Literature Citations
1. Abundant Extractable Metabolites from Temperate Tree Barks: The Specific Antimicrobial Activity of Prunus avium Extracts. Abedini, A., M. Colin, J. Hubert, E. Charpentier, A. Angelis, H. Bounasri, B. Bertaux, A. Kotland, F. Reffuveille, J.M. Nuzillard, J.H. Renault, and S.C. Gangloff. Antibiotics, 2020. 9(3): E111. PMID[32143394].
[PubMed]. TB_03_2020.
2. In Silico Study for Evaluating the Binding Mode and Interaction of 1,2,4-Triazole and its Derivatives as Potent Inhibitors against Lipoate Protein B (LipB). Adeniji, S.E., S. Uba, and A. Uzairu. Journal of King Saud University Science, 2020. 32(1): p. 475-485. ISI[000506167000064].
[WOS]. TB_03_2020.
3. Synthesis and in Vitro Evaluation of Antimycobacterial and Cytotoxic Activity of New alpha,beta-unsaturated Amide, Oxazoline and Oxazole Derivatives from L-Serine. Aguirre-Renteria, S.A., J.J.J. Carrizales-Castillo, M. Del Rayo Camacho Corona, E. Hernandez-Fernandez, E. Garza-Gonzalez, V.M. Rivas-Galindo, E. Arredondo-Espinoza, and F.G. Avalos-Alanis. Bioorganic and Medicinal Chemistry Letters, 2020. 30(9): e127074. PMID[32151467].
[PubMed]. TB_03_2020.
4. 5-Alkylamino-N-phenylpyrazine-2-carboxamides: Design, Preparation, and Antimycobacterial Evaluation. Ambrozkiewicz, W., M. Kucerova-Chlupacova, O. Jandourek, K. Konecna, P. Paterova, P. Barta, J. Vinsova, M. Dolezal, and J. Zitko. Molecules, 2020. 25(7): e1561. PMID[32231166].
[PubMed]. TB_03_2020.
5. Novel Benzothiazole Containing 4H-Pyrimido[2,1-b]benzothiazoles Derivatives: One Pot, Solvent-free Microwave Assisted Synthesis and their Biological Evaluation. Bhoi, M.N., M.A. Borad, E.A. Pithawala, and H.D. Patel. Arabian Journal of Chemistry, 2019. 12(8): p. 3799-3813. ISI[000504900300194].
[WOS]. TB_03_2020.
6. Mycobacterium tuberculosis Decaprenylphosphoryl-beta-D-ribose Oxidase Inhibitors: Expeditious Reconstruction of Suboptimal Hits into a Series with Potent in Vivo Activity. Borthwick, J.A., C. Alemparte, I. Wall, B.C. Whitehurst, A. Argyrou, G. Burley, P. de Dios-Anton, L. Guijarro, M.C. Monteiro, F. Ortega, C.J. Suckling, J.C. Pichel, M. Cacho, and R.J. Young. Journal of Medicinal Chemistry, 2020. 63(5): p. 2557-2576. PMID[31922409].
[PubMed]. TB_03_2020.
7. Bioorganometallic Derivatives of 4-Hydrazino-benzenesulphonamide as Carbonic Anhydrase Inhibitors: Synthesis, Characterisation and Biological Evaluation. Brichet, J., R. Arancibia, E. Berrino, and C.T. Supuran. Journal of Enzyme Inhibition and Medicinal Chemistry, 2020. 35(1): p. 622-628. PMID[32037900]. PMCID[PMC7034112].
[PubMed]. TB_03_2020.
8. Synthesis, Characterization, and Biological Evaluation of Novel 7-Oxo-7H-thiazolo[3,2-b]-1,2,4-triazine-2-carboxylic acid Derivatives. Cai, D., T. Li, Q. Xie, X. Yu, W. Xu, Y. Chen, Z. Jin, and C. Hu. Molecules, 2020. 25(6): E1307. PMID[32182992].
[PubMed]. TB_03_2020.
9. Design, Synthesis and Evaluation of Antitubercular Activity of Triclosan Analogues. Cinu, T.A., S.K. Sidhartha, B. Indira, B.G. Varadaraj, P.S. Vishnu, and G.G. Shenoy. Arabian Journal of Chemistry, 2019. 12(8): p. 3316-3323. ISI[000504900300154].
[WOS]. TB_03_2020.
10. Structure-based Design and Synthesis of Piperidinol-containing Molecules as New Mycobacterium abscessus Inhibitors. de Ruyck, J., C. Dupont, E. Lamy, V. Le Moigne, C. Biot, Y. Guerardel, J.L. Herrmann, M. Blaise, S. Grassin-Delyle, L. Kremer, and F. Dubar. ChemistryOpen, 2020. 9(3): p. 351-365. PMID[32211280]. PMCID[PMC7083170].
[PubMed]. TB_03_2020.
11. Synthesis, Anticancer, Antimicrobial, Anti-tuberculosis and Molecular Docking of Heterocyclic N-Ethyl-N-methylbenzenesulfonamide Derivatives. Debbabi, K.F., S.A. Al-Harbi, H.M. Al-Saidi, E.H. Aljuhani, R.N. Felaly, S.M. Abd El-Gilil, M.S. Bashandy, and H. ben Jannet. Journal of Molecular Structure, 2020. 1203: e127423. ISI[000504448700052].
[WOS]. TB_03_2020.
12. In Vitro Susceptibility Testing of GSK656 against Mycobacterium Species. Dong, W., S. Li, S. Wen, W. Jing, J. Shi, Y. Ma, F. Huo, F. Gao, Y. Pang, and J. Lu. Antimicrobial Agents and Chemotherapy, 2020. 64(2): e01577-19. PMID[31791947]. PMCID[PMC6985724].
[PubMed]. TB_03_2020.
13. Synthesis and Biological Evaluation of a Novel C8-Pyrrolobenzodiazepine (PBD) Adenosine Conjugate. A Study on the Role of the PBD Ring in the Biological Activity of PBD-conjugates. Ferguson, L., S. Bhakta, K.R. Fox, G. Wells, and F. Brucoli. Molecules, 2020. 25(5): e1243. PMID[32164166].
[PubMed]. TB_03_2020.
14. Synthesis and Efficacy of Pyrvinium-inspired Analogs against Tuberculosis and Malaria Pathogens. Gaikwad, V.R., U.B. Karale, G. Govindarajalu, N. Adhikari, E.V. Krishna, V.S. Krishna, S. Misra, D. Sriram, P.S. Sijwali, and H.B. Rode. Bioorganic and Medicinal Chemistry Letters, 2020. 30(8): e127037. PMID[32081449].
[PubMed]. TB_03_2020.
15. Synthesis and Evaluation of Coumarin Hybrids as Antimycobacterial Agents. Hassan, M.Z., A. Alsayari, H. Osman, M.A. Ali, A. Bin Muhsinah, and M.J. Ahsan. Acta Poloniae Pharmaceutica, 2019. 76(6): p. 1029-1036. ISI[000504705900010].
[WOS]. TB_03_2020.
16. Novel Pyrazine Based Anti-tubercular Agents: Design, Synthesis, Biological Evaluation and in Silico Studies. Hassan, N.W., M.N. Saudi, Y.S. Abdel-Ghany, A. Ismail, P.A. Elzahhar, D. Sriram, R. Nassra, M.M. Abdel-Aziz, and S.A. El-Hawash. Bioorganic Chemistry, 2020. 96: e103610. PMID[32028062].
[PubMed]. TB_03_2020.
17. N-Pyrazinoyl Substituted Amino Acids as Potential Antimycobacterial Agents-the Synthesis and Biological Evaluation of Enantiomers. Juhas, M., L. Kucerova, O. Horacek, O. Jandourek, V. Kubicek, K. Konecna, R. Kucera, P. Barta, J. Janousek, P. Paterova, J. Kunes, M. Dolezal, and J. Zitko. Molecules, 2020. 25(7): E1518. PMID[32230728].
[PubMed]. TB_03_2020.
18. New 2-Ethylthio-4-methylaminoquinazoline Derivatives Inhibiting Two Subunits of Cytochrome bc1 in Mycobacterium tuberculosis. Lupien, A., C.S. Foo, S. Savina, A. Vocat, J. Piton, N. Monakhova, A. Benjak, D.A. Lamprecht, A.J.C. Steyn, K. Pethe, V.A. Makarov, and S.T. Cole. Plos Pathogens, 2020. 16(1): e1008270. PMID[31971990]. PMCID[PMC6999911].
[PubMed]. TB_03_2020.
19. Novel Substituted Aniline Based Heterocyclic Dispersed Azo Dyes Coupling with 5-Methyl-2-(6-methyl-1,3-benzothiazol-2-yl)-2,4-dihydro-3H-pyrazol-3-one: Synthesis, Structural, Computational and Biological Studies. Maliyappa, M.R., J. Keshavayya, N.M. Mallikarjuna, and I. Pushpavathi. Journal of Molecular Structure, 2020. 1205: e127576. ISI[000511287400051].
[WOS]. TB_03_2020.
20. Synthesis, in Vitro, and in Vivo (Zebra Fish) Antitubercular Activity of 7,8-Dihydroquinolin-5(6H)-ylidenehydrazinecarbothioamides. Marvadi, S.K., V.S. Krishna, G. Surineni, R. Srilakshmi Reshma, B. Sridhar, D. Sriram, and S. Kantevari. Bioorganic Chemistry, 2020. 96: e103626. PMID[32007719].
[PubMed]. TB_03_2020.
21. Complexes of Cu (II) with alpha-Ketoglutaric acid and 1-(O-Tolyl) biguanide Synthesis, Characterization and Biological Activity. Mihalache, M., C. Guran, A. Meghea, V. Bercu, L. Motelica, and A.M. Holban. Revista de Chimie, 2019. 70(10): p. 3603-3610. ISI[000500795900032].
[WOS]. TB_03_2020.
22. Design, Synthesis and Biological Evaluation of 5-(2-(4-(Substituted benzo[d]isoxazol-3-yl) piperazin-1-yl)acetyl)indolin-2-one and 5-(2-(4-Substitutedpiperazin-1-yl)acetyl)indolin-2-one Analogues as Novel Anti-tubercular Agents. Naidu, K.M., R.N. Gajanan, and K. Sekhar. Arabian Journal of Chemistry, 2019. 12(8): p. 2418-2429. ISI[000504900300067].
[WOS]. TB_03_2020.
23. Synthesis of Water-soluble Prodrugs of 5-Modified 2'-deoxyuridines and their Antibacterial Activity. Negrya, S.D., M.V. Jasko, P.N. Solyev, I.L. Karpenko, O.V. Efremenkova, B.F. Vasilyeva, I.G. Sumarukova, S.N. Kochetkov, and L.A. Alexandrova. Journal of Antibiotics, 2020. 73(4): p. 236-246. PMID[31932744].
[PubMed]. TB_03_2020.
24. Structure-based Discovery of Novel Inhibitors of Mycobacterium tuberculosis Cyp121 from Indonesian Natural Products. Prasasty, V.D., S. Cindana, F.X. Ivan, H. Zahroh, and E. Sinaga. Computational Biology and Chemistry, 2020. 85: e107205. PMID[31981965].
[PubMed]. TB_03_2020.
25. Psoralen Derivatives as Inhibitors of Mycobacterium tuberculosis Proteasome. Rozman, K., E.M. Alexander, E. Ogorevc, K. Bozovicar, I. Sosic, C.C. Aldrich, and S. Gobec. Molecules, 2020. 25(6): E1305. PMID[32178473].
[PubMed]. TB_03_2020.
26. TBAJ-876, a 3,5-Dialkoxypyridine Analogue of Bedaquiline, Is Active against Mycobacterium abscessus. Sarathy, J.P., U.S. Ganapathy, M.D. Zimmerman, V. Dartois, M. Gengenbacher, and T. Dick. Antimicrobial Agents and Chemotherapy, 2020. 64(4): e02404-19. PMID[31964791].
[PubMed]. TB_03_2020.
27. Design, Synthesis and Antimycobacterial Activity of Thiazolidine-2,4-dione-based Thiosemicarbazone Derivatives. Trotsko, N., J. Golus, P. Kazimierczak, A. Paneth, A. Przekora, G. Ginalska, and M. Wujec. Bioorganic Chemistry, 2020. 97: p. e103676. PMID[32097795].
[PubMed]. TB_03_2020.
28. In Silico Design and Synthesis of Tetrahydropyrimidinones and Tetrahydropyrimidinethiones as Potential Thymidylate Kinase Inhibitors Exerting anti-TB Activity against Mycobacterium tuberculosis. Venugopala, K.N., C. Tratrat, M. Pillay, S. Chandrashekharappa, O.H.A. Al-Attraqchi, B.E. Aldhubiab, M. Attimarad, O.I. Alwassil, A.B. Nair, N. Sreeharsha, R. Venugopala, M.A. Morsy, M. Haroun, H.M. Kumalo, B. Odhav, and K. Mlisana. Drug Design, Development and Therapy, 2020. 14: p. 1027-1039. PMID[32214795]. PMCID[PMC7082623].
[PubMed]. TB_03_2020.
29. Development of New Antituberculosis Drugs among of 1,3-and 1,4-Diazines. Highlights and Perspectives. Verbitskiy, E.V., G.L. Rusinov, V.N. Charushin, and O.N. Chupakhin. Russian Chemical Bulletin, 2019. 68(12): p. 2172-2189. ISI[000512030400004].
[WOS]. TB_03_2020.
30. Antimycobacterial Rufomycin Analogues from Streptomyces atratus Strain MJM3502. Zhou, B., G. Shetye, Y. Yu, B.D. Santarsiero, L.L. Klein, C. Abad-Zapatero, N.M. Wolf, J. Cheng, Y. Jin, H. Lee, J.W. Suh, H. Lee, J. Bisson, J.B. McAlpine, S.N. Chen, S.H. Cho, S.G. Franzblau, and G.F. Pauli. Journal of Natural Products, 2020. 83(3): p. 657-667. PMID[32031795].
[PubMed]. TB_03_2020.
31. Single-step Synthesis and in Vitro Anti-mycobacterial Activity of Novel Nitrofurantoin Analogues. Zuma, N.H., F.J. Smit, R. Seldon, J. Aucamp, A. Jordaan, D.F. Warner, and D.D. N'Da. Bioorganic Chemistry, 2020. 96: e103587. PMID[32044516].
[PubMed]. TB_03_2020.
Patent Citations
32. Amino(pyridinyl)butanols as Antibacterial Agents and Their Preparation Baell, J., D. Priebbenow, L. Barbaro, and D. Che. Patent. 2020. 2019-AU50945 2020047596: 69pp.
[PubMed]. TB_03_2020.