'ONLINE DATABASE SEARCH - HIV-LS-363-MEMO
1. 59583 HIV-LS-363; PUBMED-HIV-12/11/2006
Synthesis and properties of G-quartet oligonucleotide-HIV-1 tat peptide conjugate
Kumashiro, T, Otake, T, Kawahata, T, Akagi, M, and Urata, H
Nucleic Acids Symp Ser (Oxf) 2006.(50): 177-178
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17150875&dopt=abstract
2. 59584 HIV-LS-363; PUBMED-HIV-12/11/2006
2'-Deoxy-4'-C-ethynyl-2-fluoroadenosine: A nucleoside reverse transcriptase inhibitor with highly potent activity against all HIV-1 strains, favorable toxic profiles and stability in plasma
Ohrui, H, Kohgo, S, Hayakawa, H, Kodama, E, Matsuoka, M, Nakata, T, and Mitsuya, H
Nucleic Acids Symp Ser (Oxf) 2006.(50): 1-2
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17150787&dopt=abstract
3. 59585 HIV-LS-363; PUBMED-HIV-12/11/2006
Amino disaccharides having an alpha-(1->4) or a beta-(1->4) linkage, their synthesis and evaluation as a potential inhibitor for HIV-1 TAR-Tat
Iguchi, T, Ishikawa, H, Matumoto, H, Mizuno, M, Goto, K, and Hamasaki, K
Nucleic Acids Symp Ser (Oxf) 2005.(49): 169-170
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17150687&dopt=abstract
4. 59586 HIV-LS-363; PUBMED-HIV-12/11/2006
Synthesis and antiviral activity of 1-substituted 3-(3,5-dimethylbenzyl)uracil against HIV-1
Maruyama, T, Kozai, S, Demizu, Y, Witvrouw, M, Pannecouque, C, Balzarini, J, Snoeck, R, Andrei, G, and De, Clercq E
Nucleic Acids Symp Ser (Oxf) 2004.(48): 3-4
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17150449&dopt=abstract
5. 59587 HIV-LS-363; PUBMED-HIV-12/11/2006
Discovery of HIV-1 Protease Inhibitors with Picomolar Affinities Incorporating N-Aryl-oxazolidinone-5-carboxamides as Novel P2 Ligands
Ali, A, Reddy, GS, Cao, H, Anjum, SG, Nalam, MN, Schiffer, CA, and Rana, TM
J Med Chem 2006. 49(25): 7342-7356
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17149864&dopt=abstract
6. 59588 HIV-LS-363; PUBMED-HIV-12/11/2006
Synthesis and anti-HIV evaluation of the novel 2-(m-chlorobenzyl)-4-substituted-7-methyl-1, 1, 3-trioxo-pyrazolo[4, 5-e] [1, 2, 4]thiadiazines
Yan, RZ, Liu, XY, Xu, WF, Pannecouque, C, Witvrouw, M, and De, Clercq E
Arch Pharm Res 2006. 29(11): 957-62
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17146963&dopt=abstract
7. 59589 HIV-LS-363; PUBMED-HIV-12/11/2006
Anti-HIV Activity of Steric Block Oligonucleotides
Ivanova, G, Arzumanov, AA, Turner, JJ, Reigadas, S, Toulme, JJ, Brown, DE, Lever, AM, and Gait, MJ
Ann N Y Acad Sci 2006. 1082: 103-15
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17145931&dopt=abstract
8. 59590 HIV-LS-363; SCIFINDER-HIV-12/4/2006
Design, synthesis and antiviral activity of cyclobutyl phosphonate nucleoside analogs as chain terminators against HIV
Li, Yongfeng, Schinazi, Raymond F, and Liotta, Dennis C
Abstracts of Papers, 232nd ACS National Meeting, San Francisco, CA, United States, Sept. 10-14, 2006 2006.: MEDI-244
9. 59591 HIV-LS-363; PUBMED-HIV-12/11/2006
Antiretroviral Activity, Pharmacokinetics, and Tolerability of MK-0518, a Novel Inhibitor of HIV-1 Integrase, Dosed As Monotherapy for 10 Days in Treatment-Naive HIV-1-Infected Individuals
Markowitz, M, Morales-Ramirez, JO, Nguyen, BY, Kovacs, CM, Steigbigel, RT, Cooper, DA, Liporace, R, Schwartz, R, Isaacs, R, Gilde, LR, Wenning, L, Zhao, J, and Teppler, H
J Acquir Immune Defic Syndr 2006. 43(5): 509-515
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17133211&dopt=abstract
10. 59592 HIV-LS-363; PUBMED-HIV-12/11/2006
Inhibition of HIV-1 replication by siRNA targeting conserved regions of gag/pol
Morris, KV, Chung, CH, Witke, W, and Looney, DJ
RNA Biol 2005. 2(1): 17-20
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17132935&dopt=abstract
11. 59593 HIV-LS-363; PUBMED-HIV-12/11/2006
ANTIVIRAL ACTIVITY OF NOVEL 5-PHOSPHONO-PENT-2-EN-1-YL NUCLEOSIDES AND THEIR ALKOXYALKYL PHOSPHONOESTERS
Choo, H, Beadle, JR, Kern, ER, Prichard, MN, Keith, KA, Hartline, CB, Trahan, J, Aldern, KA, Korba, BE, and Hostetler, KY
Antimicrob Agents Chemother 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17130297&dopt=abstract
12. 59594 HIV-LS-363; SCIFINDER-HIV-12/4/2006
Hiv integrase inhibitors
Vacca, Joseph P, Wai, John S, Payne, Linda S, Isaacs, Richard CA, Han, Wei, Egbertson, Melissa, and Pracitto, Richard
PATENT: WO 2006121831 ISSUE DATE: 20061116
APPLICATION: 2006 PP: 122pp.
ASSIGNEE: (Merck & Co., Inc. USA
13. 59595 HIV-LS-363; PUBMED-HIV-12/11/2006
Interactions between Buprenorphine and Antiretrovirals. II. The Protease Inhibitors Nelfinavir, Lopinavir/Ritonavir, and Ritonavir
McCance-Katz, EF, Moody, DE, Smith, PF, Morse, GD, Friedland, G, Pade, P, Baker, J, Alvanzo, A, Jatlow, P, and Rainey, PM
Clin Infect Dis 2006. 43 Suppl 4: S235-46
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17109310&dopt=abstract
14. 59596 HIV-LS-363; PUBMED-HIV-12/11/2006
Interactions between Buprenorphine and Antiretrovirals. I. The Nonnucleoside Reverse-Transcriptase Inhibitors Efavirenz and Delavirdine
McCance-Katz, EF, Moody, DE, Morse, GD, Friedland, G, Pade, P, Baker, J, Alvanzo, A, Smith, P, Ogundele, A, Jatlow, P, and Rainey, PM
Clin Infect Dis 2006. 43 Suppl 4: S224-34
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17109309&dopt=abstract
15. 59597 HIV-LS-363; PUBMED-HIV-12/11/2006
From dihydroxypyrimidine carboxylic acids to carboxamide HIV-1 integrase inhibitors: SAR around the amide moiety
Petrocchi, A, Koch, U, Matassa, VG, Pacini, B, Stillmock, KA, and Summa, V
Bioorg Med Chem Lett 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17107799&dopt=abstract
16. 59598 HIV-LS-363; SCIFINDER-HIV-12/4/2006
Polynucleotide and polypeptide sequences of HIV-1 Vif variants with antiviral activity and their therapeutic use
Bovolenta, Chiara
PATENT: WO 2006111866 ISSUE DATE: 20061026
APPLICATION: 2006 PP: 84pp.
ASSIGNEE: (Molmed SpA, Italy
17. 59599 HIV-LS-363; PUBMED-HIV-12/11/2006
Synthesis and in Vitro Biological Evaluation of Mannose-Containing Prodrugs Derived from Clinically Used HIV-Protease Inhibitors with Improved Transepithelial Transport
Roche, D, Greiner, J, Aubertin, AM, and Vierling, P
Bioconjug Chem 2006. 17(6): 1568-81
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17105238&dopt=abstract
18. 59600 HIV-LS-363; PUBMED-HIV-12/11/2006
Potent nonnucleoside reverse transcriptase inhibitors target HIV-1 Gag-Pol
Figueiredo, A, Moore, KL, Mak, J, Sluis-Cremer, N, de, Bethune MP, and Tachedjian, G
PLoS Pathog 2006. 2(11): e119
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17096588&dopt=abstract
19. 59601 HIV-LS-363; PUBMED-HIV-12/11/2006
Zinc chelation inhibits HIV Vif activity and liberates antiviral function of the cytidine deaminase APOBEC3G
Xiao, Z, Ehrlich, E, Luo, K, Xiong, Y, and Yu, XF
FASEB J 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17135358&dopt=abstract
20. 59602 HIV-LS-363; SCIFINDER-HIV-12/4/2006
Piperidinylpiperidine derivatives useful as inhibitors of chemokine receptors and their preparation and pharmaceutical compositions
Chan, Tze-Ming, Cox, Kathleen, Feng, Wenqing, Miller, Michael W, Weston, Daniel, and Mccombie, Stuart
PATENT: WO 2006091534 ISSUE DATE: 20060831
APPLICATION: 2006 PP: 92pp.
ASSIGNEE: (Schering Corporation, USA
21. 59603 HIV-LS-363; WOS-HIV-12/04/2006
Synthesis of N,S-substituted 4-chloro-2-mercapto-5-methylbenzenesulfonamide derivatives as potential anti-HIV agents
Brzozowski, Z and Slawinski, J
POLISH JOURNAL OF CHEMISTRY 2006. 80(11): 1807-1815, 9
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000242117200005
22. 59604 HIV-LS-363; WOS-HIV-12/04/2006
Synthesis and anti-HIV activity of nevirapine prodrugs
Sriram, D, Yogeeswari, P, and Kshore, MRK
PHARMAZIE 2006. 61(11): 895-897, 3
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000242002000001
23. 59605 HIV-LS-363; WOS-HIV-12/04/2006
Specific binding of a hexanucleotide to HIV-1 reverse transcriptase: a novel class of bioactive molecules
Mescalchin, A, Wunsche, W, Laufer, SD, Grohmann, D, Restle, T, and Sczakiel, G
NUCLEIC ACIDS RESEARCH 2006. 34(19): 5631-5637, 7
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000241955200038
24. 59606 HIV-LS-363; WOS-HIV-12/04/2006
4,5-dihydroxypyrimidine carboxamides and N-alkyl-5-hydroxypyrimidinone carboxamides are potent, selective HIV integrase inhibitors with good pharmacokinetic profiles in preclinical species
Summa, V, Petrocchi, A, Matassa, VG, Gardelli, C, Muraglia, E, Rowley, M, Paz, OG, Laufer, R, Monteagudo, E, and Pace, P
JOURNAL OF MEDICINAL CHEMISTRY 2006. 49(23): 6646-6649, 4
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000241894000005
25. 59607 HIV-LS-363; SCIFINDER-HIV-12/4/2006
Substituted carbamates as HIV protease inhibitors and their preparation, pharmaceutical compositions and use in the treatment of HIV infection, AIDS and AIDS-related conditions
Mclean, Ed W and Miller, John Franklin
PATENT: WO 2006104646 ISSUE DATE: 20061005
APPLICATION: 2006 PP: 73pp.
ASSIGNEE: (Smithkline Beecham Corporation, USA
26. 59608 HIV-LS-363; WOS-HIV-12/04/2006
Part 13: Synthesis and biological evaluation of piperazine derivatives with dual anti-PAF and anti-HIV-1 or pure antiretroviral activity
Serradji, N, Bensaid, O, Martin, M, Sallem, W, Dereuddre-Bosquet, N, Benmehdi, H, Redeuilh, C, Lamouri, A, Dive, G, Clayette, P, and Heymans, F
BIOORGANIC & MEDICINAL CHEMISTRY 2006. 14(23): 8109-8125, 17
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000242063500045
27. 59609 HIV-LS-363; WOS-HIV-12/04/2006
Resistance profile of a neutralizing anti-HIV monoclonal antibody, KD-247, that shows favourable synergism with anti-CCR5 inhibitors
Yoshimura, K, Shibata, J, Kimura, T, Honda, A, Maeda, Y, Koito, A, Murakami, T, Mitsuya, H, and Matsushita, S
AIDS 2006. 20 (16): 2065-2073, 9
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000242000100008
28. 59610 HIV-LS-363; WOS-HIV-12/11/2006
HIV infection of mononuclear cells is calcium-dependent
Anzinger, JJ, Mezo, I, Ji, X, Gabali, AM, Thomas, LL, and Spear, GT
VIRUS RESEARCH 2006. 122(1-2): 183-188, 6
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000242227300022
29. 59611 HIV-LS-363; WOS-HIV-12/11/2006
Tristetraprolin inhibits HIV-1 production by binding to genomic RNA
Maeda, M, Sawa, H, Tobiume, M, Tokunaga, K, Hasegawa, H, Ichinohe, T, Sata, T, Moriyama, M, Hall, WW, Kurata, T, and Takahashi, H
MICROBES AND INFECTION 2006. 8(11): 2647-2656, 10
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000242207100010
30. 59612 HIV-LS-363; WOS-HIV-12/11/2006
Inhibition of tRNA(3)(Lys)-primed reverse transcription by human APOBEC3G during human immunodeficiency virus type 1 replicationv
Guo, F, Cen, S, Niu, MJ, Saadatmand, J, and Kleiman, L
JOURNAL OF VIROLOGY 2006. 80(23): 11710-11722, 13
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000242222200028
31. 59613 HIV-LS-363; WOS-HIV-12/11/2006
Helicobacter pylori VacA toxin inhibits human immunodeficiency virus infection of primary human T cells
Oswald-Richter, K, Torres, VJ, Sundrud, MS, VanCompernolle, SE, Cover, TL, and Unutmaz, D
JOURNAL OF VIROLOGY 2006. 80(23): 11767-11775, 9
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000242222200033
32. 59614 HIV-LS-363; WOS-HIV-12/11/2006
Synthesis of new substituted 4,5-dihydro-3H-spiro[1,5]-benzoxazepine-2,4 '-piperidine and biological properties
Laras, Y, Pietrancosta, N, Moret, V, Marc, S, Garino, C, Rolland, A, Monnier, V, and Kraus, JL
AUSTRALIAN JOURNAL OF CHEMISTRY 2006. 59(11): 812-818, 7
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000242115500006