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2. Targeting HIV-1 RNase H: N'-(2-Hydroxy-benzylidene)-3,4,5-trihydroxybenzoylhydrazone as Selective Inhibitor Active against NNRTIs-resistant Variants. Corona, A., E. Ballana, S. Distinto, D. Rogolino, C. Del Vecchio, M. Carcelli, R. Badia, E. Riveira-Muñoz, F. Esposito, C. Parolin, J.A. Esté, N. Grandi, and E. Tramontano. Viruses, 2020. 12(7): E729. PMID[32640577].
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3. Inhibition of HIV Replication through siRNA Carried by CXCR4-targeted Chimeric Nanobody. Cunha-Santos, C., P.R.L. Perdigao, F. Martin, J.G. Oliveira, M. Cardoso, A. Manuel, N. Taveira, and J. Goncalves. Cellular and Molecular Life Sciences, 2020. 77(14): p. 2859-2870. PMID[31641784].
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4. 4-Deoxyphorbol Inhibits HIV-1 Infection in Synergism with Antiretroviral Drugs and Reactivates Viral Reservoirs through PKC/MEK Activation Synergizing with Vorinostat. De la Torre-Tarazona, H.E., R. Jiménez, P. Bueno, S. Camarero, L. Román, J.L. Fernández-García, M. Beltrán, L.F. Nothias, X. Cachet, J. Paolini, M. Litaudon, J. Alcami, and L.M. Bedoya. Biochemical Pharmacology, 2020. 177: 113937. PMID[32224142].
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5. Synthesis, Bioactivity and Binding Energy Calculations of Novel 3-Ethoxysalicylaldehyde Based Thiosemicarbazone Derivatives. Ishaq, M., P. Taslimi, Z. Shafiq, S. Khan, R. Ekhteiari Salmas, M.M. Zangeneh, A. Saeed, A. Zangeneh, N. Sadeghian, A. Asari, and H. Mohamad. Bioorganic Chemistry, 2020. 100: 103924. PMID[32442818].
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6. In Vitro anti-HIV Effect of Voacamine from Voacanga africana Stapf Based on the SPRi Experiment. Li, H.X., R.Q. Liu, H.M. Zhang, Z.X. Cao, L.X. Zhu, Y.Y. Li, W.J. Ding, Y.H. Chen, and Y. Deng. Russian Journal of Bioorganic Chemistry, 2020. 46(3): p. 306-311. ISI[000541338600005].
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7. Uracil-containing Heterodimers of a New Type: Synthesis and Study of Their Anti-viral Properties. Maslova, A.A., E.S. Matyugina, R. Snoeck, G. Andrei, S.N. Kochetkov, A.L. Khandazhinskaya, and M.S. Novikov. Molecules, 2020. 25(15): E3350. PMID[32717979].
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8. Oregano Oil and Its Principal Component, Carvacrol, Inhibit HIV-1 Fusion into Target Cells. Mediouni, S., J.A. Jablonski, S. Tsuda, A. Barsamian, C. Kessing, A. Richard, A. Biswas, F. Toledo, V.M. Andrade, Y. Even, M. Stevenson, T. Tellinghuisen, H. Choe, M. Cameron, T.D. Bannister, and S.T. Valente. Journal of Virology, 2020. 94(15): e00147-20. PMID[32461309]. [PMC7375364].
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9. Design, Synthesis and SAR Study of Bridged Tricyclic Pyrimidinone Carboxamides as HIV-1 Integrase Inhibitors. Patel, M., B.N. Naidu, I. Dicker, H. Higley, Z. Lin, B. Terry, T. Protack, M. Krystal, S. Jenkins, D. Parker, C. Panja, R. Rampulla, A. Mathur, N.A. Meanwell, and M.A. Walker. Bioorganic & Medicinal Chemistry, 2020. 28(13): 115541. PMID[32389483].
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10. Novel Pyranopyrazole Derivatives Comprising a Benzoxazole Core as Antimicrobial Inhibitors: Design, Synthesis, Microbial Resistance and Machine Aided Results. Reddy, G.M., A.K. Kumari, V.H. Reddy, and J.R. Garcia. Bioorganic Chemistry, 2020. 100: 103908. PMID[32413632].
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11. Discovery of Potential Dual-target Prodrugs of HIV-1 Reverse Transcriptase and Nucleocapsid Protein 7. Sun, S.K., B.S. Huang, Z. Li, Z. Wang, L. Sun, P. Gao, D.W. Kang, C.H. Chen, K.H. Lee, D. Daelemans, E. De Clercq, C. Pannecouque, P. Zhan, and X.Y. Liu. Bioorganic & Medicinal Chemistry Letters, 2020. 30(16): 127287. PMID[32631509].
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12. Chemical Profiling of HIV-1 Capsid-targeting Antiviral PF74. Wang, L., M.C. Casey, S.K.V. Vernekar, H.T. Do, R.L. Sahani, K.A. Kirby, H.J. Du, A. Hachiya, H.C. Zhang, P.R. Tedbury, J.S. Xie, S.G. Sarafianos, and Z.Q. Wang. European Journal of Medicinal Chemistry, 2020. 200: 112427. PMID[32438252].
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15. Piperidine Scaffold as the Novel P2-ligands in Cyclopropyl-containing HIV-1 Protease Inhibitors: Structure-based Design, Synthesis, Biological Evaluation and Docking Study. Zhou, H., M. Zhu, L. Ma, J. Zhou, B. Dong, G. Zhang, S. Cen, Y. Wang, and J. Wang. Plos One, 2020. 15(7): e0235483. PMID[32697773]. PMCID[PMC7375528].
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17. Design and Biological Evaluation of Novel HIV-1 Protease Inhibitors with Isopropanol as P1' Ligand to Enhance Binding with S1' Subsite. Zhu, M., L. Ma, B. Dong, G. Zhang, J. Wang, J. Zhou, S. Cen, and Y. Wang. Bioorganic & Medicinal Chemistry, 2020. 28(16): p. 115623. PMID[32690263].
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Patent Citations
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