ONLINE DATABASE SEARCH - HIV-LS-325-MEMO
1. 47531 HIV-LS-325; PUBMED-HIV-6/27/2005
Synthesis and antiviral activities of novel N-alkoxy-arylsulfonamide-based HIV protease inhibitors
Sherrill, RG, Furfine, ES, Hazen, RJ, Miller, JF, Reynolds, DJ, Sammond, DM, Spaltenstein, A, Wheelan, P, and Wright, LL
Bioorg Med Chem Lett 2005.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15975788&dopt=abstract
2. 47532 HIV-LS-325; SCIFINDER-HIV-6/20/2005
Mechanistic Insights into the Suppression of Drug Resistance by Human Immunodeficiency Virus Type 1 Reverse Transcriptase Using a-Boranophosphate Nucleoside Analogs
Deval, Jerome, Alvarez, Karine, Selmi, Boulbaba, Bermond, Marielle, Boretto, Joelle, Guerreiro, Catherine, Mulard, Laurence, and Canard, Bruno
Journal of Biological Chemistry 2005. 280(5): 3838-3846
3. 47533 HIV-LS-325; PUBMED-HIV-6/27/2005
Novel 1-[2-(Diarylmethoxy)ethyl]-2-methyl-5-nitroimidazoles as HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors. A Structure-Activity Relationship Investigation
De Martino, G, La Regina, G, Di, Pasquali A, Ragno, R, Bergamini, A, Ciaprini, C, Sinistro, A, Maga, G, Crespan, E , Artico, M, and Silvestri, R
J Med Chem 2005. 48(13): 4378-4388
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15974590&dopt=abstract
4. 47534 HIV-LS-325; PUBMED-HIV-6/27/2005
First Synthesis and Evaluation of the Inhibitory Effects of Aza Analogues of TSAO on HIV-1 Replication
Nguyen, Van Nhien A, Tomassi, C, Len, C, Marco-Contelles, JL, Balzarini, J, Pannecouque, C, De Clercq, E, and Postel, D
J Med Chem 2005. 48(13): 4276-4284
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15974581&dopt=abstract
5. 47535 HIV-LS-325; PUBMED-HIV-6/27/2005
Anti-HIV Bioactive Stilbene Dimers of Caragana rosea
Yang, GX, Zhou, JT, Li, YZ, and Hu, CQ
Planta Med 2005. 71(6): 569-71
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15971132&dopt=abstract
6. 47536 HIV-LS-325; PUBMED-HIV-6/27/2005
Thiourea-based non-nucleoside inhibitors of HIV reverse transcriptase as bifunctional organocatalysts in the asymmetric Strecker synthesis
Tsogoeva, SB, Hateley, MJ, Yalalov, DA, Meindl, K, Weckbecker, C, and Huthmacher, K
Bioorg Med Chem 2005.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15964195&dopt=abstract
7. 47537 HIV-LS-325; SCIFINDER-HIV-6/20/2005
Diazaindole-dicarbonyl-piperazinyl antiviral agents
Bender, John A, Yang, Zhong, Kadow, John F, and Meanwell, Nicholas A
PATENT: US 20050124623 ISSUE DATE: 20050609
APPLICATION: 2004-62054 PP: 87 pp.
ASSIGNEE: (USA)
8. 47538 HIV-LS-325; PUBMED-HIV-6/27/2005
Structure and anti-HIV activity of micrandilactones B and C, new nortriterpenoids possessing a unique skeleton from Schisandra micrantha
Li, RT, Han, QB, Zheng, YT, Wang, RR, Yang, LM, Lu, Y, Sang, SQ, Zheng, QT, Zhao, QS, and Sun, HD
Chem Commun (Camb) 2005.(23): 2936-8
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15957031&dopt=abstract
9. 47539 HIV-LS-325; PUBMED-HIV-6/27/2005
In vitro HIV type 1 reverse transcriptase inhibitory activities of Thai medicinal plants and Canna indica L. rhizomes
Woradulayapinij, W, Soonthornchareonnon, N, and Wiwat, C
J Ethnopharmacol 2005.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15951145&dopt=abstract
10. 47540 HIV-LS-325; SCIFINDER-HIV-6/20/2005
Inhibiting replication of a retrovirus, such as human immunodeficiency virus (HIV), through modulation of HIV Vif- or Vpu-mediated ubiquitylation of host cell proteins, such as CEM15 or CD4
Payan, Donald G and Jenkins, Yonchu
PATENT: WO 2005047476 ISSUE DATE: 20050526
APPLICATION: 2004 PP: 109 pp.
ASSIGNEE: (Rigel Pharmaceuticals, Inc. USA
11. 47541 HIV-LS-325; SCIFINDER-HIV-6/20/2005
Methods and compositions for the inhibition of HIV-1 replication in hum an cells using inhibitors of p21/CDKN1A activity or gene expression, and anti-AIDS uses
Wahl, Sharon M, Vazquez-Maldonado, Nancy, and Greenwell-Wild, Teresa
PATENT: WO 2005046732 ISSUE DATE: 20050526
APPLICATION: 2004 PP: 98 pp.
ASSIGNEE: (The United Sates of America as Represented by the Secretary of Health and Human Services, NIH USA
12. 47542 HIV-LS-325; SCIFINDER-HIV-6/20/2005
Preparation of alkylated pyrogallol calixarene type compounds as anti-viral compounds
Coveney, Donal and Costello, Benjamin
PATENT: US 20050113454 ISSUE DATE: 20050526
APPLICATION: 2003 PP: 13 pp.
ASSIGNEE: (Aids Care Pharma Limited, Ire.
13. 47543 HIV-LS-325; SCIFINDER-HIV-6/20/2005
A preparation of pyridinecarboxamide derivatives, useful for inhibiting HIV integrase
Kong, Laval Chan Chun, Zhang, Ming-Qiang, Halab, Liliane, Nguyen-Ba, Nghe, and Liu, Bingcan
PATENT: WO 2005042524 ISSUE DATE: 20050512
APPLICATION: 2004 PP: 139 pp.
ASSIGNEE: (Virochem Pharma Inc., Can.
14. 47544 HIV-LS-325; SCIFINDER-HIV-6/20/2005
Preparation of bipiperidinyl derivatives as inhibitors of CCR5 receptors
Miller, Michael W and Scott, Jack D
PATENT: WO 2005042517 ISSUE DATE: 20050512
APPLICATION: 2004 PP: 84 pp.
ASSIGNEE: (Schering Corporation, USA
15. 47545 HIV-LS-325; SCIFINDER-HIV-6/20/2005
Preparation of hydroxy pyridopyrrolopyrazine dione compounds useful as HIV integrase inhibitors
Wai, John S, Fisher, Thorsten E, Zhuang, Linghang, Staas, Donnette D, Lyle, Terry A, Kim, Boyoung, Embrey, Mark W, Wiscount, Catherine M, Tran, Lekhanh O, Egbertson, Melissa, and Savage, Kelly L
PATENT: WO 2005041664 ISSUE DATE: 20050512
APPLICATION: 2004 PP: 181 pp.
ASSIGNEE: (Merck & Co., Inc. USA
16. 47546 HIV-LS-325; SCIFINDER-HIV-6/20/2005
Identification of compounds that inhibit replication of human immunodeficiency virus
Balzarini, Jan Maria Rene, Vahlne, Anders, Hogberg, Marita, and Tong, Weimin
PATENT: US 2005096319 ISSUE DATE: 20050505
APPLICATION: 92 PP: 91 pp., Cont.-in-part of U.S. Ser. No. 783,053.
ASSIGNEE: (Belg.)
17. 47547 HIV-LS-325; SCIFINDER-HIV-6/20/2005
Potent 1,3,4-trisubstituted pyrrolidine CCR5 receptor antagonists: effects of fused heterocycles on antiviral activity and pharmacokinetic properties
Kim, Dooseop, Wang, Liping, Hale, Jeffrey J, Lynch, Christopher L, Budhu, Richard J, MacCoss, Malcolm, Mills, Sander G, Malkowitz, Lorraine, Gould, Sandra L, DeMartino, Julie A, Springer, Martin S, Hazuda, Daria, Miller, Michael, Kessler, Joseph, Hrin, Renee C, Carver, Gwen, Carella, Anthony, Henry, Karen, Lineberger, Janet, Schleif, William A, and Emini, Emilio A
Bioorganic & Medicinal Chemistry Letters 2005. 15(8): 2129-2134
18. 47548 HIV-LS-325; WOS-HIV-6/19/2005
Synthesis, antiviral activity, and mechanism of drug resistance of D- and L-2 ',3 '-didehydro-2 ',3 '-dideoxy-2 '-fluorocarbocyclic nucleosides
Wang, JN, Jin, YH, Rapp, KL, Bennett, M, Schinazi, RF, and Chu, CK
JOURNAL OF MEDICINAL CHEMISTRY 2005. 48(11): 3736-3748, 13
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000229443700011
19. 47549 HIV-LS-325; WOS-HIV-6/19/2005
Peptides derived from the reverse transcriptase of human immunodeficiency virus type 1 as novel inhibitors of the viral integrase
Gleenberg, IO, Avidan, O, Goldgur, Y, Herschhorn, A, and Hizi, A
JOURNAL OF BIOLOGICAL CHEMISTRY 2005. 280(23): 21987-21996, 10
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000229557900041
20. 47550 HIV-LS-325; SCIFINDER-HIV-6/20/2005
Synthesis of fluoroalkyl end-capped oligomers containing pendant phosphinic and phosphonic acid segments-application to novel fluorinated bioactive polymers possessing antibacterial and anti-hiv-1 activities
Sawada, Hideo, Kawai, Yoshikazu, Kawase, Tokuzo, Inaba Masashi Sugiya, Yoshiko, Sugiya, Masashi, Baba, Masanori, and Tomita, Toshio
International Journal of Polymeric Materials 2005. 54(4): 257-277
21. 47551 HIV-LS-325; WOS-HIV-6/19/2005
Discovery of natural product inhibitors of HIV-1 integrase at Merck
Singh, SB, Pelaez, F, Hazuda, DJ, and Lingham, RB
DRUGS OF THE FUTURE 2005. 30(3): 277-299, 23
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000229605600007
22. 47552 HIV-LS-325; WOS-HIV-6/19/2005
New drug targets for HIV
Bean, P
CLINICAL INFECTIOUS DISEASES 2005. 41: S96-S100, 5
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000229530700017
23. 47553 HIV-LS-325; WOS-HIV-6/26/2005
New inhibitors of the Tat-TAR RNA interaction found with a "fuzzy" pharmacophore model
Renner, S, Ludwig, V, Boden, O, Scheffer, U, Gobel, M, and Schneider, G
CHEMBIOCHEM 2005. 6(6): 1119-1125, 7
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000229730000025