova, P, Brynda, J, Lescar, J, Fabry, M, Horejsi, M, Sieglova, I, Sedlacek, J, and Bentley, GA

J Struct Biol 2005. 149(3): 332-7


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15721587&dopt=abstract


12. 44943 HIV-LS-317; PUBMED-HIV-3/9/2005

HIV-1-Associated Uracil DNA Glycosylase Activity Controls dUTP Misincorporation in Viral DNA and Is Essential to the HIV-1 Life Cycle

Priet, S, Gros, N, Navarro, JM, Boretto, J, Canard, B, Querat, G, and Sire, J

Mol Cell 2005. 17(4): 479-90


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15721252&dopt=abstract


13. 44944 HIV-LS-317; SCIFINDER-HIV-3/1/2005

Drug resistance mutations in the nucleotide binding pocket of human immunodeficiency virus type 1 reverse transcriptase differentially affect the phosphorolysis-dependent primer unblocking activity in the presence of stavudine and zidovudine and its inhibition by efavirenz

Crespan, Emmanuele, Locatelli, Giada A, Cancio, Reynel, Huebscher, Ulrich, Spadari, Silvio, and Maga, Giovanni

Antimicrobial Agents and Chemotherapy 2005. 49(1): 342-349


14. 44945 HIV-LS-317; SCIFINDER-HIV-3/1/2005

Novel anti-viral agents based upon derivatives of the aromatic heterocycle phenanthridine

Tor, Yitzhak and Luedtke, Nathan

PATENT: WO 2005016343 ISSUE DATE: 20050224

APPLICATION: 2004 PP: 58 pp.

ASSIGNEE: (The Regents of the University of California, USA


15. 44946 HIV-LS-317; PUBMED-HIV-3/9/2005

Isolation of trichogin, an antifungal protein from fresh fruiting bodies of the edible mushroom Tricholoma giganteum

Guo, Y, Wang, H, and Ng, TB

Peptides 2005. 26(4): 575-80


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15752570&dopt=abstract



16. 44947 HIV-LS-317; PUBMED-HIV-3/9/2005

Challenges for the clinical development of new nucleoside reverse transcriptase inhibitors for HIV infection

Wainberg, MA, Sawyer, JP, Montaner, JS, Murphy, RL, Kuritzkes, DR, and Raffi, F

Antivir Ther 2005. 10(1): 13-28


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15751760&dopt=abstract


17. 44948 HIV-LS-317; PUBMED-HIV-3/9/2005

Selective inhibition of HIV-1 reverse transcriptase-associated ribonuclease H activity by hydroxylated tropolones

Budihas, SR, Gorshkova, I, Gaidamakov, S, Wamiru, A, Bona, MK, Parniak, MA, Crouch, RJ, McMahon, JB, Beutler, JA, and Le, Grice SF

Nucleic Acids Res 2005. 33(4): 1249-56


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15741178&dopt=abstract


18. 44949 HIV-LS-317; PUBMED-HIV-3/9/2005

A new pinoresinol-type lignan from Ligularia kanaitizensis

Li, YS, Wang, ZT, Zhang, M, Luo, SD, and Chen, JJ

Nat Prod Res 2005. 19(2): 125-9


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15715255&dopt=abstract


19. 44950 HIV-LS-317; PUBMED-HIV-3/9/2005

Quantitative structure-activity relationship by CoMFA for cyclic urea and nonpeptide-cyclic cyanoguanidine derivatives on wild type and mutant HIV-1 protease

Avram, S, Bologa, C, and Flonta, ML

J Mol Model (Online) 2005.


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15714296&dopt=abstract


20. 44951 HIV-LS-317; WOS-HIV-2/27/2005

The trans-Golgi network-associated human ubiquitin-protein ligase POSH is essential for HIV Woe 1 production

Alroy, I, Tuvia, S, Greener, T, Gordon, D, Barr, HM, Taglicht, D, Mandil-Levin, R, Ben-Avraham, D, Konforty, D, Nir, L, Levius, O, Bicoviski, V, Dori, M, Cohen, S, Yaar, L, Erez, O, Propheta-Meiran, O, Koskas, M, Caspi-Bachar, E, Alchanati, I, Sela-Brown, A, Moskowitz, H, Tessmer, U, Schubert, U, and Reiss, Y

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA 2005. 102(5): 1478-1483, 6


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226877300042



21. 44952 HIV-LS-317; WOS-HIV-2/27/2005

Peptide nucleic acids as epigenetic inhibitors of HIV-1

Sei, S

LETTERS IN PEPTIDE SCIENCE 2003. 10(3-4): 269-286, 18


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226731200010


22. 44953 HIV-LS-317; WOS-HIV-2/27/2005

A synthetic peptide fragment derived from RANTES is a potent inhibitor of HIV-1 infectivity despite a surprising lack of CCR5 receptor affinity

Ramnarine, E, DeVico, AL, and Vigil-Cruz, SC

LETTERS IN PEPTIDE SCIENCE 2003. 10(5-6): 637-643, 7


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226731400033


23. 44954 HIV-LS-317; WOS-HIV-2/27/2005

Potent anti-R5 human immunodeficiency virus type 1 effects of a CCR5 antagonist, AK602/ONO4128/GW873140, in a novel human peripheral blood mononuclear cell nonobese diabetic-SCID, interleukin-2 receptor gamma-chain-knocked-out AIDS mouse model

Nakata, H, Maeda, K, Miyakawa, T, Shibayama, S, Matsuo, M, Takaoka, Y, Ito, M, Koyanagi, Y, and Mitsuya, H

JOURNAL OF VIROLOGY 2005. 79(4): 2087-2096, 10


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226772100012


24. 44955 HIV-LS-317; WOS-HIV-2/27/2005

Kinetics of human immunodeficiency virus type 1 decay following entry into resting CD4(+) T cells

Zhou, Y, Zhang, H, Siliciano, JD, and Siliciano, RF

JOURNAL OF VIROLOGY 2005. 79(4): 2199-2210, 12


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226772100023


25. 44956 HIV-LS-317; WOS-HIV-2/27/2005

Fungal phenalenones inhibit HIV-1 integrase

Shiomi, K, Matsui, R, Isozaki, M, Chiba, H, Sugai, T, Yamaguchi, Y, Masuma, R, Tomoda, H, Chiba, T, Yan, H, Kitamura, Y, Sugiura, W, Omura, S, and Tanaka, H

JOURNAL OF ANTIBIOTICS 2005. 58(1): 65-68, 4


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226818200008


26. 44957 HIV-LS-317; WOS-HIV-2/27/2005

Identification of diverse microbial metabolites as potent inhibitors of HIV-1 tat transactivation

Jayasuriya, H, Zink, DL, Polishook, JD, Bills, GF, Dombrowski, AW, Genilloud, O, Pelaez, FF, Herranz, L, Quamina, D, Lingham, RB, Danzeizen, R, Graham, PL, Tomassini, JE, and Singh, SB

CHEMISTRY & BIODIVERSITY 2005. 2(1): 112-122, 11


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226963500008



27. 44958 HIV-LS-317; WOS-HIV-2/27/2005

Stereoselective synthesis and antiviral activity of novel 4 '(alpha)-hydroxymethyl and 6 '(alpha)-methyl dually branched carbocyclic nucleosides

Kim, JW, Choi, BG, and Hong, JH

BULLETIN OF THE KOREAN CHEMICAL SOCIETY 2004. 25(12): 1812-1816, 5


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226854800011


28. 44959 HIV-LS-317; WOS-HIV-2/27/2005

Enantiomerical excess determination, purification and biological evaluation of (3S) and (3R) alpha,beta-butenolide analogues of isobenzofuranone

Lipka, E, Vaccher, MP, Vaccher, C, and Len, C

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 2005. 15(3): 501-504, 4


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226935700002


29. 44960 HIV-LS-317; WOS-HIV-2/27/2005

Insight into the mechanism of a peptide inhibitor of HIV reverse transcriptase dimerization

Depollier, J, Hourdou, ML, Aldrian-Herrada, G, Rothwell, P, Restle, T, and Divita, G

BIOCHEMISTRY 2005. 44(6): 1909-1918, 10


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226969400016


30. 44961 HIV-LS-317; WOS-HIV-3/6/2005

Novel [2 ',5 '-bis-O-(ter -butyldimethylsilyl)-beta-D-ribofuranosyl]-3 '-spiro-5 ''-(4 ''-amino-1 '',2 ''-oxathiole-2 '',2 ''-dioxide) derivatives with anti-HIV-1 and anti-human-cytomegalovirus activity

de Castro, S, Lobaton, E, Perez-Perez, MJ, San-Felix, A, Cordeiro, A, Andrei, G, Snoeck, R, De Clercq, E, Balzarini, J, Camarasa, MJ, and Velazquez, S

JOURNAL OF MEDICINAL CHEMISTRY 2005. 48(4): 1158-1168, 11


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227115500026


31. 44962 HIV-LS-317; WOS-HIV-3/6/2005

High-throughput screening method of inhibitors that block the interaction between 2 helical regions of HIV-1 gp41

Jin, BS, Lee, WK, Ahn, K, Lee, MK, and Yu, YG

JOURNAL OF BIOMOLECULAR SCREENING 2005. 10(1): 13-19, 7


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227050000002


32. 44963 HIV-LS-317; WOS-HIV-3/6/2005

Defensins: Natural anti-HIV peptides

Chang, TL and Klotman, ME

AIDS REVIEWS 2004. 6(3): 161-168, 8


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227043100005


33. 44964 HIV-LS-317; WOS-HIV-3/6/2005

Mechanism and inhibition of human immunodeficiency virus type 1 reverse transcriptase (HIV-1 RT) by an imidazolidine nucleotide analog

Kerr, SG, Dhareshwar, SS, Froimowitz, M, and Kalman, TI

ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 2004. 228: U174-U175, 2


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000223712800717


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