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1. 48543 HIV-LS-343; PUBMED-HIV-3/6/2006

Microwave-Accelerated Synthesis of P1'-Extended HIV-1 Protease Inhibitors Encompassing a Tertiary Alcohol in the Transition-State Mimicking Scaffold

Ekegren, JK, Ginman, N, Johansson, A, Wallberg, H, Larhed, M, Samuelsson, B, Unge, T, and Hallberg, A

J Med Chem 2006. 49(5): 1828-1832


2. 48544 HIV-LS-343; PUBMED-HIV-3/6/2006

Synthesis and Anti-HIV Activity of d- and l-Thietanose Nucleosides

Choo, H, Chen, X, Yadav, V, Wang, J, Schinazi, RF, and Chu, CK

J Med Chem 2006. 49(5): 1635-47


3. 48545 HIV-LS-343; PUBMED-HIV-3/6/2006

Novel HIV-1 Integrase Inhibitors Derived from Quinolone Antibiotics

Sato, M, Motomura, T, Aramaki, H, Matsuda, T, Yamashita, M, Ito, Y, Kawakami, H, Matsuzaki, Y, Watanabe, W, Yamataka, K, Ikeda, S, Kodama, E, Matsuoka, M, and Shinkai, H

J Med Chem 2006. 49(5): 1506-8


4. 48546 HIV-LS-343; PUBMED-HIV-3/6/2006

Synthesis, antiviral activity, and pharmacokinetic evaluation of P3 pyridylmethyl analogs of oximinoarylsulfonyl HIV-1 protease inhibitors

Randolph, JT, Huang, PP, Flosi, WJ, Degoey, D, Klein, LL, Yeung, CM, Flentge, C, Sun, M, Zhao, C, Dekhtyar, T, Mo, H, Colletti, L, Kati, W, Marsh, KC, Molla, A, and Kempf, DJ

Bioorg Med Chem 2006.


5. 48547 HIV-LS-343; PUBMED-HIV-3/6/2006

Tetrazole thioacetanilides: Potent non-nucleoside inhibitors of WT HIV reverse transcriptase and its K103N mutant

Muraglia, E, Kinzel, OD, Laufer, R, Miller, MD, Moyer, G, Munshi, V, Orvieto, F, Palumbi, MC, Pescatore, G, Rowley, M, Williams, PD, and Summa, V

Bioorg Med Chem Lett 2006.


6. 48548 HIV-LS-343; PUBMED-HIV-3/6/2006

Inhibition of human immunodeficiency virus type 1 replication with artificial transcription factors targeting the highly conserved primer-binding site

Eberhardy, SR, Goncalves, J, Coelho, S, Segal, DJ, Berkhout, B, and Barbas, CF 3rd

J Virol 2006. 80(6): 2873-83


7. 48549 HIV-LS-343; PUBMED-HIV-3/6/2006

Cyclophilin A and TRIM5{alpha} Independently Regulate Human Immunodeficiency Virus Type 1 Infectivity in Human Cells

Sokolskaja, E, Berthoux, L, and Luban, J

J Virol 2006. 80(6): 2855-62


8. 48550 HIV-LS-343; SCIFINDER-HIV-2/27/2006

C-Glycoside analogues of b-galactosylceramide with a simple ceramide substitute: Synthesis and binding to HIV-1 gp120

Augustin, Line A, Fantini, Jacques, and Mootoo, David R

Bioorganic & Medicinal Chemistry 2006. 14(4): 1182-1188

9. 48551 HIV-LS-343; PUBMED-HIV-3/6/2006

Interaction of small molecule inhibitors of HIV-1 entry with CCR5

Seibert, C, Ying, W, Gavrilov, S, Tsamis, F, Kuhmann, SE, Palani, A, Tagat, JR, Clader, JW, McCombie, SW, Baroudy, BM, Smith, SO, Dragic, T, Moore, JP, and Sakmar, TP

Virology 2006.


10. 48552 HIV-LS-343; SCIFINDER-HIV-2/27/2006

QSAR studies on the use of 5,6-dihydro-2-pyrones as HIV-1 protease inhibitors

Agrawal, Vijay K, Singh, Jyoti, Mishra, Krishna C, Khadikar, Padmakar V, and Jaliwala, Yusuf Ali

ARKIVOC (Gainesville, FL, United States) 2006.(2): 162-177

11. 48553 HIV-LS-343; SCIFINDER-HIV-2/27/2006

Preparation of amino acid-containing nucleotides as prodrugs and antiviral agents

Boojamra, Constantine G, Lin, Kuei-Ying, Mackman, Richard L, Markevitch, David Y, Petrakovsky, Oleg V, Ray, Adrian S, and Zhang, Lijun

PATENT: WO 2006015261 ISSUE DATE: 20060209

APPLICATION: 2005 PP: 173 pp.

ASSIGNEE: (Gilead Sciences, Inc. USA

12. 48554 HIV-LS-343; PUBMED-HIV-3/6/2006

Inhibition of human immunodeficiency virus type 1 infection in macrophages by an alpha-v integrin blocking antibody

Bosch, B, Clotet-Codina, I, Blanco, J, Pauls, E, Coma, G, Cedeno, S, Mitjans, F, Llano, A, Bofill, M, Clotet, B, Piulats, J, and Este, JA

Antiviral Res 2006. 69(3): 173-80


13. 48555 HIV-LS-343; SCIFINDER-HIV-2/27/2006

Induction of APOBEC3 family proteins, a defensive maneuver underlying interferon-induced anti-HIV-1 activity

Peng, Gang, Lei, Ke Jian, Jin, Wenwen, Greenwell-Wild, Teresa, and Wahl, Sharon M

Journal of Experimental Medicine 2006. 203(1): 41-46

14. 48556 HIV-LS-343; PUBMED-HIV-3/6/2006

Susceptibility to protease inhibitors in HIV-2 primary isolates from patients failing antiretroviral therapy

Rodes, B, Sheldon, J, Toro, C, Jimenez, V, Alvarez, MA, and Soriano, V

J Antimicrob Chemother 2006.


15. 48557 HIV-LS-343; PUBMED-HIV-3/6/2006

Mining the NCI antiviral compounds for HIV-1 integrase inhibitors

Deng, J, Kelley, JA, Barchi, JJ, Sanchez, T, Dayam, R, Pommier, Y, and Neamati, N

Bioorg Med Chem 2006.


16. 48558 HIV-LS-343; SCIFINDER-HIV-2/27/2006

Herbal extract with antiviral properties

Abdullahi, Jacob J

PATENT: US 2006024386 ISSUE DATE: 20060202

APPLICATION: 2005-58730

ASSIGNEE: (Nigeria)

17. 48559 HIV-LS-343; WOS-HIV-2/26/2006

Identification of sanguinarine as a novel HIV protease inhibitor from high-throughput screening of 2,000 drugs and natural products with a cell-based assay

Cheng, TJ, Goodsell, DS, and Kan, CC

LETTERS IN DRUG DESIGN & DISCOVERY 2005. 2(5): 364-371, 8


18. 48560 HIV-LS-343; WOS-HIV-2/26/2006

Structure based design of inhibitors of aspartic protease of HIV-1

Frecer, V, Jedinak, A, Tossi, A, Berti, F, Benedetti, F, Romeo, D, and Miertus, S

LETTERS IN DRUG DESIGN & DISCOVERY 2005. 2(8): 638-646, 9


19. 48561 HIV-LS-343; WOS-HIV-2/26/2006

p27(SJ), a novel protein in St John's Wort, that suppresses expression of HIV-1 genome

Darbinian-Sarkissian, N, Darbinyan, A, Otte, J, Radhakrishnan, S, Sawaya, BE, Arzumanyan, A, Chipitsyna, G, Popov, Y, Rappaport, J, Amini, S, and Khalili, K

GENE THERAPY 2006. 13(4): 288-295, 8


20. 48562 HIV-LS-343; WOS-HIV-3/5/2006

How can (-)-epigallocatechin gallate from green tea prevent HIV-1 infection? Mechanistic insights from computational modeling and the implication for rational design of anti-HIV-1 entry inhibitors

Hamza, A and Zhan, CG

JOURNAL OF PHYSICAL CHEMISTRY B 2006. 110(6): 2910-2917, 8


21. 48563 HIV-LS-343; WOS-HIV-3/5/2006

Synthesis and antiviral evaluation of carbocyclic 3 '-azidothymidine (AZT) analogues and their cycloSal-phosphate triesters

Ludek, OR, Balzarini, J, and Meier, C



22. 48564 HIV-LS-343; WOS-HIV-3/5/2006

Anti-HIV I/II activity and molecular cloning of a novel mannose/sialic acid-binding lectin from rhizome of Polygonatum cyrtonema Hua

An, J, Liu, JZ, Wu, CF, Li, J, Dai, L, Van Damme, E, Balzarini, J, De Clercq, E, Chen, F, and Bao, JK



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