ONLINE DATABASE SEARCH - HIV-LS-321-MEMO
1. 45215 HIV-LS-321; PUBMED-HIV-5/2/2005
Discovery of Small-Molecule Human Immunodeficiency Virus Type 1 Entry Inhibitors That Target the gp120-Binding Domain of CD4
Yang, QE, Stephen, AG, Adelsberger, JW , Roberts, PE, Zhu, W, Currens, MJ, Feng, Y, Crise, BJ, Gorelick, RJ, Rein, AR, Fisher, RJ, Shoemaker, RH, and Sei, S
J Virol 2005 . 79(10): 6122-6133
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15857997&dopt=abstract
2. 45216 HIV-LS-321; PUBMED-HIV-5/2/2005
Anti-HIV Protease Activity from Rosa Family Plant Extracts and Rosamultin from Rosa rugosa
Park, JC, Kim, SC, Choi, MR, Song, SH, Yoo, EJ, Kim, SH, Miyashiro, H, and Hattori, M
J Med Food 2005. 8(1): 107-109
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15857219&dopt=abstract
3. 45217 HIV-LS-321; PUBMED-HIV-5/2/2005
Targeting tn5 transposase identifies human immunodeficiency virus type 1 inhibitors
Ason, B, Knauss, DJ, Balke, AM, Merkel, G, Skalka, AM, and Reznikoff, WS
Antimicrob Agents Chemother 2005. 49(5): 2035-2043
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15855529&dopt=abstract
4. 45218 HIV-LS-321; SCIFINDER-HIV-4/25/2005
Preparation of 2-aminobenzimidazoles for the treatment of HIV/AIDS
Schohe-Loop, Rudolf, Paessens, Arnold, Bauser, Marcus, Koebberling, Johannes, Dittmer, Frank, Henninger, Kerstin, Lang, Dieter, and Paulsen, Daniela
PATENT: WO 2005019186 ISSUE DATE: 20050303
APPLICATION: 2004 PP: 59 pp.
ASSIGNEE: (Bayer Healthcare A.-G., Germany
5. 45219 HIV-LS-321; PUBMED-HIV-5/2/2005
Novel human immunodeficiency virus type 1 protease mutations potentially involved in resistance to protease inhibitors
Svicher, V, Ceccherini-Silberstein, F, Erba, F, Santoro, M, Gori, C, Bellocchi, MC, Giannella, S, Trotta, MP, Monforte, A, Antinori, A, and Perno, CF
Antimicrob Agents Chemother 2005. 49(5): 2015-2025
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15855527&dopt=abstract
6. 45220 HIV-LS-321; PUBMED-HIV-5/2/2005
Mechanism of Anti-Human Immunodeficiency Virus Activity of {beta}-D-6-Cyclopropylamino-2',3'-Didehydro-2',3'-Dideoxyguanosine
Ray, AS, Hernandez-Santiago, BI, Mathew, JS, Murakami, E, Bozeman, C, Xie, MY, Dutschman, GE, Gullen, E, Yang, Z, Hurwitz, S, Cheng, YC, Chu, CK, McClure, H, Schinazi, RF, and Anderson, KS
Antimicrob Agents Chemother 2005. 49(5): 1994-2001
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15855524&dopt=abstract
7. 45221 HIV-LS-321; SCIFINDER-HIV-4/25/2005
Preparation of 5-membered heterocycles, in particular pyrazoles and imidazoles, as p38 kinase inhibitors
Fryszman, Olga M, Lang, Hengyuan, Lan, Jiong, Chang, Edcon, and Fang, Yunfeng
PATENT: WO 2005009973 ISSUE DATE: 20050203
APPLICATION: 2004 PP: 197 pp.
ASSIGNEE: (Triad Therapeuctics, Inc. USA
8. 45222 HIV-LS-321; PUBMED-HIV-5/2/2005
Evaluation of selected South African medicinal plants for inhibitory properties against human immunodeficiency virus type 1 reverse transcriptase and integrase
Bessong, PO, Obi, CL, Andreola, ML, Rojas, LB, Pouysegu, L, Igumbor, E, Meyer, JJ, Quideau, S, and Litvak, S
J Ethnopharmacol 2005. 99(1): 83-91
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15848024&dopt=abstract
9. 45223 HIV-LS-321; PUBMED-HIV-5/2/2005
Limited development and progression of resistance of HIV-1 to the nucleoside analogue reverse transcriptase inhibitor lamivudine in human primary macrophages
Aquaro, S, Svicher, V, Ceccherini-Silberstein, F, Cenci, A, Marcuccilli, F, Giannella, S, Marcon, L, Calio, R, Balzarini, J, and Perno, CF
J Antimicrob Chemother 2005.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15845785&dopt=abstract
10. 45224 HIV-LS-321; PUBMED-HIV-5/2/2005
Inhibition of HIV-1 replication by caffeine and caffeine-related methylxanthines
Nunnari, G, Argyris, E, Fang, J, Mehlman, KE, Pomerantz, RJ, and Daniel, R
Virology 2005. 335(2): 177-184
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15840517&dopt=abstract
11. 45225 HIV-LS-321; PUBMED-HIV-5/2/2005
Oximinoarylsulfonamides as potent HIV protease inhibitors
Yeung, CM, Klein, LL, Flentge, CA, Randolph, JT, Zhao, C, Sun, M, Dekhtyar, T, Stoll, VS, and Kempf, DJ
Bioorg Med Chem Lett 2005. 15(9): 2275-2278
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15837308&dopt=abstract
12. 45226 HIV-LS-321; PUBMED-HIV-5/2/2005
Suppression of HIV-1 infection by a small molecule inhibitor of the ATM kinase
Lau, A, Swinbank, KM, Ahmed, PS, Taylor, DL, Jackson, SP, Smith, GC, and O'connor, MJ
Nat Cell Biol 2005.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15834407&dopt=abstract
13. 45227 HIV-LS-321; SCIFINDER-HIV-4/25/2005
Inhibition of HIV-1 gene expression by retroviral vector-mediated small-guide RNAs that direct specific RNA cleavage by tRNase ZL
Habu, Yuichiro, Miyano-Kurosaki, Naoko, Kitano, Michiko, Endo, Yumihiko, Yukita, Masakazu, Ohira, Shigeru, Takaku, Hiroaki, Nashimoto, Masayuki, and Takaku, Hiroshi
Nucleic Acids Research 2005. 33(1): 235-243
14. 45228 HIV-LS-321; PUBMED-HIV-5/2/2005
THE AMINO ACID N136 IN HIV-1 REVERSE TRANSCRIPTASE (RT) MAINTAINS EFFICIENT ASSOCIATION OF BOTH RT SUBUNITS AND ENABLES THE RATIONAL DESIGN OF NOVEL RT INHIBITORS
Balzarini, J, Auxerx, J, Rodriguez-Barrios, F, Chedad, A, Farkas, V, Ceccherini-Silberstein, F, Garcia-Aparicio, C, Velazquez, S, De Clercq, E, Perno, CF, Camarasa, MJ, and Gago, F
Mol Pharmacol 2005.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15833734&dopt=abstract
15. 45229 HIV-LS-321; SCIFINDER-HIV-4/25/2005
Essential regions for antiviral activities of actinohivin, a sugar-binding anti-human immunodeficiency virus protein from an actinomycete
Takahashi, Atsushi, Inokoshi, Junji, Chiba, Harumi, Omura, Satoshi, and Tanaka, Haruo
Archives of Biochemistry and Biophysics 2005. 437(2): 233-240
16. 45230 HIV-LS-321; SCIFINDER-HIV-4/25/2005
Dihydropyrimidinyl and other heterocyclic compound dipeptidyl peptidase IV (DPPIV) inhibitors
Cao, Sheldon X, Feng, Jun, Gwaltney, Stephen L, Kaldor, Stephen W, Stafford, Jeffrey A, Wallace, Michael B, Xiao, Xiao-Yi, and Zhang, Zhiyuan
PATENT: WO 2005026148 ISSUE DATE: 20050324
APPLICATION: 2004 PP: 161 pp.
ASSIGNEE: (Syrrx, Inc. USA
17. 45231 HIV-LS-321; PUBMED-HIV-5/2/2005
Blockade of chemokine-induced signalling inhibits CCR5-dependent HIV infection in vitro without blocking gp120/CCR5 interaction
Grainger, DJ and Lever, AM
Retrovirology 2005. 2(1): 23
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15807900&dopt=abstract
18. 45232 HIV-LS-321; WOS-HIV-4/24/2005
4D-QSAR models of HOE/BAY-793 analogues as HIV-1 protease inhihitors
da Cunha, EFF, Albuquerque, MG, Antunes, OAC, and de Alencastro, RB
QSAR & COMBINATORIAL SCIENCE 2005. 24(2): 240-253, 14
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000228251600006
19. 45233 HIV-LS-321; WOS-HIV-4/24/2005
Synthesis and biological evaluation of 2 ',3 '-didehydro-2 ', 3 '-dideoxy-9-deazaguanosine, a monophosphate prodrug and two analogues, 2 ',3 '-dideoxy-9-deazaguanosine and 2 ',3 '-didehydro-2 ',3 '-dideoxy-9-deazainosine
Liu, MC, Luo, MZ, Mozdziesz, DE, Dutschman, GE, Gullen, EA, Cheng, YC, and Sartorelli, AC
NUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS 2005. 24(2): 135-145, 11
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000228077200005
20. 45234 HIV-LS-321; SCIFINDER-HIV-4/25/2005
<04 Article Title>
Embrey, Mark W, Wai, John S, Funk, Timothy W, Homnick, Carl F, Perlow, Debbie S, Young, Steven D, Vacca, Joseph P, Hazuda, Daria J, Felock, Peter J, Stillmock, Kara A, Witmer, Marc V, Moyer, Gregory, Schleif, William A, Gabryelski, Lori J, Jin, Lixia, Chen, I-Wu, Ellis, Joan D, Wong, Bradley K, Lin, Jiunn H, Leonard, Yvonne M, Tsou, Nancy N, and Zhuang, Linghang
<10 Journal Title> 2005.(<24 Issue ID>): <25 Page(s)>
21. 45235 HIV-LS-321; SCIFINDER-HIV-4/25/2005
Polypeptide multimers comprising coiled coil structure and a-helical structure for use as antiviral, anti-HIV and anti-SIV agents
Weiss, Carol D, He, Yong, Vassell, Russell, and De, Rosny Eve
PATENT: WO 2005018666 ISSUE DATE: 20050303
APPLICATION: 2003 PP: 84 pp.
ASSIGNEE: (The Government of the United States of America, as Represented by the Department of Health and Human Services USA and De Rosny, Eve
22. 45236 HIV-LS-321; SCIFINDER-HIV-4/25/2005
Preparation of phenanthridine derivatives as anti-viral agents
Tor, Yitzhak and Luedtke, Nathan
PATENT: WO 2005016343 ISSUE DATE: 20050224
APPLICATION: 2004 PP: 58 pp.
ASSIGNEE: (The Regents of the University of California, USA
23. 45237 HIV-LS-321; SCIFINDER-HIV-4/25/2005
Ex Vivo Modeling of the Effects of Mycophenolic Acid on HIV Infection: Considerations for Antiviral Therapy
Kaur, Rupinderjeet, Klichko, Vladimir, and Margolis, David
AIDS Research and Human Retroviruses 2005. 21(2): 116-124
24. 45238 HIV-LS-321; SCIFINDER-HIV-4/25/2005
A preparation of antiviral and antibacterial derivatives of dithioxopyranodipyrimidine and their 10-aza-analogs
Tets, VV, Krasnov, KA, and Ashkinazi, RI
PATENT: RU 2246496 ISSUE DATE: 20050220
APPLICATION: 2003-62807 PP: No pp. given
ASSIGNEE: (Russia)
25. 45239 HIV-LS-321; SCIFINDER-HIV-4/25/2005
Preparation of nucleobase phosphonate analogs for antiviral treatment and as retroviral reverse transcriptase inhibitors
Krawczyk, Steven H
PATENT: WO 2005012324 ISSUE DATE: 20050210
APPLICATION: 2004 PP: 140 pp.
ASSIGNEE: (Gilead Sciences, Inc. USA
26. 45240 HIV-LS-321; SCIFINDER-HIV-4/25/2005
Trimeric Membrane-anchored gp41 Inhibits HIV Membrane Fusion
Lenz, Oliver, Dittmar, Matthias T, Wagner, Andreas, Ferko, Boris, Vorauer-Uhl, Karola, Stiegler, Gabriela, and Weissenhorn, Winfried
Journal of Biological Chemistry 2005. 280(6): 4095-4101
27. 45241 HIV-LS-321; WOS-HIV-4/24/2005
Amino acid derivatives, part 2: Synthesis, antiviral, and antitumor activity of simple protected amino acids functionalized at N-terminus with naphthalene side chain
Ali, IAI, Al-Masoudi, IA, Saeed, B, Al-Masoudi, NA, and La Colla, P
HETEROATOM CHEMISTRY 2005. 16(2): 148-155, 8
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000228057400008
28. 45242 HIV-LS-321; WOS-HIV-4/24/2005
Synthesis and antiviral activity of some no vel isatin derivatives
Selvam, P, Rajasekaran, A, Dharamsi, A, Ahmed, KL, Musthafa, SM, Poornima, K, Pournami, KA, Murugesh, N, Chandramohan, M, and De, Clercq E
ASIAN JOURNAL OF CHEMISTRY 2005. 17(1): 443-448, 6
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000228191800064
29. 45243 HIV-LS-321; WOS-HIV-4/24/2005
Antiviral activity of serum from the American alligator (Alligator mississippiensis)
Merchant, ME, Pallansch, M, Paulman, RL, Wells, JB, Nalca, A, and Ptak, R
ANTIVIRAL RESEARCH 2005. 66(1): 35-38, 4
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000228237800006
30. 45244 HIV-LS-321; WOS-HIV-5/1/2005
Synthesis of 1-[2-hydroxy thoxy)methyl]-6-(5,6,7,8-tetrahydronaphthylmethyl-1) thymine as novel inhibitor against drug-resistant HIV mutants
Meng, G, Kuang, YY, Ji, L, and Chen, FE
SYNTHETIC COMMUNICATIONS 2005. 35(8): 1095-1102, 8
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000228451200012
31. 45245 HIV-LS-321; WOS-HIV-5/1/2005
Marked depletion of glycosylation sites in HIV-1 gp120 under selection pressure by the mannose-specific plant lectins of Hippeastrum hybrid and Galanthus nivalis
Balzarini, J, Van Laethem, K, Hatse, S , Froeyen, M, Van Damme, E, Bolmstedt, A, Peumans, W, De Clercq, E, and Schols, D
MOLECULAR PHARMACOLOGY 2005. 67(5): 1556-1565, 10
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000228387900022
32. 45246 HIV-LS-321; WOS-HIV-5/1/2005
ATP gamma S disrupts human immunodeficiency virus type 1 virion core integrity
Gurer, C, Hoglund, A, Hoglund, S, and Luban, J
JOURNAL OF VIROLOGY 2005. 79(9): 5557-5567, 11
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000228433100033
33. 45247 HIV-LS-321; WOS-HIV-5/1/2005
Macrophage inflammatory protein 1 alpha inhibits postentry steps of human immunodeficiency virus type 1 infection via suppression of intracellular cyclic AMP
Amella, CA, Sherry, B, Shepp, DH, and Schmidtmayerova, H
JOURNAL OF VIROLOGY 2005. 79(9): 5625-5631, 7
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000228433100040
34. 45248 HIV-LS-321; WOS-HIV-5/1/2005
Some reactions of 3-chloroisoindolium salts with nucleophiles: access to isoindole derivatives and ellipticine analogues as potential antiviral agents
Hamed, AA
JOURNAL OF CHEMICAL RESEARCH-S 2005.(1): 54-58, 5
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000228312800016