Literature Citations
1. A Stereo, Regioselective Synthesis and Discovery of Antimycobaterium Tuberculosis Activity of Novel beta-Lactam Grafted Spirooxindolopyrrolidine Hybrid Heterocycles. Arumugam, N., A.I. Almansour, R.S. Kumar, V.S. Krishna, D. Sriram, and R. Padmanaban. Arabian Journal of Chemistry, 2021. 14(102938); 10pp. ISI[000614263300025].
[WOS]. TB_03_2021.
2. Phytochemical Analysis and Evaluation of Antioxidant and Antimycobacterial Activity of Colletia paradoxa from Brazil. Bastos Záchia, N.R., M. Piana, F. Dos Santos Siqueira, R. da Silva Jesus, M.L. Athayde, L. Essi, and M.M.A. de Campos. Natural Product Research, 2021. 35(5): p. 802-806. PMID[30990070].
[PubMed]. TB_03_2021.
3. Carbonyl cyanide 3-chlorophenylhydrazone (CCCP) Exhibits Direct Antibacterial Activity against Mycobacterium abscessus. Chen, S., T. Teng, Z. Zhang, Y. Shang, H. Xiao, G. Jiang, F. Wang, J. Jia, L. Dong, L. Zhao, N. Chu, and H. Huang. Infection and Drug Resistance, 2021. 14: p. 1199-1208. PMID[33790590]. PMCID[PMC8001050].
[PubMed]. TB_03_2021.
4. Structure Based Design, Synthesis, and Biological Evaluation of Imidazole Derivatives Targeting Dihydropteroate Synthase Enzyme. Daraji, D.G., D.P. Rajani, S.D. Rajani, E.A. Pithawala, S. Jayanthi, and H.D. Patel. Bioorganic and Medicinal Chemistry Letters, 2021. 36: 127819. PMID[33513385].
[PubMed]. TB_03_2021.
5. Synthesis and Evaluation of Porphyrin Glycoconjugates Varying in Linker Length: Preliminary Effects on the Photodynamic Inactivation of Mycobacterium smegmatis. Dixon, C.F., A.N. Nottingham, A.F. Lozano, J.A. Sizemore, L.A. Russell, C. Valiton, K.L. Newell, D. Babin, W.T. Bridges, M.R. Parris, D.V. Shchirov, N.L. Snyder, and J.V. Ruppel. RSC Advances, 2021. 11(12): p. 7037-7042. ISI[000617371900058].
[WOS]. TB_03_2021.
6. Easily Accessed Nitroquinolones Exhibiting Potent and Selective Anti-tubercular Activity. Dube, P.S., L.J. Legoabe, A. Jordaan, O.J. Jesumoroti, T. Tshiwawa, D.F. Warner, and R.M. Beteck. European Journal of Medicinal Chemistry, 2021. 213: 113207. PMID[33524688].
[PubMed]. TB_03_2021.
7. A Coumarin-based Analogue of Thiacetazone as Dual Covalent Inhibitor and Potential Fluorescent Label of HADA in Mycobacterium tuberculosis. Farjallah, A., L.R. Chiarelli, M. Forbak, G. Degiacomi, M. Danel, F. Goncalves, C. Carayon, C. Seguin, M. Fumagalli, M. Záhorszká, E. Vega, S. Abid, A. Grzegorzewicz, M. Jackson, A. Peixoto, J. Korduláková, M.R. Pasca, C. Lherbet, and S. Chassaing. ACS Infectious Diseases, 2021. 7(3): p. 552-565. PMID[33617235]. PMCID[PMC8022203].
[PubMed]. TB_03_2021.
8. Identification of Inhibitors of UDP-galactopyranose Mutase via Combinatorial in Situ Screening. Fu, J., H. Fu, Y. Xia, I. N'Go, J. Cao, W. Pan, and S.P. Vincent. Organic and Biomolecular Chemistry, 2021. 19(8): p. 1818-1826. PMID[33565547].
[PubMed]. TB_03_2021.
9. Efficient Pyran Derivatives Synthesis in Des Medium and Their Antimicrobial Evaluation as Inhibitors of Mycobacterium bovis (BCG). Hakiminasab, S., A. Habibi, S.M. Shahcheragh, Y. Farahani, S. Sardari, H. Dolati, S.M. Mahdavi, and M. Habibi. Journal of the Iranian Chemical Society. ISI[000620102500001].
[WOS]. TB_03_2021.
10. Simultaneous Determination of a Novel Oxazolidinone Anti-tuberculosis OTB-658 and Its Metabolites in Monkey Blood by LC-MS/MS. Jiang, J., Y. Liu, X. Liu, D. Zhang, H. Huang, B. Wang, L. Sheng, and Y. Li. Journal of Chromatography. B, Analytical Technologies in the Biomedical and Life Sciences, 2021. 1167: 122552. PMID[33588346].
[PubMed]. TB_03_2021.
11. Toxin-activating Stapled Peptides Discovered by Structural Analysis Were Identified as New Therapeutic Candidates That Trigger Antibacterial Activity against Mycobacterium tuberculosis in the Mycobacterium smegmatis Model. Kang, S.M., H. Moon, S.W. Han, B.W. Kim, D.H. Kim, B.M. Kim, and B.J. Lee. Microorganisms, 2021. 9(3): 568. PMID[33801872].
[PubMed]. TB_03_2021.
12. Comparison of the Efficacy of Two Novel Antitubercular Agents in Free and Liposome-encapsulated Formulations. Kosa, N., A. Zolcsak, I. Voszka, G. Csik, K. Horvati, L. Horvath, S. Bosze, and L. Herenyi. International Journal of Molecular Sciences, 2021. 22(5): 2457. ISI[000628295900001].
[WOS]. TB_03_2021.
13. Computational Exploration and Anti-mycobacterial Activity of Potential Inhibitors of Mycobacterium tuberculosis Acetyl Coenzyme a Carboxylase as Anti-tubercular Agents. Kuldeep, J., S.K. Sharma, B.N. Singh, and M.I. Siddiqi. SAR and QSAR in Environmental Research, 2021. 32(3): p. 191-205. PMID[33612029].
[PubMed]. TB_03_2021.
14. Synthesis, Biological Evaluation and Molecular Docking Studies of Novel Quinazolinones as Antitubercular and Antimicrobial Agents. Kumar Pandey, S., U. Yadava, A. Upadhyay, and M.L. Sharma. Bioorganic Chemistry, 2021. 108: 104611. PMID[33484939].
[PubMed]. TB_03_2021.
15. Hydride-induced Meisenheimer Complex Formation Reflects Activity of Nitro Aromatic Anti-tuberculosis Compounds. Liu, R., L. Markley, P.A. Miller, S. Franzblau, G. Shetye, R. Ma, K. Savkova, K. Mikusova, B.S. Lee, K. Pethe, G.C. Moraski, and M.J. Miller. RSC Medicinal Chemistry, 2021. 12(1): p. 62-72. ISI[000614556400005].
[WOS]. TB_03_2021.
16. Concentration Dependent SERS, DFT and Molecular Docking Studies of a Ureido Derivative with Antitubercular Properties. Mary, Y.S., Y.S. Mary, M. Krátký, J. Vinsova, C. Baraldi, and M. Cristina Gamberini. Spectrochimica Acta. Part A, Molecular and Biomolecular Spectroscopy, 2021. 249: p. 119329. PMID[33360209].
[PubMed]. TB_03_2021.
17. Isolation and Antimicrobial Activities of Phytochemicals from Parinari curatellifolia (Chrysobalanaceae). Mawire, P., W. Mozirandi, M. Heydenreich, G.F. Chi, and S. Mukanganyama. Advances in Pharmacological and Pharmaceutical Sciences, 2021. 2021: 8842629 . PMID[33763648]. PMCID[PMC7952164].
[PubMed]. TB_03_2021.
18. Synthesis, Characterization, and Biological Evaluation of New Derivatives Targeting MbtI as Antitubercular Agents. Mori, M., G. Stelitano, L.R. Chiarelli, G. Cazzaniga, A. Gelain, D. Barlocco, E. Pini, F. Meneghetti, and S. Villa. Pharmaceuticals, 2021. 14(2): 155. PMID[33668554]. PMCID[PMC7918538].
[PubMed]. TB_03_2021.
19. Allyl Piperidine-1-carbodiothioate and Benzyl 1H-imidazole 1 Carbodithioate: Two Potential Agents to Combat against Mycobacteria. Mukherjee, G., K. Mukherjee, R. Das, R.S. Mandal, I. Roy, B. Mukhopadhyay, and A.K. Sil. Journal of Applied Microbiology, 2021. 130(3): p. 786-796. PMID[32615006].
[PubMed]. TB_03_2021.
20. Stereochemical Aspects in the Synthesis of Novel N-(Purin-6-yl)dipeptides as Potential Antimycobacterial Agents. Musiyak, V.V., I.A. Nizova, E.N. Chulakov, L.S. Sadretdinova, A.A. Tumashov, G.L. Levit, and V.P. Krasnov. Amino Acids, 2021. 53(3): p. 407-415. PMID[33599833]. PMCID[PMC7889712].
[PubMed]. TB_03_2021.
21. Synthesis, Characterization and Docking Studies of N-Methyl-2,3-dihydro quinazolin-4-ones Linked 1,3-Thiazole Hybrids as Potent Anti-tubercular Agents. Nagaladinne, N., A.A. Hindustan, and D. Nayakanti. Indian Journal of Pharmaceutical Sciences, 2020. 82(6): p. 984-995. ISI[000620813100007].
[WOS]. TB_03_2021.
22. Molecular Characterization and Antimicrobial Resistance Profiles of Mycobacterium tuberculosis Complex in Environmental Substrates from Three Dairy Farms in Eastern Cape, South Africa. Ntloko, A., M.A. Adefisoye, and E. Green. International Journal of Environmental Health Research, 2021. 31(2): p. 215-224. PMID[31305130].
[PubMed]. TB_03_2021.
23. Identification of Potent Antigen 85C Inhibitors of Mycobacterium tuberculosis via in-House Lichen Library and Binding Free Energy Studies Part-II. Pant, R., A. Joshi, T. Joshi, P. Maiti, M. Nand, T. Joshi, V. Pande, and S. Chandra. Journal of Molecular Graphics and Modelling, 2021. 103: 107822. PMID[33333421].
[PubMed]. TB_03_2021.
24. The Benzimidazole SPR719 Shows Promising Concentration-dependent Activity and Synergy against Nontuberculous Mycobacteria. Pennings, L.J., M.M. Ruth, H.F.L. Wertheim, and J. van Ingen. Antimicrobial Agents and Chemotherapy, 2021. 65(4): e02469-20. PMID[33468478].
[PubMed]. TB_03_2021.
25. Biofilm Degradation of Nontuberculous Mycobacteria Formed on Stainless Steel Following Treatment with Immortelle (Helichrysum italicum) and Common Juniper (Juniperus communis) Essential Oils. Peruc, D., D. Broznic, Z. Maglica, Z. Marijanovic, L. Karleusa, and I. Gobin. Processes, 2021. 9(2): 362. ISI[000623209300001].
[WOS]. TB_03_2021.
26. Covalent Inactivation of Mycobacterium tuberculosis Isocitrate Lyase by cis-2,3-Epoxy-succinic acid. Pham, T.V., D.M. Mellott, Z. Moghadamchargari, K. Chen, I. Krieger, A. Laganowsky, J.C. Sacchettini, and T.D. Meek. ACS Chemical Biology, 2021. 16(3): p. 463-470. PMID[33688722].
[PubMed]. TB_03_2021.
27. Search for Antimicrobial Activity among Fifty-two Natural and Synthetic Compounds Identifies Anthraquinone and Polyacetylene Classes That Inhibit Mycobacterium tuberculosis. Pollo, L.A.E., E.F. Martin, V.R. Machado, D. Cantillon, L.M. Wildner, M.L. Bazzo, S.J. Waddell, M.W. Biavatti, and L.P. Sandjo. Frontiers in Microbiology, 2020. 11: 622629. PMID[33537021]. PMCID[PMC7847937].
[PubMed]. TB_03_2021
28. Click Synthesis of 1,2,3-Triazole Based Imidazoles: Antitubercular Evaluation, Molecular Docking and HSA Binding Studies. Pradeep Kumar, C.B., B.S. Prathibha, K.N.N. Prasad, M.S. Raghu, M.K. Prashanth, B.K. Jayanna, F.A. Alharthi, S. Chandrasekhar, H.D. Revanasiddappa, and K. Yogesh Kumar. Bioorganic and Medicinal Chemistry Letters, 2021. 36: 127810. PMID[33482292].
[PubMed]. TB_03_2021.
29. Antimicrobial Activity of Pyrazinamide Coordination Frameworks Synthesized by Mechanochemistry. Quaresma, S., P.C. Alves, P. Rijo, M.T. Duarte, and V. André. Molecules, 2021. 26(7): 1904. PMID[33800635]. PMCID[PMC8036749].
[PubMed]. TB_03_2021.
30. Antimicrobial and Antitumor Activity of S-methyl Dithiocarbazate Schiff Base Zinc(II) Complexes. Ramilo-Gomes, F., Y. Addis, I. Tekamo, I. Cavaco, D.L. Campos, F.R. Pavan, C.S.B. Gomes, V. Brito, A.O. Santos, F. Domingues, Â. Luís, M.M. Marques, J.C. Pessoa, S. Ferreira, S. Silvestre, and I. Correia. Journal of Inorganic Biochemistry, 2021. 216: 111331. PMID[33348167].
[PubMed]. TB_03_2021.
31. A Broad Spectrum Anti-bacterial Peptide with an Adjunct Potential for Tuberculosis Chemotherapy. Rao, K.U., D.I. Henderson, N. Krishnan, M. Puthia, I. Glegola-Madejska, L. Brive, F. Bjarnemark, A. Millqvist Fureby, K. Hjort, D.I. Andersson, E. Tenland, E. Sturegard, B.D. Robertson, and G. Godaly. Scientific Reports, 2021. 11(1): 4201. PMID[33603037]. PMCID[PMC7892554].
[PubMed]. TB_03_2021.
32. Synthesis of Novel Quinoxaline-alkynyl Derivatives and Their Anti-mycobacterium tuberculosis Activity. Raphoko, L.A., K. Lekgau, C.M. Lebepe, T.C. Leboho, T.M. Matsebatlela, and W. Nxumalo. Bioorganic and Medicinal Chemistry Letters, 2021. 35: 127784. PMID[33422606].
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33. Synthesis of Some Novel Piperidine Fused 5-Thioxo-1H-1,2,4-triazoles as Potential Antimicrobial and Antitubercular Agents. Rishikesan, R., R.P. Karuvalam, N.J. Muthipeedika, A.M. Sajith, K.R. Eeda, R. Pakkath, K.R. Haridas, V. Bhaskar, K.H. Narasimhamurthy, and A. Muralidharan. Journal of Chemical Sciences, 2021. 133(1): 3 (2021). ISI[000617327600001].
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34. Discovery of Novel Antituberculosis Agents among 3-Phenyl-5-(1-phenyl-1H-[1,2,3]triazol-4-yl)-[1,2,4]oxadiazole Derivatives Targeting Aminoacyl-tRNA Synthetases. Rybak, M.Y., A.O. Balanda, A.P. Yatsyshyna, I.M. Kotey, S.A. Starosyla, V.G. Bdzhola, L.L. Lukash, S.M. Yarmoluk, M.A. Tukalo, and G.P. Volynets. Scientific Reports, 2021. 11(7162): 10pp. PMID[33785838]. PMCID[PMC8010095].
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35.Inhibition of Biofilm Formation by the Synergistic Action of EGCG-S and Antibiotics. Shinde, S., L.H. Lee, and T. Chu. Antibiotics, 2021. 10(2): 102. PMID[33494273]. PMCID[PMC7909832].
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36. Structure Based Identification of First-in-class Fragment Inhibitors That Target the NMN Pocket of M. tuberculosis NAD(+)-dependent DNA Ligase A. Shukla, A., M. Afsar, N. Kumar, S. Kumar, and R. Ramachandran. Journal of Structural Biology, 2021. 213(1): 107655. PMID[33197566].
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37. Experimental and Computational Studies of an Antiplasmodial Derivative of Allantoin; Antimycobacterial Essential Oil from Cordia batesii WERNHAM (Boraginaceae). Tiam, E.R., D.S.N. Bikobo, I.M. Ndassa, N.M. Nyemeck Ii, A.Z. AA, L. Ayong, P.H.B. Diboué, B.L. Ndjakou, J.N. Mbing, and D.E. Pegnyemb. BMC Chemistry, 2021. 15(15): 17pp. PMID[33673871]. PMCID[PMC7934435].
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38. Synthesis, Structural Elucidation, Pharmacological and Molecular Docking Studies of Terpolymer Transition Metal Complexes. Vijayan, N., R. Princess, S.J. Raja, and J. Joseph. Journal of Molecular Structure, 2021. 1227: 129424. ISI[000609155200022].
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39. Engineering Selectivity for Reduced Toxicity of Bacterial Kinase Inhibitors Using Structure-guided Medicinal Chemistry. Wlodarchak, N., J.B. Feltenberger, Z.Q. Ye, J. Beczkiewicz, R. Procknow, G. Yan, T.M. King, J.E. Golden, and R. Striker. ACS Medicinal Chemistry Letters, 2021. 12(2): p. 228-235. ISI[000619767800006].
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40. Identification of Novel Tricyclic Benzo[1,3]oxazinyloxazolidinones as Potent Antibacterial Agents with Excellent Pharmacokinetic Profiles against Drug-resistant Pathogens. Wu, Y., B. Wang, H. Lu, H. Zhao, B. Yang, L. Li, Y. Lu, D. Zhang, N. Sun, and H. Huang. Journal of Medicinal Chemistry, 2021. 64(6): p. 3234-3248. PMID[33705128].
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41. Design and Synthesis of Mycobacterial pks13 Inhibitors: Conformationally Rigid Tetracyclic Molecules. Zhang, W., L.L. Liu, S. Lun, S.S. Wang, S. Xiao, H. Gunosewoyo, F. Yang, J. Tang, W.R. Bishai, and L.F. Yu. European Journal of Medicinal Chemistry, 2021. 213: 113202. PMID[33516983].
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Patent Citations
42. Preparation of Benzyl Amine-containing 5,6-Heteroaromatic Compounds Useful against Mycobacterial Infection. Fujitani, M., T. Iwaki, R. Nakamura, M.J. Miller, and G.C. Moraski. Patent. 2021. 2020-US50173 2021050708: 124pp.
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43. Heterocyclic Compounds as Antibacterial Agents and Their Preparation. Guillemont, J.E.G., M.M.S. Motte, M.C. Villellas Arilla, G.M.J. Lammens, A.J.D.M. Rene, M.L. Jeanty, and D.A. Lamprecht. Patent. 2021. 2020-EP75458 2021048342: 228pp.
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44. Indole Carboxamide Compounds and Use Thereof for the Treatment of Mycobacterial Infections. Kaneko, T. and N. Fotouhi. Patent. 2021. 2020-US52938 2021062319: 88pp.
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45. Thiazole Carboxamide Compounds and Use Thereof for the Treatment of Mycobacterial Infections. Kaneko, T. and N. Fotouhi. Patent. 2021. 2020-US52937 2021062318: 157pp.
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46. Azaindole Carboxamide Compounds for the Treatment of Mycobacterial Infections. Kaneko, T. and N. Fotouhi. Patent. 2021. 2020-US52934 2021062316: 394pp.
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