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HIV Drugs in Development


Drug ClassCompanyDrug NameAlt NameDrug StatusNotesAIDS#
Biological Response Modifier Hemispherx; Rega Institute For Medical ResearchAtvogen™Ampligen, AMP, Poly(I)-Poly(C12U)Phase IICompleted 000136
Entry Inhibitor Tobira TherapeuticsCenicrivirocTBR-652; TAK-652Phase IIRecruiting 224423
Entry Inhibitor Tanox; Biogen Idec; Taimed BiologiesIbalizumabTNX-355; Hu5A8Phase IIInvitation Only 209859
Entry Inhibitor Progenics PharmaceuticalsPRO-140 Phase IIOngoing 088103
Entry Inhibitor Incyte CorporationINCB-009471INCB-9471Phase IICompleted 503495
Entry and Fusion InhibitorsSchering-PloughVicrivirocSCH-417690, SCH-D, VCVPhase IIDrug Development Halted as of July 15, 2010 due to poor performance 210504
Entry and Fusion InhibitorsGenzyme CorporationAMD-070AMD-11070Phase I/IICompleted 495149
Fusion Inhibitor Cellegy PharmaceuticalsCyanovirin-N CV-N, CV-N Protein, Cianovirina-NPreclinical  045707
Fusion Inhibitor PfizerPF-00232798 Phase IICompleted
HDAC InhibitorAbbott LabsDepakote™Valporic acid, Divalproex sodium, VPAPhase IibRecruitment Unknown 057177
Integrase Inhibitor GlaxoSmithKlineGSK1349572 Phase IIIRecruiting
Integrase Inhibitor Japan Tobacco Inc.; Gilead Sciences; GlaxoSmithKlineElvitegravirEVG, GS-9137, JTK-303Phase IIIOngoing 241767
Integrase Inhibitor GlaxoSmithKlineGSK1265744 Phase IIaCompleted
MicrobicideGilead SciencesTenofovir gel (GS-1275)GS-1275; PMPA gelPhase IICompleted 021800
MicrobicidePanacos PharmaceuticalsBevirimatBVM, PA-457; MPC-4326Phase IICompleted 028530
MicrobicideUniroyal/Crompton Corp/BiosynUC781 Phase ICompleted 029940
MicrobicideStarpharmaVivaGel™SPL-7013 gelPhase II Ongoing 223863
MicrobicideReprotect, Inc.BufferGel™Carbomer 974P, Carbopol 974P, Carbopol polymerPhase IICompleted 180064
MicrobicideProcept/Interneuron/IndevusPro-2000PRO-2000/5Phase IIICompleted 032942
MicrobicidePopulation Council Center for Biomedical ResearchCarraguard™Carragaen, Carrageenan gum, Carrageenin, Irish moss extract, PC-515Phase ICompleted 000100
NNRTIGlaxoSmithKlineGSK2248761IDX-899Phase IIOn Hold
NNRTIJanssen Pharmaceutica N.V.; TibotecRilpivirineR278474, TMC-278Phase IIIOngoing 169030
NNRTIPfizerLersivirineUK453,061Phase IIOngoing 497274
NNRTIBoehringer IngelheimBILR 355 BS Phase IIStudy Terminated 212773
NRTIAchillion PharmaceuticalsElvucitabineACH-126443Phase IIOngoing 060327
NRTIPharmasset/Dupont Pharmaceuticals; VionReverset™Dexelvucitabine; DFCPhase IIStudy Terminated 000572
NRTIGlaxo Wellcome; GlaxoSmithKline; Pharmasset, Inc.RacivirRCV; (+/-)FTCPhase IICompleted 005245
NRTIBiochem Pharma; Triangle Pharmaceuticals; Gilead SciencesAmdoxovirDAPDPhase IICompleted 005431
Other Immune ModulatorGlaxoSmithKlineTucaresol Phase IICompleted 029800
Other Immune ModulatorCytodyn, Inc.Cytolin™ Phase IIOngoing

Last Updated: December 2011