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ONLINE DATABASE SEARCH - HIV-LS-334-MEMO

1. 48029 HIV-LS-334; PUBMED-HIV-10/31/2005

Discovery of 2,5-dimethoxy-substituted 5-bromopyridyl thiourea (PHI-236) as a potent broad-spectrum anti-human immunodeficiency virus microbicide

D'Cruz, OJ and Uckun, FM

Mol Hum Reprod 2005.


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16254003&dopt=abstract


2. 48030 HIV-LS-334; PUBMED-HIV-10/31/2005

Maraviroc (UK-427,857), a Potent, Orally Bioavailable, and Selective Small-Molecule Inhibitor of Chemokine Receptor CCR5 with Broad-Spectrum Anti-Human Immunodeficiency Virus Type 1 Activity

Dorr, P, Westby, M, Dobbs, S, Griffin, P, Irvine, B, Macartney, M, Mori, J, Rickett, G, Smith-Burchnell, C, Napier, C, Webster, R, Armour, D, Price, D, Stammen, B, Wood, A, and Perros, M

Antimicrob Agents Chemother 2005. 49(11): 4721-32


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16251317&dopt=abstract


3. 48031 HIV-LS-334; PUBMED-HIV-10/31/2005

TAK-652 Inhibits CCR5-Mediated Human Immunodeficiency Virus Type 1 Infection In Vitro and Has Favorable Pharmacokinetics in Humans

Baba, M, Takashima, K, Miyake, H, Kanzaki, N, Teshima, K, Wang, X, Shiraishi, M, and Iizawa, Y

Antimicrob Agents Chemother 2005. 49(11): 4584-91


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16251299&dopt=abstract


4. 48032 HIV-LS-334; PUBMED-HIV-10/31/2005

Anti-Human Immunodeficiency Virus Type 1 Activity of the Nonnucleoside Reverse Transcriptase Inhibitor GW678248 in Combination with Other Antiretrovirals against Clinical Isolate Viruses and In Vitro Selection for Resistance

Hazen, RJ, Harvey, RJ, St, Clair MH, Ferris, RG, Freeman, GA, Tidwell, JH, Schaller, LT, Cowan, JR, Short, SA, Romines, KR, Chan, JH, and Boone, LR

Antimicrob Agents Chemother 2005. 49(11): 4465-73


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16251284&dopt=abstract



5. 48033 HIV-LS-334; PUBMED-HIV-10/31/2005

Rapid access to 2'-branched-carbocyclic nucleosides and their 4'-epimers from 2-alkyl-cyclopentene-1-ones

Meillon, JC, Griffe, L, Storer, R, and Gosselin, G

Nucleosides Nucleotides Nucleic Acids 2005. 24(5-7): 695-9


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16248017&dopt=abstract


6. 48034 HIV-LS-334; PUBMED-HIV-10/31/2005

Novel phorbol esters exert dichotomous effects on inhibition of HIV-1 infection and activation of latent HIV-1 expression

Zhong, Y, Matsuya, Y, Nemoto, H, Mori, M, Saito, H, and Yamamoto, N

Antivir Chem Chemother 2005. 16(5): 303-13


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16245646&dopt=abstract


7. 48035 HIV-LS-334; PUBMED-HIV-10/31/2005

In vitro activity of SPD754, a new deoxycytidine nucleoside reverse transcriptase inhibitor (NRTI), against 215 HIV-1 isolates resistant to other NRTIs

Bethell, RC, Lie, YS, and Parkin, NT

Antivir Chem Chemother 2005. 16(5): 295-302


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16245645&dopt=abstract


8. 48036 HIV-LS-334; PUBMED-HIV-10/31/2005

Inhibition of human immunodeficiency virus-1 (HIV-1) by beta-chemokine analogues in mononuclear cells from HIV-1-infected patients with active tuberculosis

Toossi, Z, Mayanja-Kizza, H, Baseke, J, Peters, P, Wu, M, Abraha, A, Aung, H, Okwera, A, Hirsch, C, and Arts, E

Clin Exp Immunol 2005. 142(2): 327-32


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16232220&dopt=abstract


9. 48037 HIV-LS-334; PUBMED-HIV-10/31/2005

From nonpeptide toward noncarbon protease inhibitors: Metallacarboranes as specific and potent inhibitors of HIV protease

Cigler, P, Kozisek, M, Rezacova, P, Brynda, J, Otwinowski, Z, Pokorna, J, Plesek, J, Gruner, B, Doleckova-Maresova, L, Masa, M, Sedlacek, J, Bodem, J, Krausslich, HG, Kral, V, and Konvalinka, J

Proc Natl Acad Sci U S A 2005. 102(43): 15394-9


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16227435&dopt=abstract



10. 48038 HIV-LS-334; PUBMED-HIV-10/31/2005

Synthesis and biological evaluation of phosphonated carbocyclic 2'-oxa-3'-aza-nucleosides

Chiacchio, U, Iannazzo, D, Piperno, A, Romeo, R, Romeo, G, Rescifina, A, and Saglimbeni, M

Bioorg Med Chem 2005.


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16213735&dopt=abstract


11. 48039 HIV-LS-334; PUBMED-HIV-10/31/2005

Orally bioavailable highly potent HIV protease inhibitors against PI-resistant virus

Lu, Z, Bohn, J, Rano, T, Rutkowski, CA, Simcoe, AL, Olsen, DB, Schleif, WA, Carella, A, Gabryelski, L, Jin, L, Lin, JH, Emini, E, Chapman, K, and Tata, JR

Bioorg Med Chem Lett 2005. 15(23): 5311-4


HYPERLINK:

http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16203148&dopt=abstract


12. 48040 HIV-LS-334; WOS-HIV-10/23/2005

Design of HIV-1-PR inhibitors that do not create resistance: Blocking the folding of single monomers

Broglia, RA, Tiana, G, Sutto, L, Provasi, D, and Simona, F

PROTEIN SCIENCE 2005. 14(10): 2668-2681, 14


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232233400017


13. 48041 HIV-LS-334; WOS-HIV-10/23/2005

Advances in L-nucleosides as anti-HIV and anti-HBV agents

Dong, CH and Chang, JB

PROGRESS IN CHEMISTRY 2005. 17(5): 916-923, 8


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232294200021


14. 48042 HIV-LS-334; WOS-HIV-10/23/2005

Hiv-1 mutagenesis during antiretroviral therapy: Implications for successful drug treatment

Chen, RX, Quinones-Mateu, ME, and Mansky, LM

FRONTIERS IN BIOSCIENCE 2005. 10: 743-750, 8


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232319300069


15. 48043 HIV-LS-334; WOS-HIV-10/23/2005

HIV-1 gp120 V3 loop for structure-based drug design

Sirois, S, Sing, T, and Chou, KC

CURRENT PROTEIN & PEPTIDE SCIENCE 2005. 6(5): 413-422, 10


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232388000003


16. 48044 HIV-LS-334; WOS-HIV-10/23/2005

Synthesis and antiviral evaluation of novel 6 '(alpha)-methyl-branched Carbovir analogues

Kim, JW and Hong, JH

ARCHIV DER PHARMAZIE 2005. 338(9): 399-404, 6


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232313800001


17. 48045 HIV-LS-334; WOS-HIV-10/23/2005

Sophorolipids, microbial glycolipids with anti-human immunodeficiency virus and sperm-immobilizing activities

Shah, V, Doncel, GF, Seyoum, T, Eaton, KM, Zalenskaya, I, Hagver, R, Azim, A, and Gross, R

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY 2005. 49(10): 4093-4100, 8


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232244700015


18. 48046 HIV-LS-334; WOS-HIV-10/23/2005

Newly designed six-membered azasugar nucleotide-containing phosphorothioate oligonucleotides as potent human immunodeficiency virus type 1 inhibitors

Lee, DS, Jung, KE, Yoon, CH, Lim, H, and Bae, YS

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY 2005. 49(10): 4110-4120, 11


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232244700017


19. 48047 HIV-LS-334; WOS-HIV-10/23/2005

Pharmacokinetics of sifuvirtide, a novel anti-HIV-1 peptide, in monkeys and its inhibitory concentration in vitro

Dai, SJ, Dou, GF, Qian, XH, Song, HF, Tang, ZM, Liu, DS, Liu, XW, Yang, LM, Zheng, YT, and Liang, Q

ACTA PHARMACOLOGICA SINICA 2005. 26(10): 1274-1280, 7


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232346000018


20. 48048 HIV-LS-334; WOS-HIV-10/30/2005

Efficient and general method for the synthesis of benzopyrans by ethylenediamine diacetate-catalyzed reactions of resorcinols with alpha,beta-unsaturated aldehydes. One step synthesis of biologically active (+/-)-confluentin and (+/-)-daurichromenic acid

Lee, YR, Choi, JH, and Yoon, SH

TETRAHEDRON LETTERS 2005. 46(44): 7539-7543, 5


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232572200016


21. 48049 HIV-LS-334; WOS-HIV-10/30/2005

Antiviral potential of a new generation of acyclic nucleoside phosphonates, the 6-[2-(phosphonomethoxy)alkoxy]-2,4-diaminopyrimidines

De Clercq, E, Andrei, G, Balzarini, J, Leyssen, P, Naesens, L, Neyts, J, Pannecouque, C, Snoeck, R, Ying, C, Hockova, D, and Holy, A

NUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS 2005. 24(5-7): 331-341, 11


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232473500003


22. 48050 HIV-LS-334; WOS-HIV-10/30/2005

A new approach to the synthesis of 4 '-carbon-substituted nucleosides: Development of a highly active anti-HIV agent 2 ', 3 '-didehydro-3 '-deoxy-4 '-ethynylthymidine

Haraguchi, K, Takeda, S, Sumino, M, Tanaka, H, Dutschman, GE, Cheng, YC, Nitanda, T, and Baba, M

NUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS 2005. 24(5-7): 343-347, 5


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232473500004



23. 48051 HIV-LS-334; WOS-HIV-10/30/2005

Synthesis and study of conformationally restricted 3 '-deoxy-3 ',4 '-exo-methylene nucleoside analogues

Gagneron, J, Gosselin, G, and Mathe, C

NUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS 2005. 24(5-7): 383-385, 3


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232473500010


24. 48052 HIV-LS-334; WOS-HIV-10/30/2005

Design and synthesis of specific inhibitors of the 3 '-processing step of HIV-1 integrase

Chi, GC, Seo, BI, and Nair, V

NUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS 2005. 24(5-7): 481-484, 4


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232473500030


25. 48053 HIV-LS-334; WOS-HIV-10/30/2005

HIV-1 inactivation by nucleic acid aptamers

Held, DM, Kissel, JD, Patterson, JT, Nickens, DG, and Burke, DH

FRONTIERS IN BIOSCIENCE 2006. 11: 89-112, 24


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232528000008


26. 48054 HIV-LS-334; WOS-HIV-10/30/2005

Anti-HIV agents targeting the interaction of gp120 with the cellular CD4 receptor

Vermeire, K and Schols, D

EXPERT OPINION ON INVESTIGATIONAL DRUGS 2005. 14(10): 1199-1212, 14


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232509700002


27. 48055 HIV-LS-334; WOS-HIV-10/30/2005

Development of anti-HIV agents targeting dynamic supramolecular mechanism: Entry and fusion inhibitors based on CXCR4/CCR5 antagonists and gp41-C34-remodeling peptides

Tamamura, H, Otaka, A, and Fujii, N

CURRENT HIV RESEARCH 2005. 3(4): 289-301, 13


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232477900001


28. 48056 HIV-LS-334; WOS-HIV-10/30/2005

Neamine dimers targeting the HIV-1 TAR RNA

Riguet, E, Desire, J, Boden, O, Ludwig, V, Gobel, M, Bailly, C, and Decout, JL

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 2005. 15(21): 4651-4655, 5


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232465900001


29. 48057 HIV-LS-334; WOS-HIV-10/30/2005

In vitro generation of HIV type 1 subtype C isolates resistant to enfuvirtide

Cilliers, T, Moore, P, Coetzer, M, and Morris, L

AIDS RESEARCH AND HUMAN RETROVIRUSES 2005. 21(9): 776-783, 8


HYPERLINK:

http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000232528300005


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