Literature Citations
1. Synthesis and Antimicrobial Evaluation of Piperic acid Amides and their Lower Homologues. Achanta, P.S., S. Raj, S. Horam, J. Arockiaraj, R.K. Bobbala, R.R. Akkinepally, M. Pasupuleti, and A. Achanta. Drug Development Research, 2020. 81(3): p. 366-373. PMID[31800126].
[PubMed]. TB_05_2020.
2. Anti-tubercular Activity of Novel Class of Spiropyrrolidine Tethered Indenoquinoxaline Heterocyclic Hybrids. Arumugam, N., A.I. Almansour, R. Suresh Kumar, S. Ibrahim Alaqeel, V. Siva Krishna, and D. Sriram. Bioorganic Chemistry, 2020. 99: e103799. PMID[32247109].
[PubMed]. TB_05_2020.
3. Optimization of Hydantoins as Potent Antimycobacterial Decaprenylphosphoryl-Β-D-Ribose Oxidase (Dpre1) Inhibitors. Balabon, O., E. Pitta, M.K. Rogacki, E. Meiler, R. Casanueva, L. Guijarro, S. Huss, E.M. Lopez-Roman, Á. Santos-Villarejo, K. Augustyns, L. Ballell, D.B. Aguirre, R.H. Bates, F. Cunningham, M. Cacho, and P. Van der Veken. Journal of Medicinal Chemistry, 2020. 63(10): p. 5367-5386. PMID[32342688].
[PubMed]. TB_05_2020.
4. Design, Synthesis, in Vitro and in Silico Studies of 2,3-Diaryl benzofuran Derivatives as Antitubercular Agents. Bhukya, B., A. Shukla, V. Chaturvedi, P. Trivedi, S. Kumar, F. Khan, A.S. Negi, and S.K. Srivastava. Bioorganic Chemistry, 2020. 99: e103784. PMID[32361184].
[PubMed]. TB_05_2020.
5. Meridianin D Analogues Possess Antibiofilm Activity against Mycobacterium smegmatis. Brackett, S.M., K.E. Cox, S.L. Barlock, W.M. Huggins, D.F. Ackart, R.J. Bassaraba, R.J. Melander, and C. Melander. RSC Medicinal Chemistry, 2020. 11(1): p. 92-97. ISI[000526949900008].
[WOS]. TB_05_2020.
6. Identification of Substituted Amino acid Hydrazides as Novel Anti-tubercular Agents, Using a Scaffold Hopping Approach. Brown, A.K., A.K.B. Aljohani, F.M.A. Alsalem, J.L. Broadhead, J.H. Gill, Y. Lu, and J.D. Sellars. Molecules, 2020. 25(10): e2387. PMID[32455566].
[PubMed]. TB_05_2020.
7. "In Vitro" Activity of Melaleuca cajuputi against Mycobacterial Species. Bua, A., P. Molicotti, M.G. Donadu, D. Usai, L.S. Le, T.T.T. Tran, V.Q.T. Ngo, M. Marchetti, M. Usai, P. Cappuccinelli, and S. Zanetti. Natural Product Research, 2020. 34(10): p. 1494-1497. PMID[30518254].
[PubMed]. TB_05_2020.
8. Discovery of a Natural Product That Binds to the Mycobacterium tuberculosis Protein Rv1466 Using Native Mass Spectrometry. Elnaas, A.R., D. Grice, J. Han, Y. Feng, A.D. Capua, T. Mak, J.A. Laureanti, G.W. Buchko, P.J. Myler, G. Cook, R.J. Quinn, and M. Liu. Molecules, 2020. 25(10): 2384. PMID[32455540].
[PubMed]. TB_05_2020.
9. OPC-167832, a Novel Carbostyril Derivative with Potent Antituberculosis Activity as a DprE1 Inhibitor. Hariguchi, N., X. Chen, Y. Hayashi, Y. Kawano, M. Fujiwara, M. Matsuba, H. Shimizu, Y. Ohba, I. Nakamura, R. Kitamoto, T. Shinohara, Y. Uematsu, S. Ishikawa, M. Itotani, Y. Haraguchi, I. Takemura, and M. Matsumoto. Antimicrobial Agents and Chemotherapy, 2020. 64(6): p. 1-13. PMID[32229496]. PMCID[PMC7269503].
[PubMed]. TB_05_2020.
10. Brassicasterol with Dual Anti-infective Properties against HSV-1 and Mycobacterium tuberculosis, and Cardiovascular Protective Effect: Nonclinical in Vitro and in Silico Assessments. Hassan, S.T.S. Biomedicines, 2020. 8(5): e132. PMID[32456343].
[PubMed]. TB_05_2020.
11. A Preclinical Candidate Targeting Mycobacterium tuberculosis Kasa. Inoyama, D., D. Awasthi, G.C. Capodagli, K. Tsotetsi, P. Sukheja, M. Zimmerman, S.G. Li, R. Jadhav, R. Russo, X. Wang, C. Grady, T. Richmann, R. Shrestha, L. Li, Y.M. Ahn, H.P. Ho Liang, M. Mina, S. Park, D.S. Perlin, N. Connell, V. Dartois, D. Alland, M.B. Neiditch, P. Kumar, and J.S. Freundlich. Cell Chemical Biology, 2020. 27(5): p. 560-570. PMID[32197094]. PMCID[PMC7245553].
[PubMed]. TB_05_2020.
12. Synthesis of 2-Methoxy-3-(thiophen-2-ylmethyl)quinoline Containing Amino Carbinols as Antitubercular Agents. Karkara, B.B., S.S. Mishra, B.N. Singh, and G. Panda. Bioorganic Chemistry, 2020. 99: e103775. PMID[32222618].
[PubMed]. TB_05_2020.
13. Design, Synthesis, Evaluation, and Molecular Dynamic Simulation of Triclosan Mimic Diphenyl ether Derivatives as Antitubercular and Antibacterial Agents. Khade, A.B., H.I.M. Boshoff, K. Arora, K.E. Vandana, R. Verma, and G.G. Shenoy. Structural Chemistry, 2020. 31(3): p. 983-998. ISI[000529701400013].
[WOS]. TB_05_2020.
14. N-Alkyl-2-[4-(trifluoromethyl)benzoyl]hydrazine-1-carboxamides and their Analogues: Synthesis and Multitarget Biological Activity. Krátký, M., Z. Baranyai, Š. Štěpánková, K. Svrčková, M. Švarcová, J. Stolaříková, L. Horváth, S. Bősze, and J. Vinšová. Molecules, 2020. 25(10): e2268. PMID[32408517].
[PubMed]. TB_05_2020.
15. Synthesis, Characterization and Biological Potency of Butyl-pyridone Based Azo Dyes. Kumar, V., J. Keshavayya, M.N. Matada, S.M. Srinivasa, and S. Rangappa. ChemistrySelect, 2020. 5(18): p. 5460-5464. ISI[000532796500012].
[WOS]. TB_05_2020.
16. Identification of Benzothiazones Containing a Hexahydropyrrolo[3,4-c]pyrrol Moiety as Antitubercular Agents against MDR-Mtb. Ma, X.C., B. Han, A.Y. Wang, L. Yang, M.H. Huang, K. Chowdhury, J. Gu, K. Zhang, and K. Lv. RSC Advances, 2020. 10(24): p. 14410-14414. ISI[000528043700059].
[WOS]. TB_05_2020.
17. Synthesis and Antituberculosis Activity of New Acylthiosemicarbazides Designed by Structural Modification. Martínez, R., C.I. Espitia-Pinzón, M. Silva Miranda, R.M. Chávez-Santos, G. Pretelin-Castillo, A. Ramos-Orea, M. Hernández-Báez Á, S. Cotlame-Pérez, and R. Pedraza-Rodríguez. Drug Development Research, 2020. 81(3): p. 350-355. PMID[31777976].
[PubMed]. TB_05_2020.
18. Synthesis of 6-[4-(4-Propoxyphenyl)piperazin-1-yl]-9H-purine Derivatives as Antimycobacterial and Antifungal Agents: In Vitro Evaluation and in Silico Study. Nadaf, A.Q.A., M.S. Najare, M. Garbhagudi, S. Mantur, M.G. Sunagar, S. Gaonkar, S. Joshi, and I.A.M. Khazi. Chemistry and Biodiversity, 2020. 17(5): e2000053. PMID[32170847].
[PubMed]. TB_05_2020.
19. 5-Alkylthiomethyl Derivatives of 2'-Deoxyuridine: Synthesis and Antibacterial Activity. Negrya, S.D., D.A. Makarov, P.N. Solyev, I.L. Karpenko, O.V. Chekhov, A.A. Glukhova, B.F. Vasilyeva, I.G. Sumarukova, O.V. Efremenkova, S.N. Kochetkov, and L.A. Alexandrova. Russian Journal of Bioorganic Chemistry, 2020. 46(2): p. 133-138. ISI[000529094300002].
[WOS]. TB_05_2020.
20. Design, Synthesis and Antitubercular Activity of Novel Isoniazid-cyclic-amine-azachalcones Hybrids. Oliveira, J.R.S., C.Y.K. Shiguemoto, A.K. das Neves, F.M.F. Moreira, G.B. Gomes, R.T. Perdomo, S.L. Barbosa, P.G. Guerrero, J. Crodabl, and A.C.M. Baroni. Journal of the Brazilian Chemical Society, 2020. 31(6): p. 1284-1295. ISI[000530689400018].
[WOS]. TB_05_2020.
21. Inhibitory Activity of Traditional Plants against Mycobacterium smegmatis and their Action on Filamenting Temperature Sensitive Mutant Z (FtsZ)-a Cell Division Protein. Ravindran, R., G. Chakrapani, K. Mitra, and M. Doble. Plos One, 2020. 15(5): e0232482. PMID[32357366]. PMCID[PMC7195194].
[PubMed]. TB_05_2020.
22. Fragment-based Design of Mycobacterium tuberculosis InhA Inhibitors. Sabbah, M., V. Mendes, R.G. Vistal, D.M.G. Dias, M. Záhorszká, K. Mikušová, J. Korduláková, A.G. Coyne, T.L. Blundell, and C. Abell. Journal of Medicinal Chemistry, 2020. 63(9): p. 4749-4761. PMID[32240584]. PMCID[PMC7232676].
[PubMed]. TB_05_2020.
23. Synthesis of Functionalised Chromonyl-pyrimidines and their Potential as Antimycobacterial Agents. Santoso, K.T., M.W. Brett, C.Y. Cheung, G.M. Cook, B.L. Stocker, and M.S.M. Timmer. ChemistrySelect, 2020. 5(14): p. 4347-4355. ISI[000529295500032].
[WOS]. TB_05_2020.
24. Seeking Potent Anti-tubercular Agents: Design and Synthesis of Substituted-N-(6-(4-(pyrazine-2-carbonyl)piperazine/homopiperazine-1-yl)pyridin-3-yl)benzamide Derivatives as Anti-tubercular Agents. Srinivasarao, S., A. Nandikolla, A. Suresh, K. Van Calster, L. De Voogt, D. Cappoen, B. Ghosh, H. Aggarwal, S. Murugesan, and K. Sekhar. RSC Advances, 2020. 10(21): p. 12272-12288. ISI[000526839700017].
[WOS]. TB_05_2020.
25. Cytotoxicity and Antimycobacterial Properties of Pyrrolo[1,2-a]auinoline Derivatives: Molecular Target Identification and Molecular Docking Studies. Venugopala, K.N., V. Uppar, S. Chandrashekharappa, H.H. Abdallah, M. Pillay, P.K. Deb, M.A. Morsy, B.E. Aldhubiab, M. Attimarad, A.B. Nair, N. Sreeharsha, C. Tratrat, A. Yousef Jaber, R. Venugopala, R.P. Mailavaram, B.A. Al-Jaidi, M. Kandeel, M. Haroun, and B. Padmashali. Antibiotics, 2020. 9(5): e233. PMID[32392709].
[PubMed]. TB_05_2020.
26. Production of Antitubercular Depsipeptides via Biosynthetic Engineering of Cinnamoyl Units. Yang, Z., C. Sun, Z. Liu, Q. Liu, T. Zhang, J. Ju, and J. Ma. Journal of Natural Products, 2020. 83(5): p. 1666-1673. PMID[32338895].
[PubMed]. TB_05_2020.
27. Synergistic Activity of Nitroimidazole-Oxazolidinone Conjugates against Anaerobic Bacteria. Zhuang, Z., D. Wan, J. Ding, S. He, Q. Zhang, X. Wang, Y. Yuan, Y. Lu, C.Z. Ding, A.S. Lynch, A.M. Upton, C.B. Cooper, W.A. Denny, and Z. Ma. Molecules, 2020. 25(10): e2431. PMID[32456032].
[PubMed]. TB_05_2020.
Patent Citations
28. Pyrazinoic acid Conjugates and Hybrid Conjugates. Panda, S. Patent. 2020. 2019-16674651 20200140397: 65pp.
[Patent]. TB_05_2020.
29. Mmpl3 Inhibitors, Compositions and Uses Thereof. Rao, Z., J. Li, B. Zhang, and H. Yang. Patent. 2020. 2019-CN119668 2020103856: 128pp.
[Patent]. TB_05_2020.