Literature Citations
1. Exploring the Enzymatic and Antibacterial Activities of Novel Mycobacteriophage Lysin B Enzymes. Abouhmad, A., A.H. Korany, C. Grey, T. Dishisha, and R. Hatti-Kaul. International Journal of Molecular Sciences, 2020. 21(9): 3176. PMID[32365915]. PMCID[PMC7246905].
[PubMed]. TB_06_2020.
2. 3-(5-Nitrofuran-2-yl)prop-2-en-1-one Derivatives, with Potent Antituberculosis Activity, Inhibit a Novel Therapeutic Target, Arylamine N-Acetyltransferase, in Mycobacteria. Agre, N., N. Tawari, A. Maitra, A. Gupta, T. Munshi, M. Degani, and S. Bhakta. Antibiotics, 2020. 9(7): E368. PMID[32630175].
[PubMed]. TB_06_2020.
3. Exploring How Structural Changes to New Licarin a Derivatives Effects Their Bioactive Properties against Rapid Growing Mycobacteria and Biofilm Formation. Alvarenga, D.J., L.M.F. Matias, L.M. Oliveira, L. Leão, J.A. Hawkes, B.V.B. Raimundo, L.F.D. Castro, M.M.A. Campos, F.D.S. Siqueira, T.D. Santos, and D.T. Carvalho. Microbial Pathogenesis, 2020. 144: 104203. PMID[32304794].
[PubMed]. TB_06_2020.
4. Antimycobacterial Activity of Milemarinol, a New Squalene-type Triterpene, and Other Isolate? Boeno, S.I.S., M.D. Passos, M. Felix, S.D. Calixto, R.C. Almir, L.F.B. Siqueira, M.F. Muzitano, R. Braz, and I.J.C. Vieira. Natural Product Communications, 2020. 15(5): 1934578X20925589. ISI[000534526100001].
[WOS]. TB_06_2020.
5. Hemolytic and Antimicrobial Activities of a Series of Cationic Amphiphilic Copolymers Comprised of Same Centered Comonomers with Thiazole Moieties and Polyethylene Glycol Derivatives. Cuervo-Rodríguez, R., A. Muñoz-Bonilla, F. López-Fabal, and M. Fernández-García. Polymers, 2020. 12(4): 972. PMID[32331281]. PMCID[PMC7240493].
[PubMed]. TB_06_2020.
6. TCR-Like Domain Antibody against Mycobacterium tuberculosis (Mtb) Heat Shock Protein Antigen Presented by HLA-A*11 and HLA-A*24. Dass, S.A., M.N. Norazmi, A. Acosta, M.E. Sarmiento, and G.J. Tye. International Journal of Biological Macromolecules, 2020. 155: p. 305-314. PMID[32240734].
[PubMed]. TB_06_2020.
7. Indole-fused Spirochromenes as Potential Anti-tubercular Agents: Design, Synthesis and in Vitro Evaluation. Dogamanti, A., P. Chiranjeevi, V.K. Aamate, S.K. Vagolu, D. Sriram, S. Balasubramanian, and M. Sarasija. Molecular Diversity, 2020: p. 1-12. PMID[32474889].
[PubMed]. TB_06_2020.
8. (E)-2-(2-Allylidenehydrazinyl)thiazole Derivatives: Design, Green Synthesis, in Silico and in Vitro Antimycobacterial and Radical Scavenging Studies. Hublikar, M., V. Kadu, J.K. Dublad, D. Raut, S. Shirame, P. Makam, and R. Bhosale. Archiv der Pharmazie, 2020. 353(7): e2000003. PMID[32372473].
[PubMed]. TB_06_2020.
9. Benzimidazoquinazolines as New Potent anti-TB Chemotypes: Design, Synthesis, and Biological Evaluation. Jadhavar, P.S., K.I. Patel, T.M. Dhameliya, N. Saha, M.D. Vaja, V.S. Krishna, D. Sriram, and A.K. Chakraborti. Bioorganic Chemistry, 2020. 99: 103774. PMID[32224336].
[PubMed]. TB_06_2020.
10. Design, Synthesis and Biological Activity of Novel Substituted 3-Benzoic Acid Derivatives as MtDHFR Inhibitors. Kronenberger, T., G.M. Ferreira, A.D.F. de Souza, S. da Silva Santos, A. Poso, J.A. Ribeiro, M.T. Tavares, F.R. Pavan, G.H.G. Trossini, M.V.B. Dias, and R. Parise-Filho. Bioorganic and Medicinal Chemistry, 2020. 28(15): 115600. PMID[32631571].
[PubMed]. TB_06_2020.
11. Pyrazole-coumarin and Pyrazole-quinoline Chalcones as Potential Antitubercular Agents. Kumar, G., V. Siva Krishna, D. Sriram, and S.M. Jachak. Archiv der Pharmazie, 2020: e2000077. PMID[32484273].
[PubMed]. TB_06_2020.
12. Discovery of an Isothiazolinone-containing Antitubercular Natural Product Levesquamide. Liang, L., B. Haltli, D.H. Marchbank, M. Fischer, C.W. Kirby, H. Correa, T.N. Clark, C.A. Gray, and R.G. Kerr. Journal of Organic Chemistry, 2020. 85(10): p. 6450-6462. PMID[32363877].
[PubMed]. TB_06_2020.
13. Synthesis and Evaluation of Heterocycle Structures as Potential Inhibitors of Mycobacterium tuberculosis UGM. Maaliki, C., J. Fu, S. Villaume, A. Viljoen, C. Raynaud, S. Hammoud, J. Thibonnet, L. Kremer, S.P. Vincent, and E. Thiery. Bioorganic and Medicinal Chemistry, 2020. 28(13): 115579. PMID[32546296].
[PubMed]. TB_06_2020.
14. Structural Modifications of 3-Triazeneindoles and their Increased Activity Against Mycobacterium tuberculosis. Majorov, K.B., B.V. Nikonenko, P.Y. Ivanov, L.N. Telegina, A.S. Apt, and V.S. Velezheva. Antibiotics, 2020. 9(6): E356. PMID[32599854].
[PubMed]. TB_06_2020.
15. Comparative Assessment of Antifungal and Antibacterial Activities of Crude Extracts of the King Tuber Culinary-medicinal Mushroom, Pleurotus tuber-Regium (Agaricomycetes) from Cameroon. Metsebing, B.P., R. Oba, D.C. Mossebo, T.Y. Fonkui, F.T. Tsigain, M.C.D. Fotsing, T.C. Mungoh, and D.N. Ndinteh. International Journal of Medicinal Mushrooms, 2020. 22(4): p. 359-366. PMID[32558500].
[PubMed]. TB_06_2020.
16. Acetylene Containing Cyclo(L-Tyr-L-Tyr)-analogs as Mechanism-based Inhibitors of CYP121A1 from Mycobacterium tuberculosis. Ortega Ugalde, S., K. Wallraven, A. Speer, W. Bitter, T.N. Grossmann, and J.N.M. Commandeur. Biochemical Pharmacology, 2020. 177: 113938. PMID[32224137].
[PubMed]. TB_06_2020.
17. Identification of Potential Mycolyltransferase Ag85C Inhibitors of Mycobacterium tuberculosis H37Rv via Virtual High Throughput Screening and Binding Free Energy Studies. Pant, R., A. Joshi, P. Maiti, M. Nand, V. Pande, and S. Chandra. Journal of Molecular Graphics and Modelling, 2020. 98: 107584. PMID[32200279].
[PubMed]. TB_06_2020.
18. Inhaled Tigecycline Is Effective against Mycobacterium abscessus in Vitro and in Vivo. Pearce, C., M.M. Ruth, L.J. Pennings, H.F.L. Wertheim, A. Walz, W. Hoefsloot, C. Ruesen, J. Muñoz Gutiérrez, M. Gonzalez-Juarrero, and J. van Ingen. Journal of Antimicrobial Chemotherapy, 2020. 75(7): p. 1889-1894. PMID[32294173].
[PubMed]. TB_06_2020.
19. The Synthesis and Antituberculosis Activity of 5-Alkynyl Uracil Derivatives. Platonova, Y.B., A.N. Volov, and L.G. Tomilova. Bioorganic and Medicinal Chemistry Letters, 2020. 30(16): p. 127351. PMID[32631549].
[PubMed]. TB_06_2020.
20. Structure-guided Optimization of Inhibitors of Acetyltransferase Eis from Mycobacterium tuberculosis. Punetha, A., H.X. Ngo, S.Y.L. Holbrook, K.D. Green, M.J. Willby, S.A. Bonnett, K. Krieger, E.K. Dennis, J.E. Posey, T. Parish, O.V. Tsodikov, and S. Garneau-Tsodikova. ACS Chemical Biology, 2020. 15(6): p. 1581-1594. PMID[32421305].
[PubMed]. TB_06_2020.
21. Brazilian Green Propolis: Chemical Composition of Essential Oil and their in Vitro Antioxidant, Antibacterial and Antiproliferative Activities. Quintino, R.L., A.C. Reis, C.C. Fernandes, C.H.G. Martins, A.C. Colli, A.E.M. Crotti, L.S. Squarisi, A.B. Ribeiro, D.C. Tavares, and M.L.D. Miranda. Brazilian Archives of Biology and Technology, 2020. 63: e20190408. ISI[000537050300001].
[WOS]. TB_06_2020.
22. Indole Chalcones: Design, Synthesis, in vitro and in Silico Evaluation against Mycobacterium tuberculosis. Ramesh, D., A. Joji, B.G. Vijayakumar, A. Sethumadhavan, M. Mani, and T. Kannan. European Journal of Medicinal Chemistry, 2020. 198: 112358. PMID[32361610].
[PubMed]. TB_06_2020.
23. Microwave-assisted Synthesis of Some Indole and Isoniazid Derivatives as Antitubercular Agents and Molecular Docking Study. Rathod, A.S., P.V. Reddy, and J.S. Biradar. Russian Journal of Organic Chemistry, 2020. 56(4): p. 662-670. ISI[000535785500015].
[WOS]. TB_06_2020.
24. Synthesis and Evaluation of Antimycobacterial and Antiplasmodial Activities of Hirsutellide A and Its Analogues. Sahile, H.A., M.S. Martínez-Martínez, M. Dillenberger, K. Becker, and P. Imming. ACS Omega, 2020. 5(24): p. 14451-14460. PMID[32596583]. PMCID[PMC7315603].
[PubMed]. TB_06_2020.
25. Potential Anti-tuberculosis Activity of the Extracts and their Active Components of Anogeissus leiocarpa (DC.) Guill. and Perr. With Special Emphasis on Polyphenols. Salih, E.Y.A., R. Julkunen-Tiitto, O. Luukkanen, M. Sipi, M.K.M. Fahmi, and P.J. Fyhrquist. Antibiotics, 2020. 9(7): E364. PMID[32610461].
[PubMed]. TB_06_2020.
26. Cis-2 and Trans-2-eisocenoic Fatty acids are Novel Inhibitors for Mycobacterium tuberculosis Protein Tyrosine Phosphatase A. Savalas, L.R.T., B.R.N. Furqon, D. Asnawati, J. Ardhuha, P. Sedijani, S. Hadisaputra, B.N.S. Ningsih, and J. Syahri. Acta Biochimica Polonica, 2020. 67(2): p. 219-223. PMID[32559055].
[PubMed]. TB_06_2020.
27. Fluopsin C: A Potential Candidate against the Deadly Drug-resistant Microbial Infections in Humans. Sharma, D. Future Microbiology, 2020. 15: p. 381-384. PMID[32242758].
[PubMed]. TB_06_2020.
28. Discovery of 1,2,3-Triazole Based Quinoxaline-1,4-di-N-oxide Derivatives as Potential Anti-tubercular Agents. Srinivasarao, S., A. Nandikolla, A. Suresh, A.K. Ewa, A. Głogowska, B. Ghosh, B.K. Kumar, S. Murugesan, S. Pulya, H. Aggarwal, and K. Sekhar. Bioorganic Chemistry, 2020. 100: 103955. PMID[32464405].
[PubMed]. TB_06_2020.
29. Improving the Potency of N-Aryl-2,5-dimethylpyrroles against Multidrug-resistant and Intracellular Mycobacteria. Touitou, M., F. Manetti, C.M. Ribeiro, F.R. Pavan, N. Scalacci, K. Zrebna, N. Begum, D. Semenya, A. Gupta, S. Bhakta, T.D. McHugh, H. Senderowitz, M. Kyriazi, and D. Castagnolo. ACS Medicinal Chemistry Letters, 2020. 11(5): p. 638-644. PMID[32435364]. PMCID[PMC7236041].
[PubMed]. TB_06_2020.
30. Identification of 2-((2,3-Dihydrobenzo[b][1,4]dioxin-6-yl)amino)-N-phenylpropanamides as a Novel Class of Potent DprE1 Inhibitors. Whitehurst, B.C., R.J. Young, G.A. Burley, M. Cacho, P. Torres, and L. Vela-Gonzalez Del Peral. Bioorganic and Medicinal Chemistry Letters, 2020. 30(12): 127192. PMID[32312582].
[PubMed]. TB_06_2020.
31. Identification of Anti-tuberculosis Compounds from Aurone Analogs. Yang, D., Z.E. Taylor, S. Handy, S. Li, J. Liu, J. Stabenow, L. Zalduondo, C.B. Jonsson, E. Altman, and Y. Kong. Frontiers in Microbiology, 2020. 11: p. 1004. PMID[32508798]. PMCID[PMC7251074].
[PubMed]. TB_06_2020.
Patent Citations
32. Antimicrobial Peptides. Birol, I., C.C. Helbing, and S.A. Hammond. Patent. 2020. 2019-CA51778 2020118427: 83pp.
[Patent]. TB_06_2020.
33. Discovery of BD Oxidase Inhibitors for the Treatment of Mycobacterial Diseases. Miller, M.J., G.C. Moraski, and K. Pethe. Patent. 2020. 2019-IB61142 2020128981: 122pp.
[Patent]. TB_06_2020.
34. Substituted 1,2,4-Oxadiazole, Its Application and a Pharmaceutical Preparation Comprising It. Roh, J., G. Karabanovich, P. Pavek, A. Hrabalek, and V. Klimesova. Patent. 2020. 2019-IB59934 2020128675: 29pp.
[Patent]. TB_06_2020.
35. Salicyl-adenosinemonosulfamate Analogs and Uses Thereof. Tan, D.S., L.C. Standke, L.E.N. Quadri, G.V. Bythrow, W.R. Bishai, and S. Lun. Patent. 2020. 2019-US68107 2020132603: 188pp.
[Patent]. TB_06_2020.