ONLINE DATABASE SEARCH - HIV-LS-317-MEMO
1. 44932 HIV-LS-317; SCIFINDER-HIV-3/1/2005
A novel HIV-1 antiviral high throughput screening approach for the discovery of HIV-1 inhibitors
Blair, Wade S, Isaacson, Jason, Li, Xinqiang, Cao, Joan, Peng, Qinghai, Kong, George FZ, and Patick, Amy K
Antiviral Research 2005. 65(2): 107-116
2. 44933 HIV-LS-317; PUBMED-HIV-3/9/2005
Activity profiles of deoxynucleoside kinases and 5'-nucleotidases in cultured adipocytes and myoblastic cells: insights into mitochondrial toxicity of nucleoside analogs
Rylova, SN, Albertioni, F, Flygh, G, and Eriksson, S
Biochem Pharmacol 2005. 69(6): 951-60
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15748706&dopt=abstract
3. 44934 HIV-LS-317; PUBMED-HIV-3/9/2005
Artificial zinc-finger fusions targeting Sp1 binding sites and TAR potently repress transcription and replication of HIV-1
Kim, YS, Kim, JM, Jung, DL, Kang, JE, Lee, S, Kim, JS, Seol, W, Shin, HC, Kwon, HS, Lint, CV, Hernandez, N, and Hur, MW
J Biol Chem 2005.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15743774&dopt=abstract
4. 44935 HIV-LS-317; PUBMED-HIV-3/9/2005
Synthesis of Phosphonated Carbocyclic 2'-Oxa-3'-aza-nucleosides: Novel Inhibitors of Reverse Transcriptase
Chiacchio, U, Balestrieri, E, Macchi, B, Iannazzo, D, Piperno, A, Rescifina, A, Romeo, R, Saglimbeni, M, Sciortino, MT, Valveri, V, Mastino, A, and Romeo, G
J Med Chem 2005. 48(5): 1389-1394
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15743182&dopt=abstract
5. 44936 HIV-LS-317; SCIFINDER-HIV-3/1/2005
Synthesis and evaluation of CCR5 antagonists containing modified 4-piperidinyl-2-phenyl-1-(phenylsulfonylamino)-butane
Shah, Shrenik K, Chen, Natalie, Guthikonda, Ravindra N, Mills, Sander G, Malkowitz, Lorraine, Springer, Martin S, Gould, Sandra L, DeMartino, Julie A, Carella, Anthony, Carver, Gwen, Holmes, Karen, Schleif, William A, Danzeisen, Renee, Hazuda, Daria, Kessler, Joseph, Lineberger, Janet, Miller, Michael, Emini, Emilio A, and MacCoss, Malcolm
Bioorganic & Medicinal Chemistry Letters 2005. 15(4): 977-982
6. 44937 HIV-LS-317; PUBMED-HIV-3/9/2005
Synergistic anti-viral effect of oxanosine and ddI against human immunodeficiency virus
Nakamura, M, Ogawa, T, Yokono, A, Nakamori, S, Ohno, T, and Umezawa, K
Biomed Pharmacother 2005. 59(1-2): 47-50
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15740935&dopt=abstract
7. 44938 HIV-LS-317; PUBMED-HIV-3/9/2005
Design of novel bioisosteres of beta-diketo acid inhibitors of HIV-1 integrase
Sechi, M, Sannia, L, Carta, F, Palomba, M, Dallocchio, R, Dessi, A, Derudas, M, Zawahir, Z, and Neamati, N
Antivir Chem Chemother 2005. 16(1): 41-61
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15739621&dopt=abstract
8. 44939 HIV-LS-317; PUBMED-HIV-3/9/2005
Inhibition of Phosphorolysis Catalyzed by HIV-1 Reverse Transcriptase Is Responsible for the Synergy Found in Combinations of 3'-Azido-3'-deoxythymidine with Nonnucleoside Inhibitors
Cruchaga, C, Odriozola, L, Andreola, M, Tarrago-Litvak, L, and Martinez-Irujo, JJ
Biochemistry 2005. 44(9): 3535-3546
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15736963&dopt=abstract
9. 44940 HIV-LS-317; SCIFINDER-HIV-3/1/2005
Trimeric envelope protein gp41 helical conformation stabilization by peptide mimetics inhibits membrane fusion-mediated cell entry by HIV-1
Tam, James P, Yu, Qitao, Lu, Yi-An, and Yang, Jin-Long
PATENT: WO 2005007831 ISSUE DATE: 20050127
APPLICATION: 2004 PP: 71 pp.
ASSIGNEE: (Vanderbilt University, USA
10. 44941 HIV-LS-317; PUBMED-HIV-3/9/2005
In Vitro Activity of Structurally Diverse Nucleoside Analogs against Human Immunodeficiency Virus Type 1 with the K65R Mutation in Reverse Transcriptase
Parikh, UM, Koontz, DL, Chu, CK, Schinazi, RF, and Mellors, JW
Antimicrob Agents Chemother 2005. 49(3): 1139-44
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15728915&dopt=abstract
11. 44942 HIV-LS-317; PUBMED-HIV-3/9/2005
Crystal structure of a cross-reaction complex between an anti-HIV-1 protease antibody and an HIV-2 protease peptide
Rezacova, P, Brynda, J, Lescar, J, Fabry, M, Horejsi, M, Sieglova, I, Sedlacek, J, and Bentley, GA
J Struct Biol 2005. 149(3): 332-7
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15721587&dopt=abstract
12. 44943 HIV-LS-317; PUBMED-HIV-3/9/2005
HIV-1-Associated Uracil DNA Glycosylase Activity Controls dUTP Misincorporation in Viral DNA and Is Essential to the HIV-1 Life Cycle
Priet, S, Gros, N, Navarro, JM, Boretto, J, Canard, B, Querat, G, and Sire, J
Mol Cell 2005. 17(4): 479-90
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15721252&dopt=abstract
13. 44944 HIV-LS-317; SCIFINDER-HIV-3/1/2005
Drug resistance mutations in the nucleotide binding pocket of human immunodeficiency virus type 1 reverse transcriptase differentially affect the phosphorolysis-dependent primer unblocking activity in the presence of stavudine and zidovudine and its inhibition by efavirenz
Crespan, Emmanuele, Locatelli, Giada A, Cancio, Reynel, Huebscher, Ulrich, Spadari, Silvio, and Maga, Giovanni
Antimicrobial Agents and Chemotherapy 2005. 49(1): 342-349
14. 44945 HIV-LS-317; SCIFINDER-HIV-3/1/2005
Novel anti-viral agents based upon derivatives of the aromatic heterocycle phenanthridine
Tor, Yitzhak and Luedtke, Nathan
PATENT: WO 2005016343 ISSUE DATE: 20050224
APPLICATION: 2004 PP: 58 pp.
ASSIGNEE: (The Regents of the University of California, USA
15. 44946 HIV-LS-317; PUBMED-HIV-3/9/2005
Isolation of trichogin, an antifungal protein from fresh fruiting bodies of the edible mushroom Tricholoma giganteum
Guo, Y, Wang, H, and Ng, TB
Peptides 2005. 26(4): 575-80
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15752570&dopt=abstract
16. 44947 HIV-LS-317; PUBMED-HIV-3/9/2005
Challenges for the clinical development of new nucleoside reverse transcriptase inhibitors for HIV infection
Wainberg, MA, Sawyer, JP, Montaner, JS, Murphy, RL, Kuritzkes, DR, and Raffi, F
Antivir Ther 2005. 10(1): 13-28
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15751760&dopt=abstract
17. 44948 HIV-LS-317; PUBMED-HIV-3/9/2005
Selective inhibition of HIV-1 reverse transcriptase-associated ribonuclease H activity by hydroxylated tropolones
Budihas, SR, Gorshkova, I, Gaidamakov, S, Wamiru, A, Bona, MK, Parniak, MA, Crouch, RJ, McMahon, JB, Beutler, JA, and Le, Grice SF
Nucleic Acids Res 2005. 33(4): 1249-56
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15741178&dopt=abstract
18. 44949 HIV-LS-317; PUBMED-HIV-3/9/2005
A new pinoresinol-type lignan from Ligularia kanaitizensis
Li, YS, Wang, ZT, Zhang, M, Luo, SD, and Chen, JJ
Nat Prod Res 2005. 19(2): 125-9
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15715255&dopt=abstract
19. 44950 HIV-LS-317; PUBMED-HIV-3/9/2005
Quantitative structure-activity relationship by CoMFA for cyclic urea and nonpeptide-cyclic cyanoguanidine derivatives on wild type and mutant HIV-1 protease
Avram, S, Bologa, C, and Flonta, ML
J Mol Model (Online) 2005.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15714296&dopt=abstract
20. 44951 HIV-LS-317; WOS-HIV-2/27/2005
The trans-Golgi network-associated human ubiquitin-protein ligase POSH is essential for HIV Woe 1 production
Alroy, I, Tuvia, S, Greener, T, Gordon, D, Barr, HM, Taglicht, D, Mandil-Levin, R, Ben-Avraham, D, Konforty, D, Nir, L, Levius, O, Bicoviski, V, Dori, M, Cohen, S, Yaar, L, Erez, O, Propheta-Meiran, O, Koskas, M, Caspi-Bachar, E, Alchanati, I, Sela-Brown, A, Moskowitz, H, Tessmer, U, Schubert, U, and Reiss, Y
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA 2005. 102(5): 1478-1483, 6
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226877300042
21. 44952 HIV-LS-317; WOS-HIV-2/27/2005
Peptide nucleic acids as epigenetic inhibitors of HIV-1
Sei, S
LETTERS IN PEPTIDE SCIENCE 2003. 10(3-4): 269-286, 18
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226731200010
22. 44953 HIV-LS-317; WOS-HIV-2/27/2005
A synthetic peptide fragment derived from RANTES is a potent inhibitor of HIV-1 infectivity despite a surprising lack of CCR5 receptor affinity
Ramnarine, E, DeVico, AL, and Vigil-Cruz, SC
LETTERS IN PEPTIDE SCIENCE 2003. 10(5-6): 637-643, 7
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226731400033
23. 44954 HIV-LS-317; WOS-HIV-2/27/2005
Potent anti-R5 human immunodeficiency virus type 1 effects of a CCR5 antagonist, AK602/ONO4128/GW873140, in a novel human peripheral blood mononuclear cell nonobese diabetic-SCID, interleukin-2 receptor gamma-chain-knocked-out AIDS mouse model
Nakata, H, Maeda, K, Miyakawa, T, Shibayama, S, Matsuo, M, Takaoka, Y, Ito, M, Koyanagi, Y, and Mitsuya, H
JOURNAL OF VIROLOGY 2005. 79(4): 2087-2096, 10
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226772100012
24. 44955 HIV-LS-317; WOS-HIV-2/27/2005
Kinetics of human immunodeficiency virus type 1 decay following entry into resting CD4(+) T cells
Zhou, Y, Zhang, H, Siliciano, JD, and Siliciano, RF
JOURNAL OF VIROLOGY 2005. 79(4): 2199-2210, 12
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226772100023
25. 44956 HIV-LS-317; WOS-HIV-2/27/2005
Fungal phenalenones inhibit HIV-1 integrase
Shiomi, K, Matsui, R, Isozaki, M, Chiba, H, Sugai, T, Yamaguchi, Y, Masuma, R, Tomoda, H, Chiba, T, Yan, H, Kitamura, Y, Sugiura, W, Omura, S, and Tanaka, H
JOURNAL OF ANTIBIOTICS 2005. 58(1): 65-68, 4
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226818200008
26. 44957 HIV-LS-317; WOS-HIV-2/27/2005
Identification of diverse microbial metabolites as potent inhibitors of HIV-1 tat transactivation
Jayasuriya, H, Zink, DL, Polishook, JD, Bills, GF, Dombrowski, AW, Genilloud, O, Pelaez, FF, Herranz, L, Quamina, D, Lingham, RB, Danzeizen, R, Graham, PL, Tomassini, JE, and Singh, SB
CHEMISTRY & BIODIVERSITY 2005. 2(1): 112-122, 11
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226963500008
27. 44958 HIV-LS-317; WOS-HIV-2/27/2005
Stereoselective synthesis and antiviral activity of novel 4 '(alpha)-hydroxymethyl and 6 '(alpha)-methyl dually branched carbocyclic nucleosides
Kim, JW, Choi, BG, and Hong, JH
BULLETIN OF THE KOREAN CHEMICAL SOCIETY 2004. 25(12): 1812-1816, 5
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226854800011
28. 44959 HIV-LS-317; WOS-HIV-2/27/2005
Enantiomerical excess determination, purification and biological evaluation of (3S) and (3R) alpha,beta-butenolide analogues of isobenzofuranone
Lipka, E, Vaccher, MP, Vaccher, C, and Len, C
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 2005. 15(3): 501-504, 4
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226935700002
29. 44960 HIV-LS-317; WOS-HIV-2/27/2005
Insight into the mechanism of a peptide inhibitor of HIV reverse transcriptase dimerization
Depollier, J, Hourdou, ML, Aldrian-Herrada, G, Rothwell, P, Restle, T, and Divita, G
BIOCHEMISTRY 2005. 44(6): 1909-1918, 10
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000226969400016
30. 44961 HIV-LS-317; WOS-HIV-3/6/2005
Novel [2 ',5 '-bis-O-(ter -butyldimethylsilyl)-beta-D-ribofuranosyl]-3 '-spiro-5 ''-(4 ''-amino-1 '',2 ''-oxathiole-2 '',2 ''-dioxide) derivatives with anti-HIV-1 and anti-human-cytomegalovirus activity
de Castro, S, Lobaton, E, Perez-Perez, MJ, San-Felix, A, Cordeiro, A, Andrei, G, Snoeck, R, De Clercq, E, Balzarini, J, Camarasa, MJ, and Velazquez, S
JOURNAL OF MEDICINAL CHEMISTRY 2005. 48(4): 1158-1168, 11
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227115500026
31. 44962 HIV-LS-317; WOS-HIV-3/6/2005
High-throughput screening method of inhibitors that block the interaction between 2 helical regions of HIV-1 gp41
Jin, BS, Lee, WK, Ahn, K, Lee, MK, and Yu, YG
JOURNAL OF BIOMOLECULAR SCREENING 2005. 10(1): 13-19, 7
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227050000002
32. 44963 HIV-LS-317; WOS-HIV-3/6/2005
Defensins: Natural anti-HIV peptides
Chang, TL and Klotman, ME
AIDS REVIEWS 2004. 6(3): 161-168, 8
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227043100005
33. 44964 HIV-LS-317; WOS-HIV-3/6/2005
Mechanism and inhibition of human immunodeficiency virus type 1 reverse transcriptase (HIV-1 RT) by an imidazolidine nucleotide analog
Kerr, SG, Dhareshwar, SS, Froimowitz, M, and Kalman, TI
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 2004. 228: U174-U175, 2
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000223712800717