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1. 59375 HIV-LS-361; PUBMED-HIV-11/13/2006

Synthesis and anti-HIV activity evaluation of 1-[(alkenyl or alkynyl or alkyloxy)methyl]-5-alkyl-6-(1-naphthoyl)-2,4-pyrimidinediones as novel non-nucleoside HIV-1 reverse transcriptase inhibitors

Ji, L, Chen, FE, Xie, B, De, Clercq E, Balzarini, J, and Pannecouque, C

Eur J Med Chem 2006.


2. 59376 HIV-LS-361; SCIFINDER-HIV-11/7/2006

Preparation of bicyclic heterocycles, particularly pyrimido[2,1-c][1,4]oxazine-2-carboxamides, as HIV integrase inhibitors

Naidu, BNarasimhulu, Banville, Jacques, Beaulieu, Francis, Connolly, Timothy P, Krystal, Mark R, Matiskella, John D, Ouellet, Carl, Plamondon, Serge, Remillard, Roger, Sorenson, Margaret E, Ueda, Yasutsugu, and Walker, Michael A

PATENT: US 2006199956 ISSUE DATE: 20060907

APPLICATION: 2005-26389 PP: 182pp., Cont.-in-part of U.S. Ser. No. 126,891.


3. 59377 HIV-LS-361; SCIFINDER-HIV-11/7/2006

Anti-HIV quinuclidine compounds

Lecanu, Laurent, Greeson, Janet, and Papadopoulos, Vassilios

PATENT: WO 2006085890 ISSUE DATE: 20060817

APPLICATION: 2005 PP: 28pp.

ASSIGNEE: (Samaritan Pharmaceuticals, Inc. USA and Georgetown University)

4. 59378 HIV-LS-361; PUBMED-HIV-11/13/2006

Anti-HIV-1 Constituents from Leaves and Twigs of Cratoxylum arborescens

Reutrakul, V, Chanakul, W, Pohmakotr, M, Jaipetch, T, Yoosook, C, Kasisit, J, Napaswat, C, Santisuk, T, Prabpai, S, Kongsaeree, P, and Tuchinda, P

Planta Med 2006.


5. 59379 HIV-LS-361; PUBMED-HIV-11/13/2006

Arylthiopyrrole (AThP) Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors: Synthesis, Structure-Activity Relationships, and Docking Studies (Part 2)

Lavecchia, A, Costi, R, Artico, M, Miele, G, Novellino, E, Bergamini, A, Crespan, E, Maga, G, and Di, Santo R

ChemMedChem 2006.


6. 59380 HIV-LS-361; PUBMED-HIV-11/13/2006

Arylthiopyrrole (AThP) Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors: Synthesis, Structure-Activity Relationships, and Docking Studies (Part 1)

Di Santo, R, Costi, R, Artico, M, Miele, G, Lavecchia, A, Novellino, E, Bergamini, A, Cancio, R, and Maga, G

ChemMedChem 2006.


7. 59381 HIV-LS-361; PUBMED-HIV-11/13/2006

Molecular Mechanism by which K70E in HIV-1 Reverse Transcriptase Confers Resistance to Nucleoside Reverse Transcriptase Inhibitors

Sluis-Cremer, N, Sheen, CW, Zelina, S, Argoti, Torres PS, Parikh, UM, and Mellors, JW

Antimicrob Agents Chemother 2006.


8. 59382 HIV-LS-361; PUBMED-HIV-11/13/2006

Critical role of the N-loop and beta1-strand hydrophobic clusters of RANTES-derived peptides in anti-HIV activity

Vangelista, L, Longhi, R, Sironi, F, Pavone, V, and Lusso, P

Biochem Biophys Res Commun 2006.


9. 59383 HIV-LS-361; PUBMED-HIV-11/13/2006

The Role of V1V2 and other HIV-1 Envelope Domains in Resistance to Autologous Neutralization during Clade C Infection

Rong, R, Bibollet-Ruche, F, Mulenga, J, Allen, S, Blackwell, JL, and Derdeyn, CA

J Virol 2006.


10. 59384 HIV-LS-361; PUBMED-HIV-11/13/2006

Ring substituent effects on biological activity of vinyl sulfones as inhibitors of HIV-1

Meadows, DC, Sanchez, T, Neamati, N, North, TW, and Gervay-Hague, J

Bioorg Med Chem 2006.


11. 59385 HIV-LS-361; SCIFINDER-HIV-11/7/2006

Discovery, synthesis and optimization of a new series of selective HIV integrase inhibitors leading to MK-0518 currently in Phase III clinical trial for treatment of HIV/AIDS

Summa, Vincenzo

Abstracts of Papers, 232nd ACS National Meeting, San Francisco, CA, United States, Sept. 10-14, 2006 2006.: MEDI-298

12. 59386 HIV-LS-361; SCIFINDER-HIV-11/7/2006

Short-term antiviral activity of TMC278 - a novel NNRTI - in treatment-naive HIV-1-infected subjects

Goebel, Frank, Yakovlev, Alexy, Pozniak, Anton L, Vinogradova, Elena, Boogaerts, Griet, Hoetelmans, Richard, de Bethune, Marie-Pierre P, Peeters, Monika, and Woodfall, Brian

AIDS (Hagerstown, MD, United States) 2006. 20(13): 1721-1726

13. 59387 HIV-LS-361; SCIFINDER-HIV-11/7/2006

Rational design of polymerase inhibitors as antiviral drugs

Oeberg, Bo

Antiviral Research 2006. 71(2-3): 90-95

14. 59388 HIV-LS-361; SCIFINDER-HIV-11/7/2006

CoMFA study on quinolones as novel inhibitors of HIV-1 reverse transcriptase

Yi, Ping and Qiu, Minghua

Jisuanji Yu Yingyong Huaxue 2006. 23(5): 399-402

15. 59389 HIV-LS-361; SCIFINDER-HIV-11/7/2006

Synthesis, antiviral and cytotoxicity of some new sulphonamides

Selvam, P, Abileshini, B, Alagarsamy, V, Pannecouque, C, and De Clercq, E

Indian Journal of Heterocyclic Chemistry 2006. 16(1): 73-74

16. 59390 HIV-LS-361; SCIFINDER-HIV-11/7/2006

Phosphonate analogs of hiv inhibitor compounds

Boojamra, Constantine G, Lin, Kuei-Ying, Mackman, Richard L, Markevitch, David Y, Petrakovsky, Oleg V, Ray, Adrian S, and Zhang, Lijun

PATENT: WO 2006110157 ISSUE DATE: 20061019

APPLICATION: 2005 PP: 511pp.

ASSIGNEE: (Gilead Sciences, Inc. USA

17. 59391 HIV-LS-361; SCIFINDER-HIV-11/7/2006

Suppression of HIV-1 Protease Inhibitor Resistance by Phosphonate-mediated Solvent Anchoring

Cihlar, Tomas, He, Gong-Xin, Liu, Xiaohong, Chen, James M, Hatada, Marcos, Swaminathan, Swami, McDermott, Martin J, Yang, Zheng-Yu, Mulato, Andrew S, Chen, Xiaowu, Leavitt, Stephanie A, Stray, Kirsten M, and Lee, William A

Journal of Molecular Biology 2006. 363(3): 635-647

18. 59392 HIV-LS-361; SCIFINDER-HIV-11/7/2006

Fused pyrimidinones as HIV integrase inhibitors and their preparation and use in the treatment of HIV infection

Cecere, Giuseppe, Ferreira, Maria Del Rosario Rico, Jones, Philip, Pace, Paola, Petrocchi, Alessia, and Summa, Vincenzo

PATENT: WO 2006103399 ISSUE DATE: 20061005

APPLICATION: 2006 PP: 163pp.

ASSIGNEE: (Istituto De Ricerche Di Biologia Molecolare P Angeletti SpA, Italy

19. 59393 HIV-LS-361; SCIFINDER-HIV-11/7/2006

Fatty acid conjugates with HIV gp41-derived peptide for treatment of HIV infections

Wring, Stephen, Frick, Lloyd, Schneider, Stephen, Zhang, Huyi, Di, Jie, and Heilman, David

PATENT: WO 2006105201 ISSUE DATE: 20061005

APPLICATION: 2006 PP: 118pp.

ASSIGNEE: (Trimeris, Inc. USA

20. 59394 HIV-LS-361; WOS-HIV-11/6/2006

Solution structures and characterization of human immunodeficiency virus Rev responsive element IIB RNA targeting zinc finger proteins

Mishra, SH, Shelley, CM, Barrow, DJ, Darby, MK, and Germann, MW

BIOPOLYMERS 2006. 83(4): 352-364, 13


21. 59395 HIV-LS-361; WOS-HIV-11/13/2006

The engagement of activating Fc gamma Rs inhibits primate lentivirus replication in human macrophages

David, A, Saez-Cirion, A, Versmisse, P, Malbec, O, Iannascoli, B, Herschke, F, Lucas, M, Barre-Sinoussi, F, Mouscadet, JF, Daeron, M, and Pancino, G

JOURNAL OF IMMUNOLOGY 2006. 177(9): 6291-6300, 10


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