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1. 61638 HIV-LS-383; WOS-HIV-9/7/2007

Synthesis of 2-Benzothienyl Carbonyl 4-Arylpiperazines as Novel Delavirdine Analogs

Pessoa-Mahana, H. et al.

Synthetic Communications 2007. 37(7-9): 1227-1235


2. 61639 HIV-LS-383; SCIFINDER-HIV-9/10/2007

CCR5 antagonists useful for treating HIV

Ramanathan, Ragulan, Miller, Michael W, Chowdhury, Swapan K, Alton, Kevin B, Grotz, Diane, Rindgen, Diane, and Tendolkar, Amol

PATENT: US 2007203149 ISSUE DATE: 20070830

APPLICATION: 2007-22529 PP: 17pp.

ASSIGNEE: (Schering Corporation, USA

3. 61640 HIV-LS-383; SCIFINDER-HIV-9/10/2007

Pyridin-2(1H)-ones: a promising class of HIV-1 non-nucleoside reverse transcriptase inhibitors

Medina-Franco, Jose Luis, Martinez-Mayorga, Karina, Juarez-Gordiano, Cecilia, and Castillo, Rafael

ChemMedChem 2007. 2(8): 1141-1147

4. 61641 HIV-LS-383; WOS-HIV-9/7/2007

Human Polycomb Group Eed Protein Negatively Affects Hiv-1 Assembly and Release

Rakotobe, D. et al.

Retrovirology 2007. 4


5. 61642 HIV-LS-383; SCIFINDER-HIV-9/10/2007

pyrrolo[3,4-c]pyrrole derivatives as heterocyclic antiviral compounds and CCR5 receptor antagonists and their preparation, pharmaceutical compositions and use in the treatment of HIV infection, AIDS and ARC

Lemoine, Rcmy, Melville, Chris Richard, Padilla, Fernando, Rotstein, David Mark, and Wanner, Jutta

PATENT: US 2007191406 ISSUE DATE: 20070816

APPLICATION: 2007-51368 PP: 45pp.

ASSIGNEE: (Roche Palo Alto LLC, USA

6. 61643 HIV-LS-383; WOS-HIV-9/7/2007

Ccr5 Small-Molecule Antagonists and Monoclonal Antibodies Exert Potent Synergistic Antiviral Effects by Cobinding to the Receptor

Ji, C. et al.

Molecular Pharmacology 2007. 72(1): 18-28


7. 61644 HIV-LS-383; SCIFINDER-HIV-9/10/2007

Use of 6-(3-chloro-2-fluorobenzyl)-1-[(2S)-1-hydroxy-3-methylbutan-2-yl]-7-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid or salt thereof for treating retrovirus infection

Matsuzaki, Yuji, Kano, Mitsuki, and Ikeda, Satoru

PATENT: WO 2007089030 ISSUE DATE: 20070809

APPLICATION: 2007 PP: 89pp.

ASSIGNEE: (Japan Tobacco Inc., Japan

8. 61645 HIV-LS-383; WOS-HIV-9/7/2007

Rational Optimization of the Binding Affinity of Cd4 Targeting Peptidomimetics With Potential Anti Hiv Activity

Neffe, A. et al.

Journal of Medicinal Chemistry 2007. 50(15): 3482-3488


9. 61646 HIV-LS-383; SCIFINDER-HIV-9/10/2007

Preparation of imidazo[1,2-a]pyridine compds. useful in the treatment of HIV infection and other chemokine receptor-mediated diseases

Gudmundsson, Kristjan, Boggs, Sharon Davis, Miller, John Franklin, and Svolto, Angilique Christina

PATENT: WO 2007087549 ISSUE DATE: 20070802

APPLICATION: 2007 PP: 148pp.

ASSIGNEE: (Smithkline Beecham Corporation, USA

10. 61647 HIV-LS-383; SCIFINDER-HIV-9/10/2007

Imidazo[1,2-a]pyridine-3-carboxamides as anti-HIV agents and their preparation, pharmaceutical compositions and their use in monotherapy and in combination therapy of diseases

Gudmundsson, Kristjan and Turner, Elizabeth Madalena

PATENT: WO 2007087548 ISSUE DATE: 20070802

APPLICATION: 2007 PP: 104pp.

ASSIGNEE: (Smithkline Beecham Corporation, USA and Svolto, Angilique Christina

11. 61648 HIV-LS-383; SCIFINDER-HIV-9/10/2007

Synthesis of 8-halogenated adenosine compounds as antiviral agents

Chang, Junbiao, Cheng, Senxiang, Wang, Limin, Hao, Jia, Wang, Qiang, and Guo, Xiaohe

PATENT: CN 101003550 ISSUE DATE: 20070725

APPLICATION: 1016-30 PP: 14pp.

ASSIGNEE: (Henan Center of Analysis and Test, Peop. Rep. China

12. 61649 HIV-LS-383; SCIFINDER-HIV-9/10/2007

Design and cellular kinetics of dansyl-labeled CADA derivatives with anti-HIV and CD4 receptor down-modulating activity

Vermeire, Kurt, Lisco, Andrea, Grivel, Jean-Charles, Scarbrough, Emily, Dey, Kaka, Duffy, Noah, Margolis, Leonid, Bell, Thomas W, and Schols, Dominique

Biochem. Pharmacol. 2007. 74(4): 566-578

13. 61650 HIV-LS-383; SCIFINDER-HIV-9/10/2007

Hologram quantitative structure-activity relationships for a class of inhibitors of HIV-1 protease

Ferreira, Leonardo G, Leitao, Andrei, Montanari, Carlos A, and Andricopulo, Adriano D

Lett. Drug Des. Discovery 2007. 4(5): 356-364

14. 61651 HIV-LS-383; SCIFINDER-HIV-9/10/2007

A novel bis-tetrahydrofuranylurethane-containing nonpeptidic protease inhibitor (PI), GRL-98065, is potent against multiple-PI-resistant human immunodeficiency virus in vitro

Amano, Masayuki, Koh, Yasuhiro, Das, Debananda, Li, Jianfeng, Leschenko, Sofiya, Wang, Yuan-Fang, Boross, Peter I, Weber, Irene T, Ghosh, Arun K, and Mitsuya, Hiroaki

Antimicrob. Agents Chemother. 2007. 51(6): 2143-2155

15. 61652 HIV-LS-383; SCIFINDER-HIV-9/10/2007

Synthesis and anti-HIV-1 activity of new MKC-442 analogues with an alkynyl-substituted 6-benzyl group

Aly, Youssef L, Pedersen, Erik B, La Colla, Paolo, and Loddo, Roberta

Arch. Pharm. (Weinheim, Ger.) 2007. 340(5): 225-235

16. 61653 HIV-LS-383; WOS-HIV-9/7/2007

Pharmacokinetics of the Anti-Human Immunodeficiency Virus Agent 1-(Beta-D-Dioxolane)Thymine in Rhesus Monkeys

Asif, G. et al.

Antimicrobial Agents and Chemotherapy 2007. 51(7): 2424-2429


17. 61654 HIV-LS-383; WOS-HIV-9/14/2007

Novel Synthesis and Anti-Hiv-1 Activity of 2-Arylthio-6-Benzyl-2,3-Dihydro-1h-Pyrimidin-4-Ones (Aryl S-Dabos)

Aly, Y. et al.

Synthesis-Stuttgart 2007.(13): 1955-1960


18. 61655 HIV-LS-383; WOS-HIV-9/14/2007

Nuclear Factor 90(Nf90) Targeted to Tar Rna Inhibits Transcriptional Activation of Hiv-I

Agbottah, E. et al.

Retrovirology 2007. 4


19. 61656 HIV-LS-383; WOS-HIV-9/14/2007

Qsar Analysis of Caffeoyl Naphthalene Sulfonamide Derivatives as Hiv-1 Integrase Inhibitors

Sahu, K. et al.

Medicinal Chemistry Research 2007. 15(7-8): 418-430


20. 61657 HIV-LS-383; WOS-HIV-9/14/2007

All-Trans Retinoic Acid Attacks Reverse Transcriptase Resulting in Inhibition of Hiv-1 Replication

Maeda, Y. et al.

Hematology 2007. 12(3): 263-266


21. 61658 HIV-LS-383; PUBMED-HIV-9/17/2007

Discovery and Synthesis of HIV Integrase Inhibitors: Development of Potent and Orally Bioavailable N-Methyl Pyrimidones

Gardelli, C, Nizi, E, Muraglia, E, Crescenzi, B, Ferrara, M, Orvieto, F, Pace, P, Pescatore, G, Poma, M, Ferreira, MD, Scarpelli, R, Homnick, CF, Ikemoto, N, Alfieri, A, Verdirame, M, Bonelli, F, Paz, OG, Taliani, M, Monteagudo, E, Pesci, S, Laufer, R, Felock, P, Stillmock, KA, Hazuda, D, Rowley, M, and Summa, V

J Med Chem 2007.


22. 61659 HIV-LS-383; PUBMED-HIV-9/17/2007

Inhibition of Human Immunodeficiency Virus Type-1 Concerted Integration by Strand Transfer Inhibitors Which Recognize a Transient Structural Intermediate

Pandey, KK, Bera, S, Zahm, J, Vora, A, Stillmock, K, Hazuda, D, and Grandgenett, DP

J Virol 2007.


23. 61660 HIV-LS-383; PUBMED-HIV-9/17/2007

Identification of potential HIV-1 targets of minocycline

Jenwitheesuk, E and Samudrala, R

Bioinformatics 2007.


24. 61661 HIV-LS-383; PUBMED-HIV-9/17/2007

Indolyl Aryl Sulfones as HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: Role of Two Halogen Atoms at the Indole Ring in Developing New Analogues with Improved Antiviral Activity

Regina, GL, Coluccia, A, Piscitelli, F, Bergamini, A, Sinistro, A, Cavazza, A, Maga, G, Samuele, A, Zanoli, S, Novellino, E, Artico, M, and Silvestri, R

J Med Chem 2007.


25. 61662 HIV-LS-383; PUBMED-HIV-9/17/2007

Synthesis and Biological Evaluation of Alkenyldiarylmethane HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors That Possess Increased Hydrolytic Stability

Cullen, MD, Deng, BL, Hartman, TL, Watson, KM, Buckheit, RW Jr, Pannecouque, C, Clercq, ED, and Cushman, M

J Med Chem 2007.



26. 61663 HIV-LS-383; PUBMED-HIV-9/17/2007

Fluorescence correlation spectroscopy at single molecule level on the Tat-TAR complex and its inhibitors

Nandi, CK, Parui, PP, Brutschy, B, Scheffer, U, and Gobel, M

Biopolymers 2007.


27. 61664 HIV-LS-383; PUBMED-HIV-9/17/2007

Intracellular Metabolism and Persistence of the Anti-Human Immunodeficiency Virus Activity of 2', 3'-Didehydro-3'-Deoxy-4'- Ethynylthymidine, A Novel Thymidine Analog

Paintsil, E, Dutschman, GE, Hu, R, Grill, SP, Lam, W, Baba, M, Tanaka, H, and Cheng, YC

Antimicrob Agents Chemother 2007.


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