1. In Vitro Evaluation of Novel Reverse Transcriptase Inhibitors TAF (Tenofovir alafenamide) and OBP-601 (2,3-Didehydro-3-deoxy-4-ethynylthymidine) against Multi-drug Resistant Primary Isolates of HIV-2. Bartolo, I., P. Borrego, P. Gomes, F. Goncalves, U. Caixas, I.V. Pinto, and N. Taveira. Antiviral Research, 2019. 161: p. 85-89. PMID[30391482].
[PubMed]. HIV_01_2019.
2. Synthesis, anti-HBV, and anti-HIV Activities of 3 '-Halogenated Bis(hydroxymethyl)-cyclopentenyladenines. Kumamoto, H., S. Imoto, M. Amano, N. Kuwata-Higashi, M. Baba, H. Mitsuya, Y. Odanaka, S.S. Matsubayashi, H. Tanaka, and K. Haraguchi. ACS Medicinal Chemistry Letters, 2018. 9(12): p. 1211-1216. PMID[30613328]. PMCID[PMC6295849].
[PubMed]. HIV_01_2019.
3. Design, Synthesis, Molecular Modeling, in Silico ADME Studies and anti-HIV-1 Assay of New Diazocoumarin Derivatives. Livani, Z.A., M. Safakish, Z. Hajimahdi, S. Soleymani, R. Zabihollahi, M.R. Aghasadeghi, E. Alipour, and A. Zarghi. Iranian Journal of Pharmaceutical Research, 2018. 17: p. 65-77. ISI[000455744400007].
[WOS]. HIV_01_2019.
4. Benzolactam-related Compounds Promote Apoptosis of HIV-infected Human Cells via Protein Kinase C-Induced HIV Latency Reversal. Matsuda, K., T. Kobayakawa, K. Tsuchiya, S.I. Hattori, W. Nomura, H. Gatanaga, K. Yoshimura, S. Oka, Y. Endo, H. Tamamura, H. Mitsuya, and K. Maeda. Journal of Biological Chemistry, 2019. 294(1): p. 116-129. PMID[30413535]. PMCID[PMC6322896].
[PubMed]. HIV_01_2019.
5. In Vitro Inhibitory Effect of Lanostane triterpenoids of Kadsura coccinea on the Human Immunodeficiency Virus Type-1 Protease. Nguyen, H.L., T.H.T. Tran, T.T. Phuong, and T.N. Phan. Indian Journal of Pharmaceutical Sciences, 2018. 80(4): p. 755-761. ISI[000455182700021].
[WOS]. HIV_01_2019.
6. CXCR4-targeting Nanobodies Differentially Inhibit CXCR4 Function and HIV Entry. Van Hout, A., A. Klarenbeek, V. Bobkov, J. Doijen, M. Arimont, C.X. Zhao, R. Heukers, R. Rimkunas, C. de Graaf, T. Verrips, B. van der Woning, H. de Haard, J.B. Rucker, K. Vermeire, T. Handel, T. Van Loy, M.J. Smit, and D. Schols. Biochemical Pharmacology, 2018. 158: p. 402-412. PMID[30342024].
[PubMed]. HIV_01_2019.
7. Design, Synthesis and Biological Evaluation of Novel Acetamide-substituted Doravirine and its Prodrugs as Potent HIV-1 NNRTIs. Wang, Z., Z. Yu, D.W. Kang, J. Zhang, Y. Tian, D. Daelemans, E. De Clercq, C. Pannecouque, P. Zhan, and X.Y. Liu. Bioorganic & Medicinal Chemistry, 2019. 27(3): p. 447-456. PMID[30606670].
[PubMed]. HIV_01_2019.
8. Human Cervical Epithelial Cells Release Antiviral Factors and Inhibit HIV Replication in Macrophages. Xu, X.Q., L. Guo, X. Wang, Y. Liu, H. Liu, R.H. Zhou, J. Gu, J.B. Liu, P. Xu, L. Zhou, and W.Z. Ho. Journal of Innate Immunity, 2019. 11(1): p. 29-40. PMID[30032138]. PMCID[PMC6338329].
[PubMed]. HIV_01_2019.
9. Active-site Deformation in the Structure of HIV-1 RT with HBV-associated Septuple Amino acid Substitutions Rationalizes the Differential Susceptibility of HIV-1 and HBV against 4'-Modified Nucleoside RT Inhibitors. Yasutake, Y., S.I. Hattori, N. Tamura, K. Matsuda, S. Kohgo, K. Maeda, and H. Mitsuya. Biochemical and Biophysical Research Communications, 2019. 509(4): p. 943-948. PMID[30648556].
[PubMed]. HIV_01_2019.
10. The BET Bromodomain Inhibitor Apabetalone Induces Apoptosis of Latent HIV-1 Reservoir Cells Following Viral Reactivation. Zhang, X.X., J. Lin, T.Z. Liang, H. Duan, X.H. Tan, B.M. Xi, L. Li, and S.W. Liu. Acta Pharmacologica Sinica, 2019. 40(1): p. 98-110. PMID[29789664]. PMCID[PMC6318340].
[PubMed]. HIV_01_2019.
Patent Citations
This month, no relevant HIV patents were identified.