ONLINE DATABASE SEARCH - HIV-LS-355-MEMO
1. 58734 HIV-LS-355; PUBMED-HIV-8/21/2006
Design, Synthesis, Biological Evaluation, and Molecular Modeling Studies of TIBO-Like Cyclic Sulfones as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors
Di Santo, R, Costi, R, Artico, M, Ragno, R, Lavecchia, A, Novellino, E, Gavuzzo, E, La Torre, F, Cirilli, R, Cancio, R, and Maga, G
ChemMedChem 2006. 1(1): 82-95
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16892340&dopt=abstract
2. 58735 HIV-LS-355; SCIFINDER-HIV-8/14/2006
Nucleoside analogues with 6-membered carbon ring structure, synthetic method and use in antivirus thereof
Lou, Hongxiang, Zhan, Tianrong, Ma, Yudao, and Fan, Peihong
PATENT: CN 1803819 ISSUE DATE: 20060719
APPLICATION: 1004-2184 PP: 18 pp.
ASSIGNEE: (Shandong University, Peop. Rep. China
3. 58736 HIV-LS-355; PUBMED-HIV-8/21/2006
Design and Discovery of a Novel Dipeptidyl-peptidase IV (CD26)-Based Prodrug Approach
Garcia-Aparicio, C, Bonache, MC, De, Meester I, San-Felix, A, Balzarini, J, Camarasa, MJ, and Velazquez, S
J Med Chem 2006. 49(17): 5339-5351
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16913724&dopt=abstract
4. 58737 HIV-LS-355; SCIFINDER-HIV-8/14/2006
Preparation of N-[(imidazo[1,2-a]pyridin-2-yl)methyl]-3,4-dihydro-2H-pyrano[3,2-b]pyridin-4-amines that bind to chemokine receptors for use against HIV and other disorders
Gudmundsson, Kristjan
PATENT: WO 2006076131 ISSUE DATE: 20060720
APPLICATION: 2005 PP: 63 pp.
ASSIGNEE: (Smithkline Beecham Corporation, USA
5. 58738 HIV-LS-355; PUBMED-HIV-8/21/2006
Structure-Based Design of Novel HIV-1 Protease Inhibitors To Combat Drug Resistance
Ghosh, AK, Sridhar, PR, Leshchenko, S, Hussain, AK, Li, J, Kovalevsky, AY, Walters, DE, Wedekind, JE, Grum-Tokars, V, Das, D, Koh, Y, Maeda, K, Gatanaga, H, Weber, IT, and Mitsuya, H
J Med Chem 2006. 49(17): 5252-5261
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16913714&dopt=abstract
6. 58739 HIV-LS-355; SCIFINDER-HIV-8/14/2006
Preparation of 2-oxo-3-cyano-1,6a-diaza-tetrahydro-fluoranthenes as anti-HIV agents
Kesteleyn, Bart Rudolf Romanie, Raboisson, Pierre Jean-Marie, Van De Vreken, Wim, and Canard, Maxime Francis Jean-Marie Ghislain
PATENT: WO 2006072636 ISSUE DATE: 20060713
APPLICATION: 2006 PP: 42 pp.
ASSIGNEE: (Tibotec Pharmaceuticals Ltd., Ire.
7. 58740 HIV-LS-355; PUBMED-HIV-8/21/2006
Structure-activity relationships in platelet-activating factor. Part 14: Synthesis and biological evaluation of piperazine derivatives with dual anti-PAF and anti-HIV-1 activity
Sallem, W, Serradji, N, Dereuddre-Bosquet, N, Dive, G, Clayette, P, and Heymans, F
Bioorg Med Chem 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16908170&dopt=abstract
8. 58741 HIV-LS-355; PUBMED-HIV-8/21/2006
Synthesis and anti-HIV-1 activity of a novel series of 1,4,2-benzodithiazine-dioxides
Brzozowski, Z, Saczewski, F, and Neamati, N
Bioorg Med Chem Lett 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16908143&dopt=abstract
9. 58742 HIV-LS-355; PUBMED-HIV-8/21/2006
Synthesis and HIV-integrase strand transfer inhibition activity of 7-hydroxy[1,3]thiazolo[5,4-b]pyridin-5(4H)-ones
Boros, EE, Johns, BA, Garvey, EP, Koble, CS, and Miller, WH
Bioorg Med Chem Lett 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16908139&dopt=abstract
10. 58743 HIV-LS-355; SCIFINDER-HIV-8/14/2006
2',3'-Dideoxy-3'-hydroxymethylcytosine or a prodrug for the treatment of HIV
Xhou, Xiao-Xiong and Zhang, Hong
PATENT: WO 2006070004 ISSUE DATE: 20060706
APPLICATION: 2005 PP: 73 pp.
ASSIGNEE: (Medivir AB, Swed.
11. 58744 HIV-LS-355; SCIFINDER-HIV-8/14/2006
Diketo acids derivatives as integrase inhibitors: the war against the acquired immunodeficiency syndrome
Henao-Mejia, Jorge, Goez, Yenny, Patino, Pablo, and Rugeles, Maria T
Recent Patents on Anti-Infective Drug Discovery 2006. 1(2 ): 255-265
12. 58745 HIV-LS-355; PUBMED-HIV-8/21/2006
New, potent P1/P2-morpholinone-based HIV-protease inhibitors
Kazmierski, WM, Furfine, E, Spaltenstein, A, and Wright, LL
Bioorg Med Chem Lett 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16904316&dopt=abstract
13. 58746 HIV-LS-355; PUBMED-HIV-8/21/2006
Simple synthesis of novel acyclic (e)-bromovinyl nucleosides as potential antiviral agents
Kim, JW and Hong, JH
Nucleosides Nucleotides Nucleic Acids 2006. 25(8): 879-87
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16901820&dopt=abstract
14. 58747 HIV-LS-355; SCIFINDER-HIV-8/14/2006
Preparation of aminium salts of 1,2,3-triazoles as prodrugs of drugs including antiviral agents
Kadow, John F and Regueiro-Ren, Alicia
PATENT: US 2006142298 ISSUE DATE: 20060629
APPLICATION: 2005-38902 PP: 19 pp.
ASSIGNEE: (USA)
15. 58748 HIV-LS-355; SCIFINDER-HIV-8/14/2006
8-Azabicyclo[3.2.1]octane derivatives with an activity on chemokine CCR5 receptors and their preparation, pharmaceutical compositions and use for treatment of inflammatory diseases and infection caused by HIV and genetically related retroviruses
Pryde, David Cameron and Stupple, Paul Anthony
PATENT: WO 2006067584 ISSUE DATE: 20060629
APPLICATION: 2005 PP: 67 pp.
ASSIGNEE: (Pfizer Limited, UK
16. 58749 HIV-LS-355; PUBMED-HIV-8/21/2006
Towards discovering dual functional inhibitors against both wild type and K103N mutant HIV-1 reverse transcriptases: molecular docking and QSAR studies on 4,1-benzoxazepinone analogues
Zhang, Z, Zheng, M, Du, L, Shen, J, Luo, X, Zhu, W, and Jiang, H
J Comput Aided Mol Des 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16897578&dopt=abstract
17. 58750 HIV-LS-355; PUBMED-HIV-8/21/2006
Structure-activity relationships in platelet-activating factor. Part 13: Synthesis and biological evaluation of piperazine derivatives with dual anti-PAF and anti-HIV-1 or pure antiretroviral activity
Serradji, N, Bensaid, O, Martin, M, Sallem, W, Dereuddre-Bosquet, N, Benmehdi, H, Redeuilh, C, Lamouri, A, Dive, G, Clayette, P, and Heymans, F
Bioorg Med Chem 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16893650&dopt=abstract
18. 58751 HIV-LS-355; SCIFINDER-HIV-8/14/2006
Application of 2-(n-methyl-guanidino)-ethanesulfonic acid in anti-hiv virus
Jin, Yan, Zheng, Yongtang, Wang, Jianhua, and Zhang, Wei
PATENT: CN 1785168 ISSUE DATE: 20060614
APPLICATION: 1008-2873 PP: 5 pp.
ASSIGNEE: (Dalian Institute of Chemical Physics, Chinese Academy of Sciences Peop. Rep. China and Kunming Institute of Zoology, Chinese Academy of Sciences
19. 58752 HIV-LS-355; PUBMED-HIV-8/21/2006
Structure-activity relationship study of flavone compounds with anti-HIV-1 integrase activity: A density functional theory study
Lameira, J, Medeiros, IG, Reis, M, Santos, AS, and Alves, CN
Bioorg Med Chem 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16890444&dopt=abstract
20. 58753 HIV-LS-355; SCIFINDER-HIV-8/14/2006
Modified azidothymidine 5'-phosphonate for potential antiviral preparations
Kukhanova, Marina Konstantinovna, Khankajinskaya, Anastasiya Lvovna, Yasko, Maxim Vladimirovich, Shirokova, Elena Anatolievna, Shipitsyn, Alexander Valerievich, and Pokrovsky, Andrey Georgievich
PATENT: WO 2006062434 ISSUE DATE: 20060615
APPLICATION: 2005 PP: 19 pp.
ASSIGNEE: (Russia)
21. 58754 HIV-LS-355; PUBMED-HIV-8/21/2006
Antiviral activity of Arthrospira-derived spirulan-like substances
Rechter, S, Konig, T, Auerochs, S, Thulke, S, Walter, H, Dornenburg, H, Walter, C, and Marschall, M
Antiviral Res 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16884788&dopt=abstract
22. 58755 HIV-LS-355; PUBMED-HIV-8/21/2006
Inhibition of HIV-1 replication by amphotericin B methyl ester: selection for resistant variants
Waheed, AA, Ablan, SD, Mankowski, MK, Cummins, JE, Ptak, RG, Schaffner, CP, and Freed, EO
J Biol Chem 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16882663&dopt=abstract
23. 58756 HIV-LS-355; PUBMED-HIV-8/21/2006
Inhibition of HIV-1 integrase activity by synthetic peptides derived from the HIV-1 HXB2 Pol region of the viral genome
Zawahir, Z and Neamati, N
Bioorg Med Chem Lett 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16879966&dopt=abstract
24. 58757 HIV-LS-355; SCIFINDER-HIV-8/14/2006
Synthesis and antiviral evaluation of novel pyrimidine thioapionucleosides
Lee, Rae Sang, Hong, Joon Hee, and Ko, Ok Hyun
Yakhak Hoechi 2006. 50(2): 65-69
25. 58758 HIV-LS-355; PUBMED-HIV-8/21/2006
Contribution of Vpu, Env, and Nef to CD4 down-modulation and resistance of human immunodeficiency virus type 1-infected T cells to superinfection
Wildum, S, Schindler, M, Munch, J, and Kirchhoff, F
J Virol 2006. 80(16): 8047-59
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16873261&dopt=abstract
26. 58759 HIV-LS-355; SCIFINDER-HIV-8/14/2006
Preparation of HIV inhibiting bicyclic pyrimidine derivatives
Janssen, Paul Adriaan Jan, Guillemont, Jerome Emile Georges, Paugam, Mikaeel, Delest, Bruno Francois Marie, Heeres, Jan, and Lewi, Paulus Joannes
PATENT: WO 2006045828 ISSUE DATE: 20060504
APPLICATION: 2005 PP: 82 pp.
ASSIGNEE: (Tibotec Pharmaceuticals Ltd., Ire. and Arts, Frank Xavier Jozef Herwig
27. 58760 HIV-LS-355; WOS-HIV-8/20/2006
cis- and trans-decahydro-1,6-naphthyridines. Stereoselective synthesis and stereochemistry
Esipova, TV, Borisenko, AA, and Grishina, GV
RUSSIAN JOURNAL OF ORGANIC CHEMISTRY 2006. 42(6): 922-928, 7
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000239375600019
28. 58761 HIV-LS-355; WOS-HIV-8/20/2006
Chemokine receptor CCR-5 inhibitors produced by Chaetomium globosum
Yang, SW, Mierzwa, R, Terracciano, J, Patel, M, Gullo, V, Wagner, N, Baroudy, B, Puar, M, Chan, TM, McPhail, AT, and Chu, M
JOURNAL OF NATURAL PRODUCTS 2006. 69(7): 1025-1028, 4
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000239336000010