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HIV Citation List: October 1 - October 14, 2008


1. Maneglier B, Rogez-Kreuz C, Dereuddre-Bosquet N, Martal J, Devillier P, Dormont D, Clayette P.

[Anti-HIV effects of IFN-tau in human macrophages: Role of cellular antiviral factors and interleukin-6.]

Pathol Biol (Paris). 2008 Oct 6. [Epub ahead of print] French.

PMID: 18842358 [PubMed - as supplied by publisher]

2. Du L, Zhao YX, Yang LM, Zheng YT, Tang Y, Shen X, Jiang HL.

Symmetrical 1-pyrrolidineacetamide showing anti-HIV activity through a new binding site on HIV-1 integrase.

Acta Pharmacol Sin. 2008 Oct;29(10):1261-7.

PMID: 18817633 [PubMed - in process]

3. Oh CH, Liu LJ, Hong JH.

First synthesis and anti-HIV evaluation of 4'-methyl-cyclopentanyl 9-deazaadenosine.

Nucleosides Nucleotides Nucleic Acids. 2008 Oct;27(10):1144-52.

PMID: 18788044 [PubMed - in process]

4. Pollock S, Dwek RA, Burton DR, Zitzmann N.

N-Butyldeoxynojirimycin is a broadly effective anti-HIV therapy significantly enhanced by targeted liposome delivery.

AIDS. 2008 Oct 1;22(15):1961-9.

PMID: 18753929 [PubMed - in process]

5. Dolin R.

A new class of anti-HIV therapy and new challenges.

N Engl J Med. 2008 Oct 2;359(14):1509-11. No abstract available.

PMID: 18832250 [PubMed - indexed for MEDLINE]

6. Du L, Zhao Y, Chen J, Yang L, Zheng Y, Tang Y, Shen X, Jiang H.

D77, one benzoic acid derivative, functions as a novel anti-HIV-1 inhibitor targeting the interaction between integrase and cellular LEDGF/p75.

Biochem Biophys Res Commun. 2008 Oct 10;375(1):139-44. Epub 2008 Aug 6.

PMID: 18691555 [PubMed - indexed for MEDLINE]

7. Shi W, Qi Z, Pan C, Xue N, Debnath AK, Qie J, Jiang S, Liu K.

Novel anti-HIV peptides containing multiple copies of artificially designed heptad repeat motifs.

Biochem Biophys Res Commun. 2008 Oct 3;374(4):767-72. Epub 2008 Aug 3.

PMID: 18682248 [PubMed - indexed for MEDLINE]

8. Abdurahman S, Végvári A, Youssefi M, Levi M, Höglund S, Andersson E, Horal P, Svennerholm B, Balzarini J, Vahlne A.

Activity of the small modified amino acid alpha-hydroxy glycineamide on in vitro and in vivo human immunodeficiency virus type 1 capsid assembly and infectivity.

Antimicrob Agents Chemother. 2008 Oct;52(10):3737-44. Epub 2008 Jul 21.

PMID: 18644965 [PubMed - in process]

9. Garg H, Francella N, Tony KA, Augustine LA, Barchi JJ Jr, Fantini J, Puri A, Mootoo DR, Blumenthal R.

Glycoside analogs of beta-galactosylceramide, a novel class of small molecule antiviral agents that inhibit HIV-1 entry.

Antiviral Res. 2008 Oct;80(1):54-61. Epub 2008 May 19.

PMID: 18538869 [PubMed - in process]


10. Ma CM, Hattori M, Daneshtalab M, Wang L.

Chlorogenic acid derivatives with alkyl chains of different lengths and orientations: potent alpha-glucosidase inhibitors.

J Med Chem. 2008 Oct 9;51(19):6188-94. Epub 2008 Sep 11.

PMID: 18783210 [PubMed - in process]

Anti-viral and HIV

11. Wang S, Han J, Wang Y, Lu W, Chi C.

Design of peptide inhibitors for furin based on the C-terminal fragment of histone H1.2. Acta Biochim Biophys Sin (Shanghai). 2008 Oct;40(10):848-54.

PMID: 18850049 [PubMed - in process]

(HIV or AIDS) and Antiretroviral

12. He Y, Cheng J, Lu H, Li J, Hu J, Qi Z, Liu Z, Jiang S, Dai Q.

Potent HIV fusion inhibitors against Enfuvirtide-resistant HIV-1 strains.

Proc Natl Acad Sci U S A. 2008 Oct 13. [Epub ahead of print]

PMID: 18852475 [PubMed - as supplied by publisher]

13. Prichard MN, Hartline CB, Harden EA, Daily SL, Beadle JR, Valiaeva N, Kern ER, Hostetler KY.

Inhibition of Herpesvirus Replication by Hexadecyloxypropyl Esters of Purine and Pyrimidine Based Phosphonomethoxyethyl Nucleoside Phosphonates.

Antimicrob Agents Chemother. 2008 Oct 13. [Epub ahead of print]

PMID: 18852272 [PubMed - as supplied by publisher]

14. Tucker TJ, Sisko JT, Tynebor RM, Williams TM, Felock PJ, Flynn JA, Lai MT, Liang Y, McGaughey G, Liu M, Miller M, Moyer G, Munshi V, Perlow-Poehnelt R, Prasad S, Reid JC, Sanchez R, Torrent M, Vacca JP, Wan BL, Yan Y.

Discovery of 3-{5-[(6-Amino-1H-pyrazolo[3,4-b]pyridine-3-yl)methoxy]-2-chlorophenoxy}-5-chlorobenzonitrile (MK-4965): A Potent, Orally Bioavailable HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitor with Improved Potency against Key Mutant Viruses.

J Med Chem. 2008 Oct 1. [Epub ahead of print]

PMID: 18826204 [PubMed - as supplied by publisher]

Du L, Zhao YX, Yang LM, Zheng YT, Tang Y, Shen X, Jiang HL.

Symmetrical 1-pyrrolidineacetamide showing anti-HIV activity through a new binding site on HIV-1 integrase.

Acta Pharmacol Sin. 2008 Oct;29(10):1261-7.

PMID: 18817633 [PubMed - in process]

(HIV or AIDS) and (Therapeutic or Compound)

15. Maga G, Falchi F, Garbelli A, Belfiore A, Witvrouw M, Manetti F, Botta M.

Pharmacophore Modeling and Molecular Docking Led to the Discovery of Inhibitors of Human Immunodeficiency Virus-1 Replication Targeting the Human Cellular Aspartic Acid-Glutamic Acid-Alanine-Aspartic Acid Box Polypeptide 3.

J Med Chem. 2008 Oct 4. [Epub ahead of print]

PMID: 18834110 [PubMed - as supplied by publisher]

16. Sechi M, Azzena U, Delussu MP, Dallocchio R, Dessì A, Cosseddu A, Pala N, Neamati N.

Design and Synthesis of Bis-amide and Hydrazide-containing Derivatives of Malonic Acid as Potential HIV-1 Integrase Inhibitors.

Molecules. 2008 Oct 1;13(10):2442-61.

PMID: 18830166 [PubMed - in process]

17. Liu Y, Zhou E, Yu K, Zhu J, Zhang Y, Xie X, Li J, Jiang H.

Discovery of a Novel CCR5 Antagonist Lead Compound Through Fragment Assembly.

Molecules. 2008 Oct 1;13(10):2426-41.

PMID: 18830165 [PubMed - in process]

(HIV or AIDS) and Drug and Novel

18. Wendeler M, Lee HF, Bermingham A, Miller JT, Chertov O, Bona MK, Baichoo NS, Ehteshami M, Beutler J, O'Keefe BR, Götte M, Kvaratskhelia M, Le Grice S.

Vinylogous Ureas as a Novel Class of Inhibitors of Reverse Transcriptase-Associated Ribonuclease H Activity.

ACS Chem Biol. 2008 Oct 3. [Epub ahead of print]

PMID: 18831589 [PubMed - as supplied by publisher]

(HIV or AIDS) and Drug

19. Waheed AA, Ablan SD, Soheilian F, Nagashima K, Ono A, Schaffner CP, Freed EO.

Inhibition of human immunodeficiency virus type 1 assembly and release by the cholesterol-binding compound amphotericin B methyl ester: evidence for Vpu dependence.

J Virol. 2008 Oct;82(19):9776-81. Epub 2008 Jul 23.

PMID: 18653459 [PubMed - indexed for MEDLINE]

(HIV or AIDS) and Inhibition

20. Nathans R, Cao H, Sharova N, Ali A, Sharkey M, Stranska R, Stevenson M, Rana TM.

Small-molecule inhibition of HIV-1 Vif.

Nat Biotechnol. 2008 Oct;26(10):1187-92. Epub 2008 Sep 21.

PMID: 18806783 [PubMed - in process]

(HIV or AIDS) and Inhibits

21. Melamed JY, Egbertson MS, Varga S, Vacca JP, Moyer G, Gabryelski L, Felock PJ, Stillmock KA, Witmer MV, Schleif W, Hazuda DJ, Leonard Y, Jin L, Ellis JD, Young SD.

Synthesis of 5-(1-H or 1-alkyl-5-oxopyrrolidin-3-yl)-8-hydroxy-[1,6]-naphthyridine-7-carboxamide inhibitors of HIV-1 integrase.

Bioorg Med Chem Lett. 2008 Oct 1;18(19):5307-10. Epub 2008 Aug 14.

PMID: 18774711 [PubMed - in process]

(HIV or AIDS) and Inhibitor

22. De Zotti M, Formaggio F, Kaptein B, Broxterman QB, Felock PJ, Hazuda DJ, Singh SB, Brückner H, Toniolo C.

Complete Absolute Configuration of Integramide A, a Natural, 16-mer Peptide Inhibitor of HIV-1 Integrase, Elucidated by Total Synthesis.

Chembiochem. 2008 Oct 10. [Epub ahead of print] No abstract available.

PMID: 18850604 [PubMed - as supplied by publisher]

(HIV or AIDS) and Class

23. Jessen HJ, Balzarini J, Meier C.

Intracellular Trapping of cycloSal-Pronucleotides: Modification of Prodrugs with Amino Acid Esters.

J Med Chem. 2008 Oct 1. [Epub ahead of print]

PMID: 18826203 [PubMed - as supplied by publisher]

Journal Check

24. Ghosh AK, Gemma S, Baldridge A, Wang YF, Kovalevsky AY, Koh Y, Weber IT, Mitsuya H.

Flexible cyclic ethers/polyethers as novel P2-ligands for HIV-1 protease inhibitors: design, synthesis, biological evaluation, and protein-ligand X-ray studies.

J Med Chem. 2008 Oct 9;51(19):6021-33. Epub 2008 Sep 11.

PMID: 18783203 [PubMed - in process]

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