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HIV Citation List: September 16 - September 29, 2009

Pubmed citations:

1. ADS-J1 inhibits HIV-1 entry by interacting with the gp41 pocket region and blocking the fusion-active gp41 core formation.Wang H, Qi Z, Guo A, Mao Q, Lu H, An X, Xia C, Li X, Debnath AK, Wu S, Liu S, Jiang S. Antimicrob Agents Chemother. 2009 Sep 28. [Epub ahead of print] PMID: 19786602

2. Utilization of in vitro Caco-2 permeability and liver microsomal half-life screens in discovering BMS-488043, a novel HIV-1 attachment inhibitor with improved pharmacokinetic properties. Yang Z, Zadjura LM, Marino AM, D'Arienzo CJ, Malinowski J, Gesenberg C, Lin PF, Colonno RJ, Wang T, Kadow JF, Meanwell NA, Hansel SB. J Pharm Sci. 2009 Sep 24. [Epub ahead of print] PMID: 19780144

3. Inhibitors of Human Immunodeficiency Virus Type 1 (HIV-1) Attachment. 5. An Evolution from Indole to Azaindoles Leading to the Discovery of 1-(4-Benzoylpiperazin-1-yl)-2-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)ethane-1,2-dione (BMS-488043), a Drug Candidate That Demonstrates Antiviral Activity in HIV-1-Infected Subjects (infinity). Wang T, Yin Z, Zhang Z, Bender JA, Yang Z, Johnson G, Yang Z, Zadjura LM, D'Arienzo CJ, Digiugno Parker D, Gesenberg C, Yamanaka GA, Gong YF, Ho HT, Fang H, Zhou N, McAuliffe BV, Eggers BJ, Fan L, Nowicka-Sans B, Dicker IB, Gao Q, Colonno RJ, Lin PF, Meanwell NA, Kadow JF. J Med Chem. 2009 Sep 21. [Epub ahead of print] PMID: 19769332

ISI Web of Knowledge citations:

4. Quantitative Structure-Activity Relationship Studies on 2-Amino-6-arylsulfonylbenzonitriles as Human Immunodeficiency Viruses Type 1 Reverse Transcriptase Inhibitors Using Descriptors Obtained from Substituents and Whole Molecular Structures. Hemmateenejad, B; Sabet, R; Fassihi, A. CHEMICAL BIOLOGY & DRUG DESIGN, 2009; 74(4): 405-415.

5. Optimal drug combinations and minimal hitting sets.Vazquez, A. BMC SYSTEMS BIOLOGY, 2009; 3: 4930U.

6. Spiropiperidine CCR5 antagonists. Rotstein, DM; Gabriel, SD; Makra, F; Filonova, L; Gleason, S; Brotherton-Pleiss, C; Setti, LQ; Trejo-Martin, A; Lee, EK; Sankuratri, S; Ji, CH; deRosier, A; Dioszegi, M; Heilek, G; Jekle, A; Berry, P; Weller, P; Mau, CI. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009; 19(18): 5401-5406.

7. Dipyridodiazepinone derivatives; synthesis and anti HIV-1 activity. Khunnawutmanotham, N; Chimnoi, N; Thitithanyanont, A; Saparpakorn, P; Choowongkomon, K; Pungpo, P; Hannongbua, S; Techasakul, S. BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY, 2009; 5: 493CK

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