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ONLINE DATABASE SEARCH - HIV-LS-318-MEMO

1. 45023 HIV-LS-318; PUBMED-HIV-3/22/2005

Indole and carbazole alkaloids from Glycosmis montana with weak anti-HIV and cytotoxic activities

Wang, J, Zheng, Y, Efferth, T, Wang, R, Shen, Y, and Hao, X

Phytochemistry 2005. 66(6): 697-701


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771893&dopt=abstract


2. 45024 HIV-LS-318; PUBMED-HIV-3/22/2005

Development of Low Molecular Weight HIV-1 Protease Dimerization Inhibitors

Hwang, YS and Chmielewski, J

J Med Chem 2005. 48(6): 2239-42


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771466&dopt=abstract


3. 45025 HIV-LS-318; PUBMED-HIV-3/22/2005

Structure Based Activity Prediction of HIV-1 Reverse Transcriptase Inhibitors

de Jonge, MR, Koymans, LM, Vinkers, HM , Daeyaert, FF, Heeres, J, Lewi, PJ, and Janssen, PA

J Med Chem 2005. 48(6): 2176-2183


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771460&dopt=abstract


4. 45026 HIV-LS-318; PUBMED-HIV-3/22/2005

Synthesis of Novel Diarylpyrimidine Analogues and Their Antiviral Activity against Human Immunodeficiency Virus Type 1

Guillemont, J, Pasquier, E, Palandjian, P, Vernier, D, Gaurrand, S, Lewi, PJ, Heeres, J, de, Jonge MR, Koymans, LM, Daeyaert, FF, Vinkers, MH, Arnold, E, Das, K, Pauwels, R, Andries, K, de, Bethune MP, Bettens, E, Hertogs, K, Wigerinck, P, Timmerman, P, and Janssen, PA

J Med Chem 2005. 48(6): 2072-2079


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771449&dopt=abstract


5. 45027 HIV-LS-318; PUBMED-HIV-3/22/2005

Design of HIV-1 Protease Inhibitors Active on Multidrug-Resistant Virus

Surleraux, DL, de, Kock HA, Verschueren, WG, Pille, GM, Maes, LJ, Peeters, A, Vendeville, S, De, Meyer S, Azijn, H, Pauwels, R, de, Bethune MP, King, NM, Prabu-Jeyabalan, M, Schiffer, CA, and Wigerinck, PB

J Med Chem 2005. 48(6): 1965-73


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771440&dopt=abstract



6. 45028 HIV-LS-318; EMBASE-HIV-3/22/2005

The fd phage and a peptide derived from its p8 coat protein interact with the HIV-1 Tat-NLS and inhibit its biological functions

Krichevsky, A, Rusnati, M, Bugatti, A, Waigmann, E, Shohat, S, and Loyter, A

Antiviral Research 2005. 66(1): 67-78


HYPERLINK:

http://www.sciencedirect.com/science/article/B6T2H-4FJXJKJ-1/2/24393053fd342e143ba92531fd1cbf3c


7. 45029 HIV-LS-318; PUBMED-HIV-3/22/2005

Design and Optimization of Tricyclic Phtalimide Analogues as Novel Inhibitors of HIV-1 Integrase

Verschueren, WG, Dierynck, I, Amssoms, KI, Hu, L, Boonants, PM, Pille, GM, Daeyaert, FF, Hertogs, K, Surleraux, DL, and Wigerinck, PB

J Med Chem 2005. 48(6): 1930-40


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771437&dopt=abstract


8. 45030 HIV-LS-318; PUBMED-HIV-3/22/2005

Design, Synthesis, and SAR of a Novel Pyrazinone Series with Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitory Activity

Heeres, J, de, Jonge MR, Koymans, LM, Daeyaert, FF, Vinkers, M, Van, Aken KJ, Arnold, E, Das, K, Kilonda, A, Hoornaert, GJ, Compernolle, F, Cegla, M, Azzam, RA, Andries, K, de, Bethune MP, Azijn, H, Pauwels, R, Lewi, PJ, and Janssen, PA

J Med Chem 2005. 48(6): 1910-1918


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771435&dopt=abstract


9. 45031 HIV-LS-318; PUBMED-HIV-3/22/2005

In Search of a Novel Anti-HIV Drug: Multidisciplinary Coordination in the Discovery of 4-[[4-[[4-[(1E)-2-Cyanoethenyl]-2,6-dimethylphenyl]amino]-2- pyrimidinyl]amino]benzonitrile (R278474, Rilpivirine)

Janssen, PA, Lewi, PJ, Arnold, E, Daeyaert, F, de, Jonge M, Heeres, J, Koymans, L, Vinkers, M, Guillemont, J, Pasquier, E, Kukla, M, Ludovici, D, Andries, K, de, Bethune MP, Pauwels, R, Das, K, Clark, AD Jr, Frenkel, YV, Hughes, SH, Medaer, B, De, Knaep F, Bohets, H, De, Clerck F, Lampo, A, Williams, P, and Stoffels, P

J Med Chem 2005. 48(6): 1901-1909


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771434&dopt=abstract


10. 45032 HIV-LS-318; PUBMED-HIV-3/22/2005

Discovery and Selection of TMC114, a Next Generation HIV-1 Protease Inhibitor

Surleraux, DL, Tahri, A, Verschueren, WG, Pille, GM, de, Kock HA, Jonckers, TH, Peeters, A, De, Meyer S, Azijn, H, Pauwels, R, de, Bethune MP, King, NM, Prabu-Jeyabalan, M, Schiffer, CA, and Wigerinck, PB

J Med Chem 2005. 48(6): 1813-22


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771427&dopt=abstract


11. 45033 HIV-LS-318; PUBMED-HIV-3/22/2005

Atazanavir: the advent of a new generation of more convenient protease inhibitors

Barreiro, P, Rendon, A, Rodriguez-Novoa, S, and Soriano, V

HIV Clin Trials 2005. 6(1): 50-61


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15765311&dopt=abstract


12. 45034 HIV-LS-318; EMBASE-HIV-3/22/2005

HIV protease inhibitors: synthesis and activity of N-aryl-N'-hydroxyalkyl hydrazide pseudopeptides

Marastoni, M, Baldisserotto, A, Trapella, C, McDonald, J, Bortolotti, F, and Tomatis, R

European Journal of Medicinal Chemistry 2005. In Press, Corrected Proof


HYPERLINK:

http://www.sciencedirect.com/science/article/B6VKY-4FJTNRY-3/2/74e0f5bd1626524fdf52ce04faa8c929


13. 45035 HIV-LS-318; PUBMED-HIV-3/22/2005

Tipranavir: a novel second-generation nonpeptidic protease inhibitor

Kandula, VR, Khanlou, H, and Farthing, C

Expert Rev Anti Infect Ther 2005. 3(1): 9-21


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15757454&dopt=abstract


14. 45036 HIV-LS-318; PUBMED-HIV-3/22/2005

The cellular HIV-1 Rev cofactor hRIP is required for viral replication

Yu, Z, Sanchez-Velar, N, Catrina, IE, Kittler, EL, Udofia, EB, and Zapp, ML

Proc Natl Acad Sci U S A 2005. 102(11): 4027-32


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15749819&dopt=abstract


15. 45037 HIV-LS-318; EMBASE-HIV-3/22/2005

Study on the interactions between anti-HIV-1 active compounds with trans-activation response RNA by affinity capillary electrophoresis

Ding, Li, Zhang, Xin-Xiang, Chang, Wen-Bao, Lin, Wei, and Yang, Ming

Journal of Chromatography B 2005. 814(1): 99-104


HYPERLINK:

http://www.sciencedirect.com/science/article/B6X0P-4DS7T1N-4/2/97a0752715dcbf41814c8ff5d06ef9f8


16. 45038 HIV-LS-318; PUBMED-HIV-3/22/2005

Dynamic receptor-based pharmacophore model development and its application in designing novel HIV-1 integrase inhibitors

Deng, J, Lee, KW, Sanchez, T, Cui, M, Neamati, N, and Briggs, JM

J Med Chem 2005. 48(5): 1496-1505


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15743192&dopt=abstract


17. 45039 HIV-LS-318; PUBMED-HIV-3/22/2005

Integrase inhibitors to treat HIV/AIDS

Pommier, Y, Johnson, AA, and Marchand, C

Nat Rev Drug Discov 2005. 4(3): 236-48


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15729361&dopt=abstract


18. 45040 HIV-LS-318; PUBMED-HIV-3/22/2005

A novel and efficient approach to discriminate between pre- and post-transcription HIV inhibitors

Daelemans, D, Pannecouque, C, Pavlakis, GN, Tabarrini, O, and De Clercq, E

Mol Pharmacol 2005.


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15728798&dopt=abstract


19. 45041 HIV-LS-318; PUBMED-HIV-3/22/2005

5-Alkyl-2-alkylamino-6-(2,6-difluorophenylalkyl)-3,4-dihydropyrimidin-4(3H )-ones, a new series of potent, broad-spectrum non-nucleoside reverse transcriptase inhibitors belonging to the DABO family

Mai, A, Artico, M, Ragno, R, Sbardella, G, Massa, S, Musiu, C, Mura, M, Marturana, F, Cadeddu, A, Maga, G, and Colla, PL

Bioorg Med Chem 2005. 13(6): 2065-2077


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15727860&dopt=abstract


20. 45042 HIV-LS-318; PUBMED-HIV-3/22/2005

Hexitol nucleic acid-containing aptamers are efficient ligands of HIV-1 TAR RNA

Kolb, G, Reigadas, S, Boiziau, C, van Aerschot, A, Arzumanov, A, Gait, MJ, Herdewijn, P, and Toulme, JJ

Biochemistry 2005. 44(8): 2926-2933


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15723535&dopt=abstract


21. 45043 HIV-LS-318; WOS-HIV-3/13/2005

Adaptive inhibitors of the HIV-1 protease

Ohtaka, H and Freire, E

PROGRESS IN BIOPHYSICS & MOLECULAR BIOLOGY 2005. 88(2): 193-208, 16


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227204200002


22. 45044 HIV-LS-318; WOS-HIV-3/13/2005

Cluster analysis and three-dimensional QSAR studies of HIV-1 integrase inhibitors

Yuan, HB and Parrill, A

JOURNAL OF MOLECULAR GRAPHICS & MODELLING 2005. 23(4): 317-328, 12


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227150400003



23. 45045 HIV-LS-318; WOS-HIV-3/13/2005

A novel once-daily protease inhibitor

Piliero, PJ

DRUGS OF TODAY 2004. 40(11): 901-912, 12


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227168600002


24. 45046 HIV-LS-318; WOS-HIV-3/13/2005

The N-terminus of HIV-1 Tat protein is essential for Tat-TAR RNA interaction

Chaloin, O, Peter, JC, Briand, JP, Masquida, B, Desgranges, C, Muller, S, and Hoebeke, J

CELLULAR AND MOLECULAR LIFE SCIENCES 2005. 62(3): 355-361, 7


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227149600010


25. 45047 HIV-LS-318; WOS-HIV-3/13/2005

Human immunodeficiency virus-reverse transcriptase inhibition and hepatitis C virus RNA-dependent RNA polymerase inhibition activities of fullerene derivatives

Mashino, T, Shimotohno, K, Ikegami, N, Nishikawa, D, Okuda, K, Takahashi, K, Nakamura, S, and Mochizuki, M

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 2005. 15(4): 1107-1109, 3


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227135400047


26. 45048 HIV-LS-318; WOS-HIV-3/13/2005

Analysis of interactions of DNA polymerase beta and reverse transcriptases of human immunodeficiency and mouse leukemia viruses with dNTP analogs containing a modified sugar residue

Lebedeva, NA, Seredina, TA, Silnikov, VN, Abramova, TV, Levina, AS, Khodyreva, SN, Rechkunova, NI, and Lavrik, OI

BIOCHEMISTRY-MOSCOW 2005. 70(1): 1-7, 7


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227139600001


27. 45049 HIV-LS-318; WOS-HIV-3/20/2005

Substrate properties of dinucleoside 5 ',5 ''-oligophosphates in the reactions catalyzed by HIV reverse transcriptase, E-coli DNA polymerase I, and E-coli RNA polymerase

Skoblov, AY, Sosunov, VV, Victorova, LS, Skoblov, YS, and Kukhanova, MK

RUSSIAN JOURNAL OF BIOORGANIC CHEMISTRY 2005. 31(1): 48-57, 10


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227321000006


28. 45050 HIV-LS-318; WOS-HIV-3/20/2005

SIRT1 regulates HIV transcription via Tat deacetylation

Pagans, S, Pedal, A, North, BJ, Kaehlcke, K, Marshall, BL, Dorr, A, Hetzer-Egger, C, Henklein, P, Frye, R, McBurney, MW, Hruby, H, Jung, M, Verdin, E, and Ott, M

PLOS BIOLOGY 2005. 3(2): 210-220, 11


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227404100006


29. 45051 HIV-LS-318; WOS-HIV-3/20/2005

Sulfonated naphthyl porphyrins as agents against HIV-1

Dixon, DW, Gill, AF, Giribabu, L, Vzorov, AN, Alam, AB, and Compans, RW

JOURNAL OF INORGANIC BIOCHEMISTRY 2005. 99(3): 813-821, 9


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227374900017


30. 45052 HIV-LS-318; WOS-HIV-3/20/2005

HIV protease inhibitors-induced atherosclerosis: Prevention by alpha-tocopherol

Munteanu, A, Ricciarelli, R, and Zingg, JM

IUBMB LIFE 2004. 56(10): 629-631, 3


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227425000008


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