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1. 58734 HIV-LS-355; PUBMED-HIV-8/21/2006

Design, Synthesis, Biological Evaluation, and Molecular Modeling Studies of TIBO-Like Cyclic Sulfones as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors

Di Santo, R, Costi, R, Artico, M, Ragno, R, Lavecchia, A, Novellino, E, Gavuzzo, E, La Torre, F, Cirilli, R, Cancio, R, and Maga, G

ChemMedChem 2006. 1(1): 82-95


2. 58735 HIV-LS-355; SCIFINDER-HIV-8/14/2006

Nucleoside analogues with 6-membered carbon ring structure, synthetic method and use in antivirus thereof

Lou, Hongxiang, Zhan, Tianrong, Ma, Yudao, and Fan, Peihong

PATENT: CN 1803819 ISSUE DATE: 20060719

APPLICATION: 1004-2184 PP: 18 pp.

ASSIGNEE: (Shandong University, Peop. Rep. China

3. 58736 HIV-LS-355; PUBMED-HIV-8/21/2006

Design and Discovery of a Novel Dipeptidyl-peptidase IV (CD26)-Based Prodrug Approach

Garcia-Aparicio, C, Bonache, MC, De, Meester I, San-Felix, A, Balzarini, J, Camarasa, MJ, and Velazquez, S

J Med Chem 2006. 49(17): 5339-5351


4. 58737 HIV-LS-355; SCIFINDER-HIV-8/14/2006

Preparation of N-[(imidazo[1,2-a]pyridin-2-yl)methyl]-3,4-dihydro-2H-pyrano[3,2-b]pyridin-4-amines that bind to chemokine receptors for use against HIV and other disorders

Gudmundsson, Kristjan

PATENT: WO 2006076131 ISSUE DATE: 20060720

APPLICATION: 2005 PP: 63 pp.

ASSIGNEE: (Smithkline Beecham Corporation, USA

5. 58738 HIV-LS-355; PUBMED-HIV-8/21/2006

Structure-Based Design of Novel HIV-1 Protease Inhibitors To Combat Drug Resistance

Ghosh, AK, Sridhar, PR, Leshchenko, S, Hussain, AK, Li, J, Kovalevsky, AY, Walters, DE, Wedekind, JE, Grum-Tokars, V, Das, D, Koh, Y, Maeda, K, Gatanaga, H, Weber, IT, and Mitsuya, H

J Med Chem 2006. 49(17): 5252-5261


6. 58739 HIV-LS-355; SCIFINDER-HIV-8/14/2006

Preparation of 2-oxo-3-cyano-1,6a-diaza-tetrahydro-fluoranthenes as anti-HIV agents

Kesteleyn, Bart Rudolf Romanie, Raboisson, Pierre Jean-Marie, Van De Vreken, Wim, and Canard, Maxime Francis Jean-Marie Ghislain

PATENT: WO 2006072636 ISSUE DATE: 20060713

APPLICATION: 2006 PP: 42 pp.

ASSIGNEE: (Tibotec Pharmaceuticals Ltd., Ire.

7. 58740 HIV-LS-355; PUBMED-HIV-8/21/2006

Structure-activity relationships in platelet-activating factor. Part 14: Synthesis and biological evaluation of piperazine derivatives with dual anti-PAF and anti-HIV-1 activity

Sallem, W, Serradji, N, Dereuddre-Bosquet, N, Dive, G, Clayette, P, and Heymans, F

Bioorg Med Chem 2006.


8. 58741 HIV-LS-355; PUBMED-HIV-8/21/2006

Synthesis and anti-HIV-1 activity of a novel series of 1,4,2-benzodithiazine-dioxides

Brzozowski, Z, Saczewski, F, and Neamati, N

Bioorg Med Chem Lett 2006.


9. 58742 HIV-LS-355; PUBMED-HIV-8/21/2006

Synthesis and HIV-integrase strand transfer inhibition activity of 7-hydroxy[1,3]thiazolo[5,4-b]pyridin-5(4H)-ones

Boros, EE, Johns, BA, Garvey, EP, Koble, CS, and Miller, WH

Bioorg Med Chem Lett 2006.


10. 58743 HIV-LS-355; SCIFINDER-HIV-8/14/2006

2',3'-Dideoxy-3'-hydroxymethylcytosine or a prodrug for the treatment of HIV

Xhou, Xiao-Xiong and Zhang, Hong

PATENT: WO 2006070004 ISSUE DATE: 20060706

APPLICATION: 2005 PP: 73 pp.

ASSIGNEE: (Medivir AB, Swed.

11. 58744 HIV-LS-355; SCIFINDER-HIV-8/14/2006

Diketo acids derivatives as integrase inhibitors: the war against the acquired immunodeficiency syndrome

Henao-Mejia, Jorge, Goez, Yenny, Patino, Pablo, and Rugeles, Maria T

Recent Patents on Anti-Infective Drug Discovery 2006. 1(2 ): 255-265

12. 58745 HIV-LS-355; PUBMED-HIV-8/21/2006

New, potent P1/P2-morpholinone-based HIV-protease inhibitors

Kazmierski, WM, Furfine, E, Spaltenstein, A, and Wright, LL

Bioorg Med Chem Lett 2006.


13. 58746 HIV-LS-355; PUBMED-HIV-8/21/2006

Simple synthesis of novel acyclic (e)-bromovinyl nucleosides as potential antiviral agents

Kim, JW and Hong, JH

Nucleosides Nucleotides Nucleic Acids 2006. 25(8): 879-87


14. 58747 HIV-LS-355; SCIFINDER-HIV-8/14/2006

Preparation of aminium salts of 1,2,3-triazoles as prodrugs of drugs including antiviral agents

Kadow, John F and Regueiro-Ren, Alicia

PATENT: US 2006142298 ISSUE DATE: 20060629

APPLICATION: 2005-38902 PP: 19 pp.


15. 58748 HIV-LS-355; SCIFINDER-HIV-8/14/2006

8-Azabicyclo[3.2.1]octane derivatives with an activity on chemokine CCR5 receptors and their preparation, pharmaceutical compositions and use for treatment of inflammatory diseases and infection caused by HIV and genetically related retroviruses

Pryde, David Cameron and Stupple, Paul Anthony

PATENT: WO 2006067584 ISSUE DATE: 20060629

APPLICATION: 2005 PP: 67 pp.

ASSIGNEE: (Pfizer Limited, UK

16. 58749 HIV-LS-355; PUBMED-HIV-8/21/2006

Towards discovering dual functional inhibitors against both wild type and K103N mutant HIV-1 reverse transcriptases: molecular docking and QSAR studies on 4,1-benzoxazepinone analogues

Zhang, Z, Zheng, M, Du, L, Shen, J, Luo, X, Zhu, W, and Jiang, H

J Comput Aided Mol Des 2006.


17. 58750 HIV-LS-355; PUBMED-HIV-8/21/2006

Structure-activity relationships in platelet-activating factor. Part 13: Synthesis and biological evaluation of piperazine derivatives with dual anti-PAF and anti-HIV-1 or pure antiretroviral activity

Serradji, N, Bensaid, O, Martin, M, Sallem, W, Dereuddre-Bosquet, N, Benmehdi, H, Redeuilh, C, Lamouri, A, Dive, G, Clayette, P, and Heymans, F

Bioorg Med Chem 2006.


18. 58751 HIV-LS-355; SCIFINDER-HIV-8/14/2006

Application of 2-(n-methyl-guanidino)-ethanesulfonic acid in anti-hiv virus

Jin, Yan, Zheng, Yongtang, Wang, Jianhua, and Zhang, Wei

PATENT: CN 1785168 ISSUE DATE: 20060614

APPLICATION: 1008-2873 PP: 5 pp.

ASSIGNEE: (Dalian Institute of Chemical Physics, Chinese Academy of Sciences Peop. Rep. China and Kunming Institute of Zoology, Chinese Academy of Sciences

19. 58752 HIV-LS-355; PUBMED-HIV-8/21/2006

Structure-activity relationship study of flavone compounds with anti-HIV-1 integrase activity: A density functional theory study

Lameira, J, Medeiros, IG, Reis, M, Santos, AS, and Alves, CN

Bioorg Med Chem 2006.


20. 58753 HIV-LS-355; SCIFINDER-HIV-8/14/2006

Modified azidothymidine 5'-phosphonate for potential antiviral preparations

Kukhanova, Marina Konstantinovna, Khankajinskaya, Anastasiya Lvovna, Yasko, Maxim Vladimirovich, Shirokova, Elena Anatolievna, Shipitsyn, Alexander Valerievich, and Pokrovsky, Andrey Georgievich

PATENT: WO 2006062434 ISSUE DATE: 20060615

APPLICATION: 2005 PP: 19 pp.

ASSIGNEE: (Russia)

21. 58754 HIV-LS-355; PUBMED-HIV-8/21/2006

Antiviral activity of Arthrospira-derived spirulan-like substances

Rechter, S, Konig, T, Auerochs, S, Thulke, S, Walter, H, Dornenburg, H, Walter, C, and Marschall, M

Antiviral Res 2006.


22. 58755 HIV-LS-355; PUBMED-HIV-8/21/2006

Inhibition of HIV-1 replication by amphotericin B methyl ester: selection for resistant variants

Waheed, AA, Ablan, SD, Mankowski, MK, Cummins, JE, Ptak, RG, Schaffner, CP, and Freed, EO

J Biol Chem 2006.


23. 58756 HIV-LS-355; PUBMED-HIV-8/21/2006

Inhibition of HIV-1 integrase activity by synthetic peptides derived from the HIV-1 HXB2 Pol region of the viral genome

Zawahir, Z and Neamati, N

Bioorg Med Chem Lett 2006.


24. 58757 HIV-LS-355; SCIFINDER-HIV-8/14/2006

Synthesis and antiviral evaluation of novel pyrimidine thioapionucleosides

Lee, Rae Sang, Hong, Joon Hee, and Ko, Ok Hyun

Yakhak Hoechi 2006. 50(2): 65-69

25. 58758 HIV-LS-355; PUBMED-HIV-8/21/2006

Contribution of Vpu, Env, and Nef to CD4 down-modulation and resistance of human immunodeficiency virus type 1-infected T cells to superinfection

Wildum, S, Schindler, M, Munch, J, and Kirchhoff, F

J Virol 2006. 80(16): 8047-59


26. 58759 HIV-LS-355; SCIFINDER-HIV-8/14/2006

Preparation of HIV inhibiting bicyclic pyrimidine derivatives

Janssen, Paul Adriaan Jan, Guillemont, Jerome Emile Georges, Paugam, Mikaeel, Delest, Bruno Francois Marie, Heeres, Jan, and Lewi, Paulus Joannes

PATENT: WO 2006045828 ISSUE DATE: 20060504

APPLICATION: 2005 PP: 82 pp.

ASSIGNEE: (Tibotec Pharmaceuticals Ltd., Ire. and Arts, Frank Xavier Jozef Herwig

27. 58760 HIV-LS-355; WOS-HIV-8/20/2006

cis- and trans-decahydro-1,6-naphthyridines. Stereoselective synthesis and stereochemistry

Esipova, TV, Borisenko, AA, and Grishina, GV



28. 58761 HIV-LS-355; WOS-HIV-8/20/2006

Chemokine receptor CCR-5 inhibitors produced by Chaetomium globosum

Yang, SW, Mierzwa, R, Terracciano, J, Patel, M, Gullo, V, Wagner, N, Baroudy, B, Puar, M, Chan, TM, McPhail, AT, and Chu, M

JOURNAL OF NATURAL PRODUCTS 2006. 69(7): 1025-1028, 4


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