ONLINE DATABASE SEARCH - HIV-LS-318-MEMO
1. 45023 HIV-LS-318; PUBMED-HIV-3/22/2005
Indole and carbazole alkaloids from Glycosmis montana with weak anti-HIV and cytotoxic activities
Wang, J, Zheng, Y, Efferth, T, Wang, R, Shen, Y, and Hao, X
Phytochemistry 2005. 66(6): 697-701
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771893&dopt=abstract
2. 45024 HIV-LS-318; PUBMED-HIV-3/22/2005
Development of Low Molecular Weight HIV-1 Protease Dimerization Inhibitors
Hwang, YS and Chmielewski, J
J Med Chem 2005. 48(6): 2239-42
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771466&dopt=abstract
3. 45025 HIV-LS-318; PUBMED-HIV-3/22/2005
Structure Based Activity Prediction of HIV-1 Reverse Transcriptase Inhibitors
de Jonge, MR, Koymans, LM, Vinkers, HM , Daeyaert, FF, Heeres, J, Lewi, PJ, and Janssen, PA
J Med Chem 2005. 48(6): 2176-2183
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771460&dopt=abstract
4. 45026 HIV-LS-318; PUBMED-HIV-3/22/2005
Synthesis of Novel Diarylpyrimidine Analogues and Their Antiviral Activity against Human Immunodeficiency Virus Type 1
Guillemont, J, Pasquier, E, Palandjian, P, Vernier, D, Gaurrand, S, Lewi, PJ, Heeres, J, de, Jonge MR, Koymans, LM, Daeyaert, FF, Vinkers, MH, Arnold, E, Das, K, Pauwels, R, Andries, K, de, Bethune MP, Bettens, E, Hertogs, K, Wigerinck, P, Timmerman, P, and Janssen, PA
J Med Chem 2005. 48(6): 2072-2079
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771449&dopt=abstract
5. 45027 HIV-LS-318; PUBMED-HIV-3/22/2005
Design of HIV-1 Protease Inhibitors Active on Multidrug-Resistant Virus
Surleraux, DL, de, Kock HA, Verschueren, WG, Pille, GM, Maes, LJ, Peeters, A, Vendeville, S, De, Meyer S, Azijn, H, Pauwels, R, de, Bethune MP, King, NM, Prabu-Jeyabalan, M, Schiffer, CA, and Wigerinck, PB
J Med Chem 2005. 48(6): 1965-73
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771440&dopt=abstract
6. 45028 HIV-LS-318; EMBASE-HIV-3/22/2005
The fd phage and a peptide derived from its p8 coat protein interact with the HIV-1 Tat-NLS and inhibit its biological functions
Krichevsky, A, Rusnati, M, Bugatti, A, Waigmann, E, Shohat, S, and Loyter, A
Antiviral Research 2005. 66(1): 67-78
HYPERLINK:
http://www.sciencedirect.com/science/article/B6T2H-4FJXJKJ-1/2/24393053fd342e143ba92531fd1cbf3c
7. 45029 HIV-LS-318; PUBMED-HIV-3/22/2005
Design and Optimization of Tricyclic Phtalimide Analogues as Novel Inhibitors of HIV-1 Integrase
Verschueren, WG, Dierynck, I, Amssoms, KI, Hu, L, Boonants, PM, Pille, GM, Daeyaert, FF, Hertogs, K, Surleraux, DL, and Wigerinck, PB
J Med Chem 2005. 48(6): 1930-40
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771437&dopt=abstract
8. 45030 HIV-LS-318; PUBMED-HIV-3/22/2005
Design, Synthesis, and SAR of a Novel Pyrazinone Series with Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitory Activity
Heeres, J, de, Jonge MR, Koymans, LM, Daeyaert, FF, Vinkers, M, Van, Aken KJ, Arnold, E, Das, K, Kilonda, A, Hoornaert, GJ, Compernolle, F, Cegla, M, Azzam, RA, Andries, K, de, Bethune MP, Azijn, H, Pauwels, R, Lewi, PJ, and Janssen, PA
J Med Chem 2005. 48(6): 1910-1918
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771435&dopt=abstract
9. 45031 HIV-LS-318; PUBMED-HIV-3/22/2005
In Search of a Novel Anti-HIV Drug: Multidisciplinary Coordination in the Discovery of 4-[[4-[[4-[(1E)-2-Cyanoethenyl]-2,6-dimethylphenyl]amino]-2- pyrimidinyl]amino]benzonitrile (R278474, Rilpivirine)
Janssen, PA, Lewi, PJ, Arnold, E, Daeyaert, F, de, Jonge M, Heeres, J, Koymans, L, Vinkers, M, Guillemont, J, Pasquier, E, Kukla, M, Ludovici, D, Andries, K, de, Bethune MP, Pauwels, R, Das, K, Clark, AD Jr, Frenkel, YV, Hughes, SH, Medaer, B, De, Knaep F, Bohets, H, De, Clerck F, Lampo, A, Williams, P, and Stoffels, P
J Med Chem 2005. 48(6): 1901-1909
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771434&dopt=abstract
10. 45032 HIV-LS-318; PUBMED-HIV-3/22/2005
Discovery and Selection of TMC114, a Next Generation HIV-1 Protease Inhibitor
Surleraux, DL, Tahri, A, Verschueren, WG, Pille, GM, de, Kock HA, Jonckers, TH, Peeters, A, De, Meyer S, Azijn, H, Pauwels, R, de, Bethune MP, King, NM, Prabu-Jeyabalan, M, Schiffer, CA, and Wigerinck, PB
J Med Chem 2005. 48(6): 1813-22
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771427&dopt=abstract
11. 45033 HIV-LS-318; PUBMED-HIV-3/22/2005
Atazanavir: the advent of a new generation of more convenient protease inhibitors
Barreiro, P, Rendon, A, Rodriguez-Novoa, S, and Soriano, V
HIV Clin Trials 2005. 6(1): 50-61
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15765311&dopt=abstract
12. 45034 HIV-LS-318; EMBASE-HIV-3/22/2005
HIV protease inhibitors: synthesis and activity of N-aryl-N'-hydroxyalkyl hydrazide pseudopeptides
Marastoni, M, Baldisserotto, A, Trapella, C, McDonald, J, Bortolotti, F, and Tomatis, R
European Journal of Medicinal Chemistry 2005. In Press, Corrected Proof
HYPERLINK:
http://www.sciencedirect.com/science/article/B6VKY-4FJTNRY-3/2/74e0f5bd1626524fdf52ce04faa8c929
13. 45035 HIV-LS-318; PUBMED-HIV-3/22/2005
Tipranavir: a novel second-generation nonpeptidic protease inhibitor
Kandula, VR, Khanlou, H, and Farthing, C
Expert Rev Anti Infect Ther 2005. 3(1): 9-21
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15757454&dopt=abstract
14. 45036 HIV-LS-318; PUBMED-HIV-3/22/2005
The cellular HIV-1 Rev cofactor hRIP is required for viral replication
Yu, Z, Sanchez-Velar, N, Catrina, IE, Kittler, EL, Udofia, EB, and Zapp, ML
Proc Natl Acad Sci U S A 2005. 102(11): 4027-32
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15749819&dopt=abstract
15. 45037 HIV-LS-318; EMBASE-HIV-3/22/2005
Study on the interactions between anti-HIV-1 active compounds with trans-activation response RNA by affinity capillary electrophoresis
Ding, Li, Zhang, Xin-Xiang, Chang, Wen-Bao, Lin, Wei, and Yang, Ming
Journal of Chromatography B 2005. 814(1): 99-104
HYPERLINK:
http://www.sciencedirect.com/science/article/B6X0P-4DS7T1N-4/2/97a0752715dcbf41814c8ff5d06ef9f8
16. 45038 HIV-LS-318; PUBMED-HIV-3/22/2005
Dynamic receptor-based pharmacophore model development and its application in designing novel HIV-1 integrase inhibitors
Deng, J, Lee, KW, Sanchez, T, Cui, M, Neamati, N, and Briggs, JM
J Med Chem 2005. 48(5): 1496-1505
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15743192&dopt=abstract
17. 45039 HIV-LS-318; PUBMED-HIV-3/22/2005
Integrase inhibitors to treat HIV/AIDS
Pommier, Y, Johnson, AA, and Marchand, C
Nat Rev Drug Discov 2005. 4(3): 236-48
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15729361&dopt=abstract
18. 45040 HIV-LS-318; PUBMED-HIV-3/22/2005
A novel and efficient approach to discriminate between pre- and post-transcription HIV inhibitors
Daelemans, D, Pannecouque, C, Pavlakis, GN, Tabarrini, O, and De Clercq, E
Mol Pharmacol 2005.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15728798&dopt=abstract
19. 45041 HIV-LS-318; PUBMED-HIV-3/22/2005
5-Alkyl-2-alkylamino-6-(2,6-difluorophenylalkyl)-3,4-dihydropyrimidin-4(3H )-ones, a new series of potent, broad-spectrum non-nucleoside reverse transcriptase inhibitors belonging to the DABO family
Mai, A, Artico, M, Ragno, R, Sbardella, G, Massa, S, Musiu, C, Mura, M, Marturana, F, Cadeddu, A, Maga, G, and Colla, PL
Bioorg Med Chem 2005. 13(6): 2065-2077
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15727860&dopt=abstract
20. 45042 HIV-LS-318; PUBMED-HIV-3/22/2005
Hexitol nucleic acid-containing aptamers are efficient ligands of HIV-1 TAR RNA
Kolb, G, Reigadas, S, Boiziau, C, van Aerschot, A, Arzumanov, A, Gait, MJ, Herdewijn, P, and Toulme, JJ
Biochemistry 2005. 44(8): 2926-2933
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15723535&dopt=abstract
21. 45043 HIV-LS-318; WOS-HIV-3/13/2005
Adaptive inhibitors of the HIV-1 protease
Ohtaka, H and Freire, E
PROGRESS IN BIOPHYSICS & MOLECULAR BIOLOGY 2005. 88(2): 193-208, 16
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227204200002
22. 45044 HIV-LS-318; WOS-HIV-3/13/2005
Cluster analysis and three-dimensional QSAR studies of HIV-1 integrase inhibitors
Yuan, HB and Parrill, A
JOURNAL OF MOLECULAR GRAPHICS & MODELLING 2005. 23(4): 317-328, 12
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227150400003
23. 45045 HIV-LS-318; WOS-HIV-3/13/2005
A novel once-daily protease inhibitor
Piliero, PJ
DRUGS OF TODAY 2004. 40(11): 901-912, 12
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227168600002
24. 45046 HIV-LS-318; WOS-HIV-3/13/2005
The N-terminus of HIV-1 Tat protein is essential for Tat-TAR RNA interaction
Chaloin, O, Peter, JC, Briand, JP, Masquida, B, Desgranges, C, Muller, S, and Hoebeke, J
CELLULAR AND MOLECULAR LIFE SCIENCES 2005. 62(3): 355-361, 7
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227149600010
25. 45047 HIV-LS-318; WOS-HIV-3/13/2005
Human immunodeficiency virus-reverse transcriptase inhibition and hepatitis C virus RNA-dependent RNA polymerase inhibition activities of fullerene derivatives
Mashino, T, Shimotohno, K, Ikegami, N, Nishikawa, D, Okuda, K, Takahashi, K, Nakamura, S, and Mochizuki, M
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 2005. 15(4): 1107-1109, 3
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227135400047
26. 45048 HIV-LS-318; WOS-HIV-3/13/2005
Analysis of interactions of DNA polymerase beta and reverse transcriptases of human immunodeficiency and mouse leukemia viruses with dNTP analogs containing a modified sugar residue
Lebedeva, NA, Seredina, TA, Silnikov, VN, Abramova, TV, Levina, AS, Khodyreva, SN, Rechkunova, NI, and Lavrik, OI
BIOCHEMISTRY-MOSCOW 2005. 70(1): 1-7, 7
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227139600001
27. 45049 HIV-LS-318; WOS-HIV-3/20/2005
Substrate properties of dinucleoside 5 ',5 ''-oligophosphates in the reactions catalyzed by HIV reverse transcriptase, E-coli DNA polymerase I, and E-coli RNA polymerase
Skoblov, AY, Sosunov, VV, Victorova, LS, Skoblov, YS, and Kukhanova, MK
RUSSIAN JOURNAL OF BIOORGANIC CHEMISTRY 2005. 31(1): 48-57, 10
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227321000006
28. 45050 HIV-LS-318; WOS-HIV-3/20/2005
SIRT1 regulates HIV transcription via Tat deacetylation
Pagans, S, Pedal, A, North, BJ, Kaehlcke, K, Marshall, BL, Dorr, A, Hetzer-Egger, C, Henklein, P, Frye, R, McBurney, MW, Hruby, H, Jung, M, Verdin, E, and Ott, M
PLOS BIOLOGY 2005. 3(2): 210-220, 11
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227404100006
29. 45051 HIV-LS-318; WOS-HIV-3/20/2005
Sulfonated naphthyl porphyrins as agents against HIV-1
Dixon, DW, Gill, AF, Giribabu, L, Vzorov, AN, Alam, AB, and Compans, RW
JOURNAL OF INORGANIC BIOCHEMISTRY 2005. 99(3): 813-821, 9
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227374900017
30. 45052 HIV-LS-318; WOS-HIV-3/20/2005
HIV protease inhibitors-induced atherosclerosis: Prevention by alpha-tocopherol
Munteanu, A, Ricciarelli, R, and Zingg, JM
IUBMB LIFE 2004. 56(10): 629-631, 3
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227425000008